Process Research and Development for an Efficient Synthesis of the HIV Protease Inhibitor BMS-232632
Xu, Zhongmin, Singh, Janak, Schwinden, Mark D, Zheng, Bin, Kissick, Thomas P, Patel, Bharat, Humora, Michael J, Quiroz, Fernando, Dong, Lin, Hsieh, Dau-Ming, Heikes, James E, Pudipeddi, Madhusudhan, Lindrud, Mark D, Srivastava, Sushil K, Kronenthal, David R, Mueller, Richard H
Published in Organic process research & development (01.05.2002)
Published in Organic process research & development (01.05.2002)
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Efficient Asymmetric Synthesis of the Vasopeptidase Inhibitor BMS-189921
Singh, Janak, Kronenthal, David R, Schwinden, Mark, Godfrey, Jollie D, Fox, Rita, Vawter, Edward J, Zhang, Bo, Kissick, Thomas P, Patel, Bharat, Mneimne, Omar, Humora, Michael, Papaioannou, Chris G, Szymanski, Walter, Wong, Michael K. Y, Chen, Chien K, Heikes, James E, DiMarco, John D, Qiu, Jun, Deshpande, Rajendra P, Gougoutas, Jack Z, Mueller, Richard H
Published in Organic letters (21.08.2003)
Published in Organic letters (21.08.2003)
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Improved synthesis of aryl 1,1-dimethylpropargyl ethers
Godfrey, Jollie D., Mueller, Richard H., Sedergran, Thomas C., Soundararajan, Nachimuthu, Colandrea, Vincent J.
Published in Tetrahedron letters (29.08.1994)
Published in Tetrahedron letters (29.08.1994)
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Regioselective enzymatic aminoacylation of lobucavir to give an intermediate for lobucavir prodrug
Hanson, Ronald L, Shi, Zhongping, Brzozowski, David B, Banerjee, Amit, Kissick, Thomas P, Singh, Janak, Pullockaran, Annie J, North, Jeffrey T, Fan, Junying, Howell, Jeffrey, Durand, Susan C, Montana, Michael A, Kronenthal, David R, Mueller, Richard H, Patel, Ramesh N
Published in Bioorganic & medicinal chemistry (01.12.2000)
Published in Bioorganic & medicinal chemistry (01.12.2000)
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Journal Article
Regioselective Activation of Aminothiazole(iminoxyacetic acid)acetic Acid: An Efficient Synthesis of the Monobactam Aztreonam
Singh, Janak, Denzel, Theodor W, Fox, Rita, Kissick, Thomas P, Herter, Rolf, Wurdinger, Joseph, Schierling, Peter, Papaioannou, Chris G, Moniot, Jerome L, Mueller, Richard H, Cimarusti, Christopher M
Published in Organic process research & development (01.11.2002)
Published in Organic process research & development (01.11.2002)
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Regioselective Coupling of Tetraalkylammonium Salts of 6-Iodo-2-aminopurine to a Cyclobutyl Triflate: Efficient Preparation of Homochiral BMS-180,194, a Potent Antiviral Carbocyclic Nucleoside
Bisacchi, Gregory S., Singh, Janak, Godfrey, Jollie D., Kissick, Thomas P., Mitt, Toomas, Malley, Mary F., Di Marco, John D., Gougoutas, Jack Z., Mueller, Richard H., Zahler, Robert
Published in Journal of organic chemistry (01.05.1995)
Published in Journal of organic chemistry (01.05.1995)
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Synthesis and anti-MRSA Activity of Novel Cephalosporin Derivatives
D'Andrea, Stan V., Bonner, Daniel, Bronson, Joanne J., Clark, Junius, Denbleyker, Ken, Fung-Tomc, Joan, Hoeft, Shelley E., Hudyma, Thomas W., Matiskella, John D., Miller, Raymond F., Misco, Peter F., Pucci, Michael, Sterzycki, Roman, Tsai, Yuan, Ueda, Yasutsuga, Wichtowski, John A., Singh, Janak, Kissick, Thomas P., North, Jeffery T., Pullockaran, Annie, Humora, Michael, Boyhan, Brenda, Vu, Truc, Fritz, Alan, Heikes, J., Fox, Rita, Godfrey, Jollie D., Perrone, Robert, Kaplan, Murray, Kronenthal, David, Mueller, Richard H.
Published in Tetrahedron (28.07.2000)
Published in Tetrahedron (28.07.2000)
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Journal Article
A Practical Asymmetric Synthesis of the Antiviral Agent Lobucavir, BMS-180194
Singh, Janak, Bisacchi, Gregory S, Ahmad, Saleem, Godfrey, Jollie D, Kissick, Thomas P, Mitt, Toomas, Kocy, Octavian, Vu, Truc, Papaioannou, Chris G, Wong, Michael K, Heikes, James E, Zahler, Robert, Mueller, Richard H
Published in Organic process research & development (01.11.1998)
Published in Organic process research & development (01.11.1998)
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Journal Article
NOVEL METHODS FOR SYNTHESES OF SUBSTITUTED OXAZOLES BY CYCLIZATION OF VINYL BROMIDES
DAS, J, REID, JA, KRONENTHAL, DR, SINGH, J, PANSEGRAU, PD, MUELLER, RH
Published in Tetrahedron letters (15.12.1992)
Published in Tetrahedron letters (15.12.1992)
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Diastereoselective Reaction of a Grignard Reagent with Chiral Imides: A Practical Preparation of a Key Intermediate in the Synthesis of Ifetroban Sodium
Mueller, Richard H, Wang, Shaopeng, Pansegrau, Paul D, Jannotti, Joy Q, Poss, Michael A, Thottathil, John K, Singh, Janak, Humora, Michael J, Kissick, Thomas P, Boyhan, Brenda
Published in Organic process research & development (01.01.1997)
Published in Organic process research & development (01.01.1997)
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Journal Article
A Practical Asymmetric Synthesis of the Antiviral Agent Lobucavir, BMS-180194
Singh, Janak, Bisacchi, Gregory S, Ahmad, Saleem, Godfrey, Jollie D, Kissick, Thomas P, Mitt, Toomas, Kocy, Octavian, Vu, Truc, Papaioannou, Chris G, Wong, Michael K, Heikes, James E, Zahler, Robert, Mueller, Richard H
Published in Organic process research & development (01.05.1999)
Published in Organic process research & development (01.05.1999)
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Journal Article
Claisen rearrangement of allyl esters
Ireland, Robert E, Mueller, Richard H
Published in Journal of the American Chemical Society (01.08.1972)
Published in Journal of the American Chemical Society (01.08.1972)
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Journal Article
Stereospecific microbial reduction of 4,5-dihydro-4-(4-methoxyphenyl)-6-(trifluoromethyl-1H-1)-benzazepin-2-one
Patel, Ramesh N., Robison, Robert S., Szarka, Laszo J., Kloss, John, Thottathil, John K., Mueller, Richard H.
Published in Enzyme and microbial technology (1991)
Published in Enzyme and microbial technology (1991)
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Journal Article
Synthesis of l-β-hydroxyvaline from α-keto-β-hydroxyisovalerate using leucine dehydrogenase from Bacillus species
Hanson, Ronald L., Singh, Janak, Kissick, Thomas P., Patel, Ramesh N., Szarka, Laszlo J., Mueller, Richard H.
Published in Bioorganic chemistry (01.06.1990)
Published in Bioorganic chemistry (01.06.1990)
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IMPROVED PROCEDURE FOR THE ONE-STEP SYNTHESIS OF ALPHA-KETOESTERS
SINGH, J, KISSICK, TP, MUELLER, RH
Published in Organic preparations and procedures international (01.08.1989)
Published in Organic preparations and procedures international (01.08.1989)
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