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SHAHUL HAMEED, P, SOLAPURE, Suresh, GHOSH, Anirban, AWASTHY, Disha, SHANBHAG, Gajanan, SHEIKH, Gulebahar, MCMIKEN, Helen, PUTTUR, Jayashree, REDDY, Jitendar, WERNGREN, Jim, READ, Jon, KUMAR, Mahesh, MUKHERJEE, Kakoli, MANJUNATHA, R, CHINNAPATTU, Murugan, MADHAVAPEDDI, Prashanti, MANJREKAR, Praveena, BASU, Reetobrata, GAONKAR, Sheshagiri, SHARMA, Sreevalli, HOFFNER, Sven, HUMNABADKAR, Vaishali, SUBBULAKSHMI, Venkita, NANDI, Vrinda, PANDUGA, Vijender, WATERSON, David, SHANDIL, Radha, BALGANESH, Meenakshi, SAMBANDAMURTHY, Vasan K, ANAND KUMAR RAICHURKAR, DESHPANDE, Abhijeet
Published in Antimicrobial Agents and Chemotherapy (01.01.2014)
Published in Antimicrobial Agents and Chemotherapy (01.01.2014)
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KISHORE REDDY, B. K, LANDGE, Sudhir, AMBADY, Anisha, GHOSH, Anirban, TUNDUGURU, Ragadeepthi, KAUR, Parvinder, SINGH, Ragini, KUMAR, Naveen, BHARATH, Sowmya, SUNDARAM, Aishwarya, BHAT, Jyothi, SAMBANDAMURTHY, Vasan K, RAVISHANKAR, Sudha, BJÖRKELID, Christofer, ALWYN JONES, T, DAS, Kaveri, BANDODKAR, Balachandra, MALOLANARASIMHAN, Krishnan, MUKHERJEE, Kakoli, RAMACHANDRAN, Vasanthi, PATIL, Vikas, SHINDE, Vikas, TANTRY, Subramanyam, KALE, Manoj, RAICHURKAR, Anandkumar, MENASINAKAI, Sreenivasaiah, NAINA VINAY MUDUGAL
Published in Antimicrobial agents and chemotherapy (01.06.2014)
Published in Antimicrobial agents and chemotherapy (01.06.2014)
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Essentiality and functional analysis of type I and type III pantothenate kinases of Mycobacterium tuberculosis
AWASTHY, Disha, AMBADY, Anisha, BHAT, Jyothi, SHEIKH, Gulebahar, RAVISHANKAR, Sudha, SUBBULAKSHMI, Venkita, MUKHERJEE, Kakoli, SAMBANDAMURTHY, Vasan, SHARMA, Umender
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Published in Microbiology (Society for General Microbiology) (01.09.2010)
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Peptide Deformylase Inhibitors as Potent Antimycobacterial Agents
TEO, Jeanette W. P, THAYALAN, Pamela, HASAN, Samiul, CYNAMON, Michael, RYDER, Neil S, XIA YANG, WEIDMANN, Beat, BRACKEN, Kathryn, DICK, Thomas, MUKHERJEE, Kakoli, BEER, David, YAP, Amelia S. L, NANJUNDAPPA, Mahesh, NGEW, Xinyi, DURAISWAMY, Jeyaraj, LIUNG, Sarah, DARTOIS, Veronique, SCHREIBER, Mark
Published in Antimicrobial Agents and Chemotherapy (01.11.2006)
Published in Antimicrobial Agents and Chemotherapy (01.11.2006)
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Proteins released during high toxin production in Clostridium difficile
Mukherjee, Kakoli, Karlsson, Sture, Burman, Lars G, Akerlund, Thomas
Published in Microbiology (Society for General Microbiology) (01.07.2002)
Published in Microbiology (Society for General Microbiology) (01.07.2002)
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Discovery of Imidazo[1,2‑a]pyridine Ethers and Squaramides as Selective and Potent Inhibitors of Mycobacterial Adenosine Triphosphate (ATP) Synthesis
Tantry, Subramanyam J, Markad, Shankar D, Shinde, Vikas, Bhat, Jyothi, Balakrishnan, Gayathri, Gupta, Amit K, Ambady, Anisha, Raichurkar, Anandkumar, Kedari, Chaitanyakumar, Sharma, Sreevalli, Mudugal, Naina V, Narayan, Ashwini, Naveen Kumar, C. N, Nanduri, Robert, Bharath, Sowmya, Reddy, Jitendar, Panduga, Vijender, Prabhakar, K. R, Kandaswamy, Karthikeyan, Saralaya, Ramanatha, Kaur, Parvinder, Dinesh, Neela, Guptha, Supreeth, Rich, Kirsty, Murray, David, Plant, Helen, Preston, Marian, Ashton, Helen, Plant, Darren, Walsh, Jarrod, Alcock, Peter, Naylor, Kathryn, Collier, Matthew, Whiteaker, James, McLaughlin, Robert E, Mallya, Meenakshi, Panda, Manoranjan, Rudrapatna, Suresh, Ramachandran, Vasanthi, Shandil, Radha, Sambandamurthy, Vasan K, Mdluli, Khisi, Cooper, Christopher B, Rubin, Harvey, Yano, Takahiro, Iyer, Pravin, Narayanan, Shridhar, Kavanagh, Stefan, Mukherjee, Kakoli, Balasubramanian, V, Hosagrahara, Vinayak P, Solapure, Suresh, Ravishankar, Sudha, Hameed P, Shahul
Published in Journal of medicinal chemistry (23.02.2017)
Published in Journal of medicinal chemistry (23.02.2017)
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Discovery of MDV6058 (PF-06952229), a selective and potent TGF?R1 inhibitor: Design, synthesis and optimization
Pujala, Brahmam, Ramachandran, Sreekanth A., Sonawane, Mukesh, Kamble, Maruti M., Panpatil, Dayanand, Adhikari, Swati, Soni, Sanjeev, Subbareddy, Venkata, Shinde, Bharat U., Nayak, Anjan K., Bansal, Chandni, Gupta, Ashu, Mukherjee, Kakoli, Agarwal, Anil K., Guerrero, Javier, Herrera, Francisco J., Bernales, Sebastian, Guha, Mausumee, Chakravarty, Sarvajit, Pham, Son M., Rai, Roopa
Published in Bioorganic & medicinal chemistry letters (01.11.2022)
Published in Bioorganic & medicinal chemistry letters (01.11.2022)
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Structural and Biochemical Characterization of Compounds Inhibiting Mycobacterium tuberculosis Pantothenate Kinase
Björkelid, Christofer, Bergfors, Terese, Raichurkar, Anand Kumar V., Mukherjee, Kakoli, Malolanarasimhan, Krishnan, Bandodkar, Balachandra, Jones, T. Alwyn
Published in The Journal of biological chemistry (21.06.2013)
Published in The Journal of biological chemistry (21.06.2013)
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Discovery of MDV6058 (PF-06952229), a selective and potent TGFβR1 inhibitor: Design, synthesis and optimization
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Published in Bioorganic & medicinal chemistry letters (01.11.2022)
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Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate
Hameed P., Shahul, Solapure, Suresh, Patil, Vikas, Henrich, Philipp P., Magistrado, Pamela A., Bharath, Sowmya, Murugan, Kannan, Viswanath, Pavithra, Puttur, Jayashree, Srivastava, Abhishek, Bellale, Eknath, Panduga, Vijender, Shanbag, Gajanan, Awasthy, Disha, Landge, Sudhir, Morayya, Sapna, Koushik, Krishna, Saralaya, Ramanatha, Raichurkar, Anandkumar, Rautela, Nikhil, Roy Choudhury, Nilanjana, Ambady, Anisha, Nandishaiah, Radha, Reddy, Jitendar, Prabhakar, K. R., Menasinakai, Sreenivasaiah, Rudrapatna, Suresh, Chatterji, Monalisa, Jiménez-Díaz, María Belén, Martínez, María Santos, Sanz, Laura María, Coburn-Flynn, Olivia, Fidock, David A., Lukens, Amanda K., Wirth, Dyann F., Bandodkar, Balachandra, Mukherjee, Kakoli, McLaughlin, Robert E., Waterson, David, Rosenbrier-Ribeiro, Lyn, Hickling, Kevin, Balasubramanian, V., Warner, Peter, Hosagrahara, Vinayak, Dudley, Adam, Iyer, Pravin S., Narayanan, Shridhar, Kavanagh, Stefan, Sambandamurthy, Vasan K.
Published in Nature communications (31.03.2015)
Published in Nature communications (31.03.2015)
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Design, synthesis and optimization of bis-amide derivatives as CSF1R inhibitors
Ramachandran, Sreekanth A., Jadhavar, Pradeep S., Miglani, Sandeep K., Singh, Manvendra P., Kalane, Deepak P., Agarwal, Anil K., Sathe, Balaji D., Mukherjee, Kakoli, Gupta, Ashu, Haldar, Srijan, Raja, Mohd, Singh, Siddhartha, Pham, Son M., Chakravarty, Sarvajit, Quinn, Kevin, Belmar, Sebastian, Alfaro, Ivan E., Higgs, Christopher, Bernales, Sebastian, Herrera, Francisco J., Rai, Roopa
Published in Bioorganic & medicinal chemistry letters (15.05.2017)
Published in Bioorganic & medicinal chemistry letters (15.05.2017)
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Abstract B30: Talazoparib efficacy is enhanced by noncytotoxic doses of temozolomide-mediated DNA damage in prostate cancer cell lines
Lindquist, Jeffrey N., Phan, Vernon T., Riquelme, Eduardo, Mukherjee, Kakoli, Farías, Olivia, Gupta, Ashu, Raja, Mohd, Rai, Roopa, Uppal, Hirdesh, Protter, Andrew A.
Published in Molecular cancer research (01.04.2017)
Published in Molecular cancer research (01.04.2017)
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Synthesis and structure activity relationship of imidazo[1,2-a]pyridine-8-carboxamides as a novel antimycobacterial lead series
Ramachandran, Sreekanth, Panda, Manoranjan, Mukherjee, Kakoli, Choudhury, Nilanjana Roy, Tantry, Subramanyam J., Kedari, Chaitanya Kumar, Ramachandran, Vasanthi, Sharma, Sreevalli, Ramya, V.K., Guptha, Supreeth, Sambandamurthy, Vasan K.
Published in Bioorganic & medicinal chemistry letters (01.09.2013)
Published in Bioorganic & medicinal chemistry letters (01.09.2013)
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Novel N‑Linked Aminopiperidine-Based Gyrase Inhibitors with Improved hERG and in Vivo Efficacy against Mycobacterium tuberculosis
Hameed P, Shahul, Patil, Vikas, Solapure, Suresh, Sharma, Umender, Madhavapeddi, Prashanti, Raichurkar, Anandkumar, Chinnapattu, Murugan, Manjrekar, Praveena, Shanbhag, Gajanan, Puttur, Jayashree, Shinde, Vikas, Menasinakai, Sreenivasaiah, Rudrapatana, Suresh, Achar, Vijayashree, Awasthy, Disha, Nandishaiah, Radha, Humnabadkar, Vaishali, Ghosh, Anirban, Narayan, Chandan, Ramya, V. K, Kaur, Parvinder, Sharma, Sreevalli, Werngren, Jim, Hoffner, Sven, Panduga, Vijender, Kumar, C. N. Naveen, Reddy, Jitendar, Kumar KN, Mahesh, Ganguly, Samit, Bharath, Sowmya, Bheemarao, Ugarkar, Mukherjee, Kakoli, Arora, Uma, Gaonkar, Sheshagiri, Coulson, Michelle, Waterson, David, Sambandamurthy, Vasan K, de Sousa, Sunita M
Published in Journal of medicinal chemistry (12.06.2014)
Published in Journal of medicinal chemistry (12.06.2014)
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Aminoazabenzimidazoles, a Novel Class of Orally Active Antimalarial Agents
Hameed P, Shahul, Chinnapattu, Murugan, Shanbag, Gajanan, Manjrekar, Praveena, Koushik, Krishna, Raichurkar, Anandkumar, Patil, Vikas, Jatheendranath, Sandesh, Rudrapatna, Suresh S, Barde, Shubhada P, Rautela, Nikhil, Awasthy, Disha, Morayya, Sapna, Narayan, Chandan, Kavanagh, Stefan, Saralaya, Ramanatha, Bharath, Sowmya, Viswanath, Pavithra, Mukherjee, Kakoli, Bandodkar, Balachandra, Srivastava, Abhishek, Panduga, Vijender, Reddy, Jitender, Prabhakar, K. R, Sinha, Achyut, Jiménez-Díaz, María Belén, Martínez, María Santos, Angulo-Barturen, Iñigo, Ferrer, Santiago, Sanz, Laura María, Gamo, Francisco Javier, Duffy, Sandra, Avery, Vicky M, Magistrado, Pamela A, Lukens, Amanda K, Wirth, Dyann F, Waterson, David, Balasubramanian, V, Iyer, Pravin S, Narayanan, Shridhar, Hosagrahara, Vinayak, Sambandamurthy, Vasan K, Ramachandran, Sreekanth
Published in Journal of medicinal chemistry (10.07.2014)
Published in Journal of medicinal chemistry (10.07.2014)
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Scaffold morphing leading to evolution of 2,4-diaminoquinolines and aminopyrazolopyrimidines as inhibitors of the ATP synthesis pathway
Tantry, Subramanyam J., Shinde, Vikas, Balakrishnan, Gayathri, Markad, Shankar D., Gupta, Amit K., Bhat, Jyothi, Narayan, Ashwini, Raichurkar, Anandkumar, Jena, Lalit Kumar, Sharma, Sreevalli, Kumar, Naveen, Nanduri, Robert, Bharath, Sowmya, Reddy, Jitendar, Panduga, Vijender, Prabhakar, K. R., Kandaswamy, Karthikeyan, Kaur, Parvinder, Dinesh, Neela, Guptha, Supreeth, Saralaya, Ramanatha, Panda, Manoranjan, Rudrapatna, Suresh, Mallya, Meenakshi, Rubin, Harvey, Yano, Takahiro, Mdluili, Khisi, Cooper, Christopher B., Balasubramanian, V., Sambandamurthy, Vasan K., Ramachandran, Vasanthi, Shandil, Radha, Kavanagh, Stefan, Narayanan, Shridhar, Iyer, Pravin, Mukherjee, Kakoli, Hosagrahara, Vinayak P., Solapure, Suresh, Hameed, Shahul P., Ravishankar, Sudha
Published in MedChemComm (01.01.2016)
Published in MedChemComm (01.01.2016)
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Assays, surrogates, and alternative technologies for a TB lead identification program targeting DNA gyrase ATPase
Humnabadkar, Vaishali, Madhavapeddi, Prashanti, Basavarajappa, Halesha, Sheikh, Md Gulebahar, Rane, Rajendra, Basu, Reetobrata, Verma, Prateek, Sundaram, Aishwarya, Mukherjee, Kakoli, de Sousa, Sunita M
Published in Journal of biomolecular screening (01.02.2015)
Published in Journal of biomolecular screening (01.02.2015)
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