Identification and Structure−Activity Relationships of Chromene-Derived Selective Estrogen Receptor Modulators for Treatment of Postmenopausal Symptoms
Jain, Nareshkumar, Xu, Jiayi, Kanojia, Ramesh M, Du, Fuyong, Jian-Zhong, Guo, Pacia, Emmanuel, Lai, Muh-Tsann, Musto, Amy, Allan, George, Reuman, Michael, Li, Xun, Hahn, DoWon, Cousineau, Martin, Peng, Sean, Ritchie, David, Russell, Ronald, Lundeen, Scott, Sui, Zhihua
Published in Journal of medicinal chemistry (10.12.2009)
Published in Journal of medicinal chemistry (10.12.2009)
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The discovery of a potent orally efficacious indole androgen receptor antagonist through in vivo screening
Lanter, James C., Fiordeliso, James J., Jiang, Weiqin, Allan, George F., Lai, Muh-Tsann, Linton, Olivia, Hahn, Do Won, Lundeen, Scott G., Sui, Zhihua
Published in Bioorganic & medicinal chemistry letters (2007)
Published in Bioorganic & medicinal chemistry letters (2007)
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Diverse Effects of Tyrosine Kinase Inhibitors on Follicle-Stimulating Hormone-Stimulated Estradiol and Progesterone Production from Rat Granulosa Cells in Serum-Containing Medium and Serum-Free Medium Containing Epidermal Growth Factor
Haynes-Johnson, Donna, Lai, Muh-Tsann, Campen, Carolyn, Palmer, Stephen
Published in Biology of reproduction (01.07.1999)
Published in Biology of reproduction (01.07.1999)
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Pharmacological characterization of an imidazolopyrazole as novel selective androgen receptor modulator
Zhang, Xuqing, Allan, George F., Tannenbaum, Pamela, Sbriscia, Tifanie, Linton, Olivia, Lai, Muh-Tsann, Haynes-Johnson, Donna, Bhattacharjee, Sheela, Lundeen, Scott G., Sui, Zhihua
Published in The Journal of steroid biochemistry and molecular biology (01.03.2013)
Published in The Journal of steroid biochemistry and molecular biology (01.03.2013)
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Novel Chromene-Derived Selective Estrogen Receptor Modulators Useful for Alleviating Hot Flushes and Vaginal Dryness
Jain, Nareshkumar, Kanojia, Ramesh M, Xu, Jiayi, Jian-Zhong, Guo, Pacia, Emmanuel, Lai, Muh-Tsann, Du, Fuyong, Musto, Amy, Allan, George, Hahn, Lundeen, Scott, Sui, Zhihua
Published in Journal of medicinal chemistry (01.06.2006)
Published in Journal of medicinal chemistry (01.06.2006)
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A selective androgen receptor modulator with minimal prostate hypertrophic activity restores lean body mass in aged orchidectomized male rats
Allan, George, Sbriscia, Tifanie, Linton, Olivia, Lai, Muh-Tsann, Haynes-Johnson, Donna, Bhattacharjee, Sheela, Ng, Raymond, Sui, Zhihua, Lundeen, Scott
Published in The Journal of steroid biochemistry and molecular biology (01.06.2008)
Published in The Journal of steroid biochemistry and molecular biology (01.06.2008)
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A selective androgen receptor modulator that reduces prostate tumor size and prevents orchidectomy-induced bone loss in rats
Allan, George, Lai, Muh-Tsann, Sbriscia, Tifanie, Linton, Olivia, Haynes-Johnson, Donna, Bhattacharjee, Sheela, Dodds, Robert, Fiordeliso, James, Lanter, James, Sui, Zhihua, Lundeen, Scott
Published in The Journal of steroid biochemistry and molecular biology (2007)
Published in The Journal of steroid biochemistry and molecular biology (2007)
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Journal Article
A selective androgen receptor modulator with minimal prostate hypertrophic activity enhances lean body mass in male rats and stimulates sexual behavior in female rats
Allan, George F, Tannenbaum, Pamela, Sbriscia, Tifanie, Linton, Olivia, Lai, Muh-Tsann, Haynes-Johnson, Donna, Bhattacharjee, Sheela, Zhang, Xuqing, Sui, Zhihua, Lundeen, Scott G
Published in Endocrine (01.08.2007)
Published in Endocrine (01.08.2007)
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Molecular properties and preclinical pharmacology of JNJ-1250132, a steroidal progesterone receptor modulator that inhibits binding of the receptor to DNA in vitro
Allan, George F., Palmer, Elizabeth, Musto, Amy, Lai, Muh-Tsann, Clancy, Joanna, Palmer, Stephen
Published in Steroids (01.07.2006)
Published in Steroids (01.07.2006)
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β-Alkylthio indolyl carbinols: Potent nonsteroidal antiandrogens with oral efficacy in a prostate cancer model
Lanter, James C., Fiordeliso, James J., Alford, Vernon C., Zhang, Xuqing, Wells, Kenneth M., Russell, Ronald K., Allan, George F., Lai, Muh-Tsann, Linton, Olivia, Lundeen, Scott, Sui, Zhihua
Published in Bioorganic & medicinal chemistry letters (01.05.2007)
Published in Bioorganic & medicinal chemistry letters (01.05.2007)
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Journal Article
Potent pituitary-gonadal axis suppression and extremely low anaphylactoid activity of a new gonadotropin releasing hormone (GnRH) receptor antagonist “azaline B”
Campen, Carolyn A., Lai, Muh-Tsann, Kraft, Pat, Kirchner, Tom, Phillips, Audrey, Hahn, Do Won, Rivier, Jean
Published in Biochemical pharmacology (11.05.1995)
Published in Biochemical pharmacology (11.05.1995)
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Nonsteroidal progesterone receptor ligands with unprecedented receptor selectivity
Palmer, Stephen, Campen, Carolyn A, Allan, George F, Rybczynski, Philip, Haynes-Johnson, Donna, Hutchins, Amy, Kraft, Patricia, Kiddoe, Margaret, Lai, Muh-Tsann, Lombardi, Elizabeth, Pedersen, Phyllis, Hodgen, Gary, Combs, Donald W
Published in The Journal of steroid biochemistry and molecular biology (01.12.2000)
Published in The Journal of steroid biochemistry and molecular biology (01.12.2000)
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Synthesis and progesterone receptor binding affinity of substituted 1-phenyl-7-benzyl-4,5,6,7-tetrahydro-1H-indazoles
CONNOLLY, P. J, WETTER, S. K, PHILLIPS, A, BEERS, K. N, HAMEL, S. C, HAYNES-JOHNSON, D, KIDDOE, M, KRAFT, P, MUH TSANN LAI, CAMPEN, C, PALMER, S
Published in Bioorganic & medicinal chemistry letters (07.10.1997)
Published in Bioorganic & medicinal chemistry letters (07.10.1997)
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Journal Article
Novel Chromene-Derived Selective Estrogen Receptor Modulators Useful for Alleviating Hot Flushes and Vaginal Dryness
JAIN, Nareshkumar, KANOJIA, Ramesh M., XU, Jiayi, JIAN-ZHONG, Guo, PACIA, Emmanuel, LAI, Muh-Tsann, DU, Fuyong, MUSTO, Amy, ALLAN, George, HAHN, LUNDEEN, Scott, SUI, Zhihua
Published in Journal of medicinal chemistry (01.06.2006)
Published in Journal of medicinal chemistry (01.06.2006)
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Journal Article
Synthesis and progesterone receptor binding affinity of substituted 1-phenyl-7-benzyl-4,5,6,7-tetrahydro-1 [formula omitted]-indazoles
Connolly, Peter J., Wetter, Steven K., Beers, Kimberly N., Hamel, Stephanie C., Haynes-Johnson, Donna, Kiddoe, Margaret, Kraft, Pat, Tsann Lai, Muh, Campen, Carolyn, Palmer, Stephen, Phillips, Audrey
Published in Bioorganic & medicinal chemistry letters (01.10.1997)
Published in Bioorganic & medicinal chemistry letters (01.10.1997)
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