Distinct roles of metabotropic glutamate receptor dimerization in agonist activation and G-protein coupling
El Moustaine, Driss, Granier, Sébastien, Doumazane, Etienne, Scholler, Pauline, Rahmeh, Rita, Bron, Patrick, Mouillac, Bernard, Banères, Jean-Louis, Rondard, Philippe, Pin, Jean-Philippe
Published in Proceedings of the National Academy of Sciences - PNAS (02.10.2012)
Published in Proceedings of the National Academy of Sciences - PNAS (02.10.2012)
Get full text
Journal Article
Structural insights into biased G protein-coupled receptor signaling revealed by fluorescence spectroscopy
Rahmeh, Rita, Damian, Marjorie, Cottet, Martin, Orcel, Hélène, Mendre, Christiane, Durroux, Thierry, Sharma, K. Shivaji, Durand, Grégory, Pucci, Bernard, Trinquet, Eric, Zwier, Jurriaan M, Deupi, Xavier, Bron, Patrick, Banères, Jean-Louis, Mouillac, Bernard, Granier, Sébastien
Published in Proceedings of the National Academy of Sciences - PNAS (24.04.2012)
Published in Proceedings of the National Academy of Sciences - PNAS (24.04.2012)
Get full text
Journal Article
The ligand-bound state of a G protein-coupled receptor stabilizes the interaction of functional cholesterol molecules
Lemel, Laura, Nieścierowicz, Katarzyna, García-Fernández, M. Dolores, Darré, Leonardo, Durroux, Thierry, Busnelli, Marta, Pezet, Mylène, Rébeillé, Fabrice, Jouhet, Juliette, Mouillac, Bernard, Domene, Carmen, Chini, Bice, Cherezov, Vadim, Moreau, Christophe J.
Published in Journal of lipid research (01.01.2021)
Published in Journal of lipid research (01.01.2021)
Get full text
Journal Article
Ghrelin receptor conformational dynamics regulate the transition from a preassembled to an active receptor:Gq complex
Damian, Marjorie, Mary, Sophie, Maingot, Mathieu, M’Kadmi, Céline, Gagne, Didier, Leyris, Jean-Philippe, Denoyelle, Séverine, Gaibelet, Gérald, Gavara, Laurent, de Souza Costa, Mauricio Garcia, Perahia, David, Trinquet, Eric, Mouillac, Bernard, Galandrin, Ségolène, Galès, Céline, Fehrentz, Jean-Alain, Floquet, Nicolas, Martinez, Jean, Marie, Jacky, Banères, Jean-Louis
Published in Proceedings of the National Academy of Sciences - PNAS (03.02.2015)
Published in Proceedings of the National Academy of Sciences - PNAS (03.02.2015)
Get full text
Journal Article
Functional Rescue of a Nephrogenic Diabetes Insipidus Causing Mutation in the V2 Vasopressin Receptor by Specific Antagonist and Agonist Pharmacochaperones
Szalai, Laura, Sziráki, András, Erdélyi, László Sándor, Kovács, Kinga Bernadett, Tóth, Miklós, Tóth, András Dávid, Turu, Gábor, Bonnet, Dominique, Mouillac, Bernard, Hunyady, László, Balla, András
Published in Frontiers in pharmacology (25.01.2022)
Published in Frontiers in pharmacology (25.01.2022)
Get full text
Journal Article
V1b vasopressin receptor trafficking and signaling: Role of arrestins, G proteins and Src kinase
Perkovska, Sanja, Méjean, Catherine, Ayoub, Mohammed Akli, Li, Juan, Hemery, Floriane, Corbani, Maithé, Laguette, Nadine, Ventura, Maria‐Angeles, Orcel, Hélène, Durroux, Thierry, Mouillac, Bernard, Mendre, Christiane
Published in Traffic (Copenhagen, Denmark) (01.01.2018)
Published in Traffic (Copenhagen, Denmark) (01.01.2018)
Get full text
Journal Article
Red Fluorescent Turn-On Ligands for Imaging and Quantifying G Protein-Coupled Receptors in Living Cells
Karpenko, Iuliia A., Kreder, Rémy, Valencia, Christel, Villa, Pascal, Mendre, Christiane, Mouillac, Bernard, Mély, Yves, Hibert, Marcel, Bonnet, Dominique, Klymchenko, Andrey S.
Published in Chembiochem : a European journal of chemical biology (10.02.2014)
Published in Chembiochem : a European journal of chemical biology (10.02.2014)
Get full text
Journal Article
Biased Agonist Pharmacochaperones of the AVP V2 Receptor May Treat Congenital Nephrogenic Diabetes Insipidus
JEAN-ALPHONSE, Frédéric, PERKOVSKA, Sanja, MENDRE, Christiane, FRANTZ, Marie-Céline, DURROUX, Thierry, MEJEAN, Catherine, MORIN, Denis, LOISON, Stéphanie, BONNET, Dominique, HIBERT, Marcel, MOUILLAC, Bernard
Published in Journal of the American Society of Nephrology (01.10.2009)
Published in Journal of the American Society of Nephrology (01.10.2009)
Get full text
Journal Article
Oxytocin and Vasopressin V1a and V2 Receptors Form Constitutive Homo- and Heterodimers during Biosynthesis
Terrillon, Sonia, Durroux, Thierry, Mouillac, Bernard, Breit, Andreas, Ayoub, Mohammed A, Taulan, Magali, Jockers, Ralf, Barberis, Claude, Bouvier, Michel
Published in Molecular endocrinology (Baltimore, Md.) (01.04.2003)
Published in Molecular endocrinology (Baltimore, Md.) (01.04.2003)
Get full text
Journal Article
Cryo-electron microscopy structure of the antidiuretic hormone arginine-vasopressin V2 receptor signaling complex
Bous, Julien, Orcel, Hélène, Floquet, Nicolas, Leyrat, Cédric, Lai-Kee-Him, Joséphine, Gaibelet, Gérald, Ancelin, Aurélie, Saint-Paul, Julie, Trapani, Stefano, Louet, Maxime, Sounier, Rémy, Déméné, Hélène, Granier, Sébastien, Bron, Patrick, Mouillac, Bernard
Published in Science advances (21.05.2021)
Published in Science advances (21.05.2021)
Get full text
Journal Article
Probing the Existence of G Protein-Coupled Receptor Dimers by Positive and Negative Ligand-Dependent Cooperative Binding
Albizu, Laura, Balestre, Marie-Noëlle, Breton, Christophe, Pin, Jean-Philippe, Manning, Maurice, Mouillac, Bernard, Barberis, Claude, Durroux, Thierry
Published in Molecular pharmacology (01.11.2006)
Published in Molecular pharmacology (01.11.2006)
Get full text
Journal Article
Toward Efficient Drug Screening by Homogeneous Assays Based on the Development of New Fluorescent Vasopressin and Oxytocin Receptor Ligands
Albizu, Laura, Teppaz, Géraldine, Seyer, René, Bazin, Hervé, Ansanay, Hervé, Manning, Maurice, Mouillac, Bernard, Durroux, Thierry
Published in Journal of medicinal chemistry (04.10.2007)
Published in Journal of medicinal chemistry (04.10.2007)
Get full text
Journal Article
Inhibition of oxytocin receptor function by direct binding of progesterone
Zingg, Hans H, Grazzini, Eric, Guillon, Gilles, Mouillac, Bernard
Published in Nature (London) (02.04.1998)
Published in Nature (London) (02.04.1998)
Get full text
Journal Article
Leukotriene BLT2 Receptor Monomers Activate the Gi2 GTP-binding Protein More Efficiently than Dimers
Arcemisbéhère, Laure, Sen, Tuhinadri, Boudier, Laure, Balestre, Marie-Noëlle, Gaibelet, Gérald, Detouillon, Emilie, Orcel, Hélène, Mendre, Christiane, Rahmeh, Rita, Granier, Sébastien, Vivès, Corinne, Fieschi, Franck, Damian, Marjorie, Durroux, Thierry, Banères, Jean-Louis, Mouillac, Bernard
Published in The Journal of biological chemistry (26.02.2010)
Published in The Journal of biological chemistry (26.02.2010)
Get full text
Journal Article
The constitutively active V2 receptor mutants conferring NSIAD are weakly sensitive to agonist and antagonist regulation
Tenenbaum, Julie, Ayoub, Mohammed A, Perkovska, Sanja, Adra-Delenne, Anne-Laure, Mendre, Christiane, Ranchin, Bruno, Bricca, Giamperro, Geelen, Ghislaine, Mouillac, Bernard, Durroux, Thierry, Morin, Denis
Published in PloS one (21.12.2009)
Published in PloS one (21.12.2009)
Get full text
Journal Article
Differential Coupling of the Vasopressin V1b Receptor through Compartmentalization within the Plasma Membrane
Orcel, Hélène, Albizu, Laura, Perkovska, Sanja, Durroux, Thierry, Mendre, Christiane, Ansanay, Hervé, Mouillac, Bernard, Rabié, Alain
Published in Molecular pharmacology (01.03.2009)
Published in Molecular pharmacology (01.03.2009)
Get full text
Journal Article
Identification of the Binding Sites of the SR49059 Nonpeptide Antagonist into the V1a Vasopressin Receptor Using Sulfydryl-reactive Ligands and Cysteine Mutants as Chemical Sensors
Tahtaoui, Chouaïb, Balestre, Marie-Noëlle, Klotz, Philippe, Rognan, Didier, Barberis, Claude, Mouillac, Bernard, Hibert, Marcel
Published in The Journal of biological chemistry (10.10.2003)
Published in The Journal of biological chemistry (10.10.2003)
Get full text
Journal Article