Asymmetric nucleophilic fluorination under hydrogen bonding phase-transfer catalysis
Pupo, Gabriele, Ibba, Francesco, Ascough, David M H, Vicini, Anna Chiara, Ricci, Paolo, Christensen, Kirsten E, Pfeifer, Lukas, Morphy, John Richard, Brown, John M, Paton, Robert S, Gouverneur, Véronique
Published in Science (American Association for the Advancement of Science) (11.05.2018)
Published in Science (American Association for the Advancement of Science) (11.05.2018)
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Identification and optimisation of novel sulfonamide, selective vasopressin V₁B receptor antagonists
Baker, James, Bingham, Matilda, Blackburn-Munro, Ruth, Cai, Jiaqiang, Craighead, Mark, Gilfillan, Robert, Goan, Kate, Jaap, David, Milne, Rachel, Richard Morphy, J, Napier, Susan, Presland, Jeremy, Spinks, Gayle, Thomson, Fiona
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
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Synthesis and SAR studies of novel 2-(6-aminomethylaryl-2-aryl-4-oxo-quinazolin-3(4H)-yl)acetamide Vasopressin V₁b receptor antagonists
Napier, Susan E, Letourneau, Jeffrey J, Ansari, Nasrin, Auld, Douglas S, Baker, James, Best, Stuart, Campbell-Wan, Leigh, Chan, Ray, Craighead, Mark, Desai, Hema, Ho, Koc-Kan, MacSweeney, Cliona, Milne, Rachel, Richard Morphy, J, Neagu, Irina, Ohlmeyer, Michael H.J, Pick, Jack, Presland, Jeremy, Riviello, Chris, Zanetakos, Heather A, Zhao, Jiuqiao, Webb, Maria L
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
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Design, synthesis, and structure–activity relationships of indole-3-carboxamides as novel water soluble cannabinoid CB1 receptor agonists
Adam, Julia M., Cairns, Jim, Caulfield, Wilson, Cowley, Phillip, Cumming, Iain, Easson, Morag, Edwards, Darren, Ferguson, Morag, Goodwin, Richard, Jeremiah, Fiona, Kiyoi, Takao, Mistry, Ashvin, Moir, Elizabeth, Morphy, Richard, Tierney, Jason, York, Mark, Baker, James, Cottney, Jean E., Houghton, Andrea K., Westwood, Paul J., Walker, Glenn
Published in MedChemComm (01.07.2010)
Published in MedChemComm (01.07.2010)
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Synthesis and SAR studies of novel 2-(6-aminomethylaryl-2-aryl-4-oxo-quinazolin-3(4 H)-yl)acetamide Vasopressin V 1b receptor antagonists
Napier, Susan E., Letourneau, Jeffrey J., Ansari, Nasrin, Auld, Douglas S., Baker, James, Best, Stuart, Campbell-Wan, Leigh, Chan, Ray, Craighead, Mark, Desai, Hema, Ho, Koc-Kan, MacSweeney, Cliona, Milne, Rachel, Richard Morphy, J., Neagu, Irina, Ohlmeyer, Michael H.J., Pick, Jack, Presland, Jeremy, Riviello, Chris, Zanetakos, Heather A., Zhao, Jiuqiao, Webb, Maria L.
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
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Journal Article
Identification and optimisation of novel sulfonamide, selective vasopressin V 1B receptor antagonists
Baker, James, Bingham, Matilda, Blackburn-Munro, Ruth, Cai, Jiaqiang, Craighead, Mark, Gilfillan, Robert, Goan, Kate, Jaap, David, Milne, Rachel, Richard Morphy, J., Napier, Susan, Presland, Jeremy, Spinks, Gayle, Thomson, Fiona
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
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Synthesis of Tertiary Amines Using a Polystyrene (REM) Resin
Brown, Angus R, Rees, David C, Rankovic, Zoran, Morphy, J. Richard
Published in Journal of the American Chemical Society (09.04.1997)
Published in Journal of the American Chemical Society (09.04.1997)
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Synthesis and SAR studies of 3-phenoxypropyl piperidine analogues as ORL1 (NOP) receptor agonists
Palin, Ronald, Barn, David R., Clark, John K., Cottney, Jean E., Cowley, Phillip M., Crockatt, Marc, Evans, Louise, Feilden, Helen, Goodwin, Richard R., Griekspoor, Frank, Grove, Simon J.A., Houghton, Andrea K., Jones, Philip S., Morphy, Richard J., Smith, Alasdair R.C., Sundaram, Hardy, Vrolijk, David, Weston, Mark A., Wishart, Grant, Wren, Paul
Published in Bioorganic & medicinal chemistry letters (01.02.2005)
Published in Bioorganic & medicinal chemistry letters (01.02.2005)
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The First Potent and Selective Inhibitors of the Glycine Transporter Type 2
Caulfield, Wilson L, Collie, Iain T, Dickins, Rachel S, Epemolu, Ola, McGuire, Ross, Hill, David R, McVey, Gillian, Morphy, J. Richard, Rankovic, Zoran, Sundaram, Hardy
Published in Journal of medicinal chemistry (16.08.2001)
Published in Journal of medicinal chemistry (16.08.2001)
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