Effect of N-methyl substitution of the peptide bonds in luteinizing hormone-releasing hormone agonists
Haviv, Fortuna, Fitzpatrick, Timothy D, Swenson, Rolf E, Nichols, Charles J, Mort, Nicholas A, Bush, Eugene N, Diaz, Gilbert, Bammert, Gary, Nguyen, A
Published in Journal of medicinal chemistry (01.02.1993)
Published in Journal of medicinal chemistry (01.02.1993)
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Synthesis and Activity of New Aryl- and Heteroaryl-Substituted Pyrazole Inhibitors of the Transforming Growth Factor-β Type I Receptor Kinase Domain
Sawyer, J. Scott, Anderson, Bryan D, Beight, Douglas W, Campbell, Robert M, Jones, Michael L, Herron, David K, Lampe, John W, McCowan, Jefferson R, McMillen, William T, Mort, Nicholas, Parsons, Stephen, Smith, Edward C. R, Vieth, Michal, Weir, Leonard C, Yan, Lei, Zhang, Faming, Yingling, Jonathan M
Published in Journal of medicinal chemistry (11.09.2003)
Published in Journal of medicinal chemistry (11.09.2003)
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Synthesis and activity of new aryl- and heteroaryl-substituted 5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole inhibitors of the transforming growth factor-β type I receptor kinase domain
SAWYER, J. Scott, BEIGHT, Douglas W, PARSONS, Stephen, SMITH, Edward C. R, WAGNER, Jill R, LEI YAN, FAMING ZHANG, YINGLING, Jonathan M, BRITT, Karen S, ANDERSON, Bryan D, CAMPBELL, Robert M, GOODSON, Theodore JR, HERRON, David K, LI, Hong-Yu, MCMILLEN, William T, MORT, Nicholas
Published in Bioorganic & medicinal chemistry letters (05.07.2004)
Published in Bioorganic & medicinal chemistry letters (05.07.2004)
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Kinetic Characterization of Novel Pyrazole TGF-β Receptor I Kinase Inhibitors and Their Blockade of the Epithelial−Mesenchymal Transition
Peng, Sheng-Bin, Yan, Lei, Xia, Xiaoling, Watkins, Scott A, Brooks, Harold B, Beight, Douglas, Herron, David K, Jones, Michael L, Lampe, John W, McMillen, William T, Mort, Nicholas, Sawyer, J. Scott, Yingling, Jonathan M
Published in Biochemistry (Easton) (22.02.2005)
Published in Biochemistry (Easton) (22.02.2005)
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Journal Article
The effect of NMeTyr5 substitution in luteinizing hormone-releasing hormone antagonists
Haviv, Fortuna, Fitzpatrick, Timothy D, Nichols, Charles J, Swenson, Rolf E, Mort, Nicholas A, Bush, Eugene N, Diaz, Gilbert, Nguyen, A. T, Holst, Mark R
Published in Journal of medicinal chemistry (01.04.1993)
Published in Journal of medicinal chemistry (01.04.1993)
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Journal Article
Synthesis and activity of new aryl- and heteroaryl-substituted 5,6-dihydro-4 H-pyrrolo[1,2- b]pyrazole inhibitors of the transforming growth factor-β type I receptor kinase domain
Scott Sawyer, J., Beight, Douglas W., Britt, Karen S., Anderson, Bryan D., Campbell, Robert M., Goodson, Theodore, Herron, David K., Li, Hong-Yu, McMillen, William T., Mort, Nicholas, Parsons, Stephen, Smith, Edward C.R., Wagner, Jill R., Yan, Lei, Zhang, Faming, Yingling, Jonathan M.
Published in Bioorganic & medicinal chemistry letters (2004)
Published in Bioorganic & medicinal chemistry letters (2004)
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Journal Article
THE EFFECT OF NMETYR(5) SUBSTITUTION IN LUTEINIZING-HORMONE-RELEASING HORMONE ANTAGONISTS
HAVIV, F, FITZPATRICK, TD, NICHOLS, CJ, SWENSON, RE, MORT, NA, BUSH, EN, DIAZ, G, NGUYEN, AT, HOLST, MR, CYBULSKI, VA, LEAL, JA, BAMMERT, G, RHUTASEL, NS, DODGE, PW, JOHNSON, ES, CANNON, JB, KNITTLE, J, GREER, J
Published in Journal of medicinal chemistry (02.04.1993)
Published in Journal of medicinal chemistry (02.04.1993)
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Journal Article
Novel pyrrole derivatives as pharmaceutical agents
MORT NICHOLAS ANTHONY, BEIGHT DOUGLAS WADE, GODFREY ALEXANDER GLENN, MCMILLEN WILLIAM THOMAS, YINGLING JONATHAN MICHAEL, SAWYER JASON SCOTT, LIAO JUNKAI, LI HONG-YU, CIAPETTI PAOLA, SMITH EDWARD C. R, HERRON DAVID KENT, MILLER SHAWN CHRISTOPHER, DECOLLO TODD VINCENT, GOODSON THEODORE JUNIOR
Year of Publication 04.01.2012
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Year of Publication 04.01.2012
Patent
N-TERMINUS MODIFIED ANALOG OF LHRH
SWENSON ROLF E, HAVIV FORTUNA, FITZPATRICK TIMOTHY D, NICHOLS CHARLES J, MORT NICHOLAS A
Year of Publication 30.06.2005
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Year of Publication 30.06.2005
Patent
MACROLIDE LHRH ANTAGONISTS
DALTON CHRISTOPHER R, GREER JONATHON, HAVIV FORTUNA, FREY LISA MARIE, CRAWFORD BRADLEY W, SAUER DARYL R, RANDOLPH JOHN, MORT NICHOLAS A, KAMINSKI MICHELE A, BRUNCKO MILAN
Year of Publication 31.10.2005
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Year of Publication 31.10.2005
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ANTAGONISTAS MACROLIDOS DE LHRH
MORT, NICHOLAS A, CRAWFORD, BRADLEY W, CHRISTOPHER R. DALTON, SAUER, DARYL R, RANDOLPH, JOHN, BRUNCKO, MILAN, KAMINSKI, MICHELE A, HAVIV, FORTUNA, FREY, LISA MARIE, GREER, JONATHON
Year of Publication 30.06.2005
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Year of Publication 30.06.2005
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MAKROLID-LHRH-ANTAGONISTEN
DALTON, CHRISTOPHER, R, CRAWFORD, BRADLEY, W, FREY, LISA, MARIE, RANDOLPH, JOHN, BRUNCKO, MILAN, HAVIV, FORTUNA, KAMINSKI, MICHELE, A, GREER, JONATHON, MORT, NICHOLAS, A, SAUER, DARYL, R
Year of Publication 15.03.2005
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Year of Publication 15.03.2005
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MACROLIDE LHRH ANTAGONISTS
DALTON, CHRISTOPHER, R, CRAWFORD, BRADLEY, W, FREY, LISA, MARIE, RANDOLPH, JOHN, BRUNCKO, MILAN, HAVIV, FORTUNA, KAMINSKI, MICHELE, A, GREER, JONATHON, MORT, NICHOLAS, A, SAUER, DARYL, R
Year of Publication 23.02.2005
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Year of Publication 23.02.2005
Patent
6-POSITION MODIFIED DECAPEPTIDE LHRH ANTAGONISTS
MORT, NICHOLAS A, GREER, JONATHAN, SWENSON, ROLF E, HAVIV, FORTUNA, NICHOLS, CHARLES J, FITZPATRICK, TIMOTHY D
Year of Publication 18.11.1998
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Year of Publication 18.11.1998
Patent
6-position modified decapeptide LHRH antagonists
HAVIV; FORTUNA, GREER; JONATHAN, SWENSON; ROLF E, NICHOLS; CHARLES J, MORT; NICHOLAS A, FITZPATRICK; TIMOTHY D
Year of Publication 16.12.1997
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Year of Publication 16.12.1997
Patent
3',3'-N-bis-substituted macrolide LHRH antagonists
RAWFORD, BRADLEY W, DALTON, CHRISTOPHER R, MORT, NICHOLAS A, SAUER, DARYL R, ANDOLPH, JOHN, KAMINSKI, MICHELE A, BRUNCKO, MILAN, HAVIV, FORTUNA, GREER, JONATHON
Year of Publication 28.03.2003
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Year of Publication 28.03.2003
Patent
Macrolide LHRH antagonists
WAID; PHILIP, HAVIV; FORTUNA, GREER; JONATHAN, SAUER; DARYL, NICHOLS; CHARLES J, MORT; NICHOLAS A, RANDOLPH; JOHN T, DALTON; CHRISTOPHER R
Year of Publication 01.02.2000
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Year of Publication 01.02.2000
Patent
N-TERMINUS MODIFIED ANALOGS OF LHRH
MORT, NICHOLAS A, SWENSON, ROLF E, HAVIV, FORTUNA, NICHOLS, CHARLES, J, FITZPATRICK, TIMOTHY D
Year of Publication 23.10.1996
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Year of Publication 23.10.1996
Patent