Antisense Oligonucleotides
De Mesmaeker, Alain, Haener, Robert, Martin, Pierre, Moser, Heinz E
Published in Accounts of chemical research (01.09.1995)
Published in Accounts of chemical research (01.09.1995)
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Journal Article
DNA binding ligands targeting drug-resistant Gram-positive bacteria. Part 1: Internal benzimidazole derivatives
Bürli, Roland W, McMinn, Dustin, Kaizerman, Jacob A, Hu, Wenhao, Ge, Yigong, Pack, Quinn, Jiang, Vernon, Gross, Matthew, Garcia, Martin, Tanaka, Richard, Moser, Heinz E
Published in Bioorganic & medicinal chemistry letters (08.03.2004)
Published in Bioorganic & medicinal chemistry letters (08.03.2004)
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Journal Article
Matrix-assisted laser desorption ionization time-of-flight mass spectrometry: a powerful tool for the mass and sequence analysis of natural and modified oligonucleotides
Pieles, Uwe, Zürcher, Werner, Schär, Martin, Moser, Heinz
Published in Nucleic acids research (11.07.1993)
Published in Nucleic acids research (11.07.1993)
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Journal Article
DNA binding ligands targeting drug-resistant Gram-positive bacteria. Part 2: C-terminal benzimidazoles and derivatives
Bürli, Roland W, Jones, Peter, McMinn, Dustin, Le, Quan, Duan, Jian-Xin, Kaizerman, Jacob A, Difuntorum, Stacey, Moser, Heinz E
Published in Bioorganic & medicinal chemistry letters (08.03.2004)
Published in Bioorganic & medicinal chemistry letters (08.03.2004)
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Journal Article
Dual Recognition of Double-Stranded DNA by 2′-Aminoethoxy-Modified Oligonucleotides
Cuenoud, Bernard, Casset, Florence, Hüsken, Dieter, Natt, François, Wolf, Romain M., Altmann, Karl-Heinz, Martin, Pierre, Moser, Heinz E.
Published in Angewandte Chemie (International ed.) (18.05.1998)
Published in Angewandte Chemie (International ed.) (18.05.1998)
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Sequence-Specific Cleavage of Double Helical DNA by Triple Helix Formation
Moser, Heinz E., Dervan, Peter B.
Published in Science (American Association for the Advancement of Science) (30.10.1987)
Published in Science (American Association for the Advancement of Science) (30.10.1987)
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Journal Article
DNA Binding Ligands with Improved in Vitro and in Vivo Potency against Drug-Resistant Staphylococcus aureus
Hu, Wenhao, Bürli, Roland W, Kaizerman, Jacob A, Johnson, Kirk W, Gross, Matthew I, Iwamoto, Mari, Jones, Peter, Lofland, Denene, Difuntorum, Stacey, Chen, Hsiu, Bozdogan, Bülent, Appelbaum, Peter C, Moser, Heinz E
Published in Journal of medicinal chemistry (26.08.2004)
Published in Journal of medicinal chemistry (26.08.2004)
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Journal Article
DNA Binding Ligands with Excellent Antibiotic Potency Against Drug-Resistant Gram-Positive Bacteria
Bürli, Roland W., Ge, Yigong, White, Sarah, Baird, Eldon E., Touami, Sofia M., Taylor, Matthew, Kaizerman, Jacob A., Moser, Heinz E.
Published in Bioorganic & medicinal chemistry letters (16.09.2002)
Published in Bioorganic & medicinal chemistry letters (16.09.2002)
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Journal Article
DNA Binding Ligands Targeting Drug-Resistant Bacteria: Structure, Activity, and Pharmacology
Kaizerman, Jacob A, Gross, Matthew I, Ge, Yigong, White, Sarah, Hu, Wenhao, Duan, Jian-Xin, Baird, Eldon E, Johnson, Kirk W, Tanaka, Richard D, Moser, Heinz E, Bürli, Roland W
Published in Journal of medicinal chemistry (28.08.2003)
Published in Journal of medicinal chemistry (28.08.2003)
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Journal Article
DNA binding ligands with in vivo efficacy in murine models of bacterial infection: optimization of internal aromatic amino acids
BÜRLI, Roland W, KAIZERMAN, Jacob A, TOUAMI, Sofia, GROSS, Matthew, JIANG, Vernon, YIGONG GE, MOSER, Heinz E, DUAN, Jian-Xin, JONES, Peter, JOHNSON, Kirk W, IWAMOTO, Mari, TRUONG, Kiet, WENHAO HU, STANTON, Timothy, CHEN, Alfred
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Journal Article
Second Generation of Antisense Oligonucleotides: From Nuclease Resistance to Biological Efficacy in Animals
Karl-Heinz Altmann, Henri Sasmor, Uwe Pieles, Judy Phillipsd, Paul Nicklind, Fram;ois Natt, Marcel Miiller, Brett P.B Monia, Pierre Martina, Dieter A Hiisken, Robert Hanera, Thomas Geiger, Susan M. Freier, Doriano Fabbro, Nicholas M. Dean, Heinz E Moser
Published in Chimia (24.04.1996)
Published in Chimia (24.04.1996)
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Journal Article
Double strand cleavage of genomic DNA at a single site by triple helix formation
Strobel, Scott A., Moser, Heinz E., Dervan, Peter B.
Published in Journal of the American Chemical Society (01.11.1988)
Published in Journal of the American Chemical Society (01.11.1988)
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Journal Article
Creating RNA Bulges: Cleavage of RNA in RNA/DNA Duplexes by Metal Ion Catalysis
Hüsken, Dieter, Goodall, Greg, Blommers, Marcel J. J, Jahnke, Wolfgang, Hall, Jonathan, Häner, Robert, Moser, Heinz E
Published in Biochemistry (Easton) (24.12.1996)
Published in Biochemistry (Easton) (24.12.1996)
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Distribution of a 20-mer phosphorothioate oligonucleotide, CGP69846A (ISIS 5132), into airway leukocytes and epithelial cells following intratracheal delivery to Brown-Norway rats
DANAHAY, H, GIDDINGS, J, CHRISTIAN, R. A, MOSER, H. E, PHILLIPS, J. A
Published in Pharmaceutical research (01.10.1999)
Published in Pharmaceutical research (01.10.1999)
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Journal Article
A novel fluorogenic substrate for ribonucleases. Synthesis and enzymatic characterization
Zelenko, Ottilie, Neumann, Ulf, Brill, Wolfgang, Pieles, Uwe, Moser, Heinz E., Hofsteenge, Jan
Published in Nucleic acids research (25.07.1994)
Published in Nucleic acids research (25.07.1994)
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Journal Article
Sequence analysis of phosphorothioate oligonucleotides via matrix-assisted laser desorption ionization time-of-flight mass spectrometry
Schuette, Jodi M., Pieles, Uwe, Maleknia, Simin D., Srivatsa, G.Susan, Cole, Douglas L., Moser, Heinz E., Afeyan, Noubar B.
Published in Journal of pharmaceutical and biomedical analysis (01.09.1995)
Published in Journal of pharmaceutical and biomedical analysis (01.09.1995)
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