Stereo- and regiodefined DNA-encoded chemical libraries enable efficient tumour-targeting applications
Favalli, Nicholas, Bassi, Gabriele, Pellegrino, Christian, Millul, Jacopo, De Luca, Roberto, Cazzamalli, Samuele, Yang, Su, Trenner, Anika, Mozaffari, Nour L., Myburgh, Renier, Moroglu, Mustafa, Conway, Stuart J., Sartori, Alessandro A., Manz, Markus G., Lerner, Richard A., Vogt, Peter K., Scheuermann, Jörg, Neri, Dario
Published in Nature chemistry (01.06.2021)
Published in Nature chemistry (01.06.2021)
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Controlling Intramolecular Interactions in the Design of Selective, High-Affinity Ligands for the CREBBP Bromodomain
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Published in Journal of medicinal chemistry (22.07.2021)
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Publisher Correction: Stereo- and regiodefined DNA-encoded chemical libraries enable efficient tumour-targeting applications
Favalli, Nicholas, Bassi, Gabriele, Pellegrino, Christian, Millul, Jacopo, De Luca, Roberto, Cazzamalli, Samuele, Yang, Su, Trenner, Anika, Mozaffari, Nour L., Myburgh, Renier, Moroglu, Mustafa, Conway, Stuart J., Sartori, Alessandro A., Manz, Markus G., Lerner, Richard A., Vogt, Peter K., Scheuermann, Jörg, Neri, Dario
Published in Nature chemistry (01.07.2021)
Published in Nature chemistry (01.07.2021)
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A Single‐Stranded DNA‐Encoded Chemical Library Based on a Stereoisomeric Scaffold Enables Ligand Discovery by Modular Assembly of Building Blocks
Bassi, Gabriele, Favalli, Nicholas, Vuk, Miriam, Catalano, Marco, Martinelli, Adriano, Trenner, Anika, Porro, Antonio, Yang, Su, Tham, Chuin Lean, Moroglu, Mustafa, Yue, Wyatt W., Conway, Stuart J., Vogt, Peter K., Sartori, Alessandro A., Scheuermann, Jörg, Neri, Dario
Published in Advanced science (01.11.2020)
Published in Advanced science (01.11.2020)
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BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability
Jennings, Laura E., Schiedel, Matthias, Hewings, David S., Picaud, Sarah, Laurin, Corentine M.C., Bruno, Paul A., Bluck, Joseph P., Scorah, Amy R., See, Larissa, Reynolds, Jessica K., Moroglu, Mustafa, Mistry, Ishna N., Hicks, Amy, Guzanov, Pavel, Clayton, James, Evans, Charles N.G., Stazi, Giulia, Biggin, Philip C., Mapp, Anna K., Hammond, Ester M., Humphreys, Philip G., Filippakopoulos, Panagis, Conway, Stuart J.
Published in Bioorganic & medicinal chemistry (15.07.2018)
Published in Bioorganic & medicinal chemistry (15.07.2018)
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Chemical Epigenetics: The Impact of Chemical and Chemical Biology Techniques on Bromodomain Target Validation
Schiedel, Matthias, Moroglu, Mustafa, Ascough, David M. H., Chamberlain, Anna E. R., Kamps, Jos J. A. G., Sekirnik, Angelina R., Conway, Stuart J.
Published in Angewandte Chemie International Edition (09.12.2019)
Published in Angewandte Chemie International Edition (09.12.2019)
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ENT1 억제 활성을 갖는 마크로시클릭 화합물의 제조 방법
MOROGLU MUSTAFA, SHANG DEJU, HUANG XIN, LEMOINE HUGUES, TALBOT ERIC, ROCHE DIDIER, YUAN CUICUI, DELIGNY MICHAEL
Year of Publication 20.06.2024
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Year of Publication 20.06.2024
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Selective Fragments for the CREBBP Bromodomain Identified from an Encoded Self‐assembly Chemical Library
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Published in ChemMedChem (16.09.2020)
Published in ChemMedChem (16.09.2020)
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신규 화합물
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Year of Publication 19.05.2023
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Year of Publication 19.05.2023
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Chemische Epigenetik: der Einfluss chemischer und chemo‐biologischer Techniken auf die Zielstruktur‐Validierung von Bromodomänen
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Published in Angewandte Chemie (01.12.2019)
Published in Angewandte Chemie (01.12.2019)
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Chemische Epigenetik: der Einfluss chemischer und chemo‐biologischer Techniken auf die Zielstruktur‐Validierung von Bromodomänen
Schiedel, Matthias, Moroglu, Mustafa, Ascough, David M. H., Chamberlain, Anna E. R., Kamps, Jos J. A. G., Sekirnik, Angelina R., Conway, Stuart J.
Published in Angewandte Chemie (09.12.2019)
Published in Angewandte Chemie (09.12.2019)
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Year of Publication 13.04.2023
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Year of Publication 13.04.2023
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MACLEAN, John, TALBOT, Eric, MILLER, Neil, MOROGLU, Mustafa, MORPHY, Richard, ROWLEY, Michael, KULAGOWSKI, Jan, LADDUWAHETTY, Tammy, RUTTER, Richard
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Year of Publication 02.11.2023
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Year of Publication 02.11.2023
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COMPOUNDS AS PARP1 INHIBITIORS
SHEN, Zhenhai, BATEMAN, Joseph M, RAHEMTULLA, Benjamin F, MOROGLU, Mustafa, LADDUWAHETTY, Tammy, WANG, Tingzhong, TALBOT, Eric P A
Year of Publication 02.11.2023
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Year of Publication 02.11.2023
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