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Published in Bone (New York, N.Y.) (01.06.2009)
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Kumar, Rebecca N, Wu, En-Ling, Stosor, Valentina, Moore, William J, Achenbach, Chad, Ison, Michael G, Angarone, Michael P
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OMERO: flexible, model-driven data management for experimental biology
Allan, Chris, Burel, Jean-Marie, Moore, Josh, Blackburn, Colin, Linkert, Melissa, Loynton, Scott, MacDonald, Donald, Moore, William J, Neves, Carlos, Patterson, Andrew, Porter, Michael, Tarkowska, Aleksandra, Loranger, Brian, Avondo, Jerome, Lagerstedt, Ingvar, Lianas, Luca, Leo, Simone, Hands, Katherine, Hay, Ron T, Patwardhan, Ardan, Best, Christoph, Kleywegt, Gerard J, Zanetti, Gianluigi, Swedlow, Jason R
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Synthesis and Activity of Substituted 4-(Indazol-3-yl)phenols as Pathway-Selective Estrogen Receptor Ligands Useful in the Treatment of Rheumatoid Arthritis
Steffan, Robert J, Matelan, Edward, Ashwell, Mark A, Moore, William J, Solvibile, William R, Trybulski, Eugene, Chadwick, Christopher C, Chippari, Susan, Kenney, Thomas, Eckert, Amy, Borges-Marcucci, Lisa, Keith, James C, Xu, Zhang, Mosyak, Lydia, Harnish, Douglas C
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Discovery and Optimization of Potent, Cell-Active Pyrazole-Based Inhibitors of Lactate Dehydrogenase (LDH)
Rai, Ganesha, Brimacombe, Kyle R, Mott, Bryan T, Urban, Daniel J, Hu, Xin, Yang, Shyh-Ming, Lee, Tobie D, Cheff, Dorian M, Kouznetsova, Jennifer, Benavides, Gloria A, Pohida, Katie, Kuenstner, Eric J, Luci, Diane K, Lukacs, Christine M, Davies, Douglas R, Dranow, David M, Zhu, Hu, Sulikowski, Gary, Moore, William J, Stott, Gordon M, Flint, Andrew J, Hall, Matthew D, Darley-Usmar, Victor M, Neckers, Leonard M, Dang, Chi V, Waterson, Alex G, Simeonov, Anton, Jadhav, Ajit, Maloney, David J
Published in Journal of medicinal chemistry (22.11.2017)
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Discovery of Potent Myeloid Cell Leukemia‑1 (Mcl-1) Inhibitors That Demonstrate in Vivo Activity in Mouse Xenograft Models of Human Cancer
Lee, Taekyu, Christov, Plamen P, Shaw, Subrata, Tarr, James C, Zhao, Bin, Veerasamy, Nagarathanam, Jeon, Kyu Ok, Mills, Jonathan J, Bian, Zhiguo, Sensintaffar, John L, Arnold, Allison L, Fogarty, Stuart A, Perry, Evan, Ramsey, Haley E, Cook, Rebecca S, Hollingshead, Melinda, Davis Millin, Myrtle, Lee, Kyung-min, Koss, Brian, Budhraja, Amit, Opferman, Joseph T, Kim, Kwangho, Arteaga, Carlos L, Moore, William J, Olejniczak, Edward T, Savona, Michael R, Fesik, Stephen W
Published in Journal of medicinal chemistry (25.04.2019)
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Discovery of Potent Orally Bioavailable WD Repeat Domain 5 (WDR5) Inhibitors Using a Pharmacophore-Based Optimization
Teuscher, Kevin B, Meyers, Kenneth M, Wei, Qiangqiang, Mills, Jonathan J, Tian, Jianhua, Alvarado, Joseph, Sai, Jiqing, Van Meveren, Mayme, South, Taylor M, Rietz, Tyson A, Zhao, Bin, Moore, William J, Stott, Gordon M, Tansey, William P, Lee, Taekyu, Fesik, Stephen W
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Published in Clinical infectious diseases (29.01.2022)
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Structure-Based Discovery of Potent, Orally Bioavailable Benzoxazepinone-Based WD Repeat Domain 5 Inhibitors
Teuscher, Kevin B., Mills, Jonathan J., Tian, Jianhua, Han, Changho, Meyers, Kenneth M., Sai, Jiqing, South, Taylor M., Crow, Mackenzie M., Van Meveren, Mayme, Sensintaffar, John L., Zhao, Bin, Amporndanai, Kangsa, Moore, William J., Stott, Gordon M., Tansey, William P., Lee, Taekyu, Fesik, Stephen W.
Published in Journal of medicinal chemistry (28.12.2023)
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Discovery and Structure-Based Optimization of Potent and Selective WD Repeat Domain 5 (WDR5) Inhibitors Containing a Dihydroisoquinolinone Bicyclic Core
Tian, Jianhua, Teuscher, Kevin B, Aho, Erin R, Alvarado, Joseph R, Mills, Jonathan J, Meyers, Kenneth M, Gogliotti, Rocco D, Han, Changho, Macdonald, Jonathan D, Sai, Jiqing, Shaw, J. Grace, Sensintaffar, John L, Zhao, Bin, Rietz, Tyson A, Thomas, Lance R, Payne, William G, Moore, William J, Stott, Gordon M, Kondo, Jumpei, Inoue, Masahiro, Coffey, Robert J, Tansey, William P, Stauffer, Shaun R, Lee, Taekyu, Fesik, Stephen W
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Discovery of a Myeloid Cell Leukemia 1 (Mcl-1) Inhibitor That Demonstrates Potent In Vivo Activities in Mouse Models of Hematological and Solid Tumors
Tarr, James C., Salovich, James M., Aichinger, Martin, Jeon, KyuOk, Veerasamy, Nagarathanam, Sensintaffar, John L., Arnhof, Heribert, Samwer, Matthias, Christov, Plamen P., Kim, Kwangho, Wunberg, Tobias, Schweifer, Norbert, Trapani, Francesca, Arnold, Allison, Martin, Florian, Zhao, Bin, Miriyala, Nagaraju, Sgubin, Danielle, Fogarty, Stuart, Moore, William J., Stott, Gordon M., Olejniczak, Edward T., Engelhardt, Harald, Rudolph, Dorothea, Lee, Taekyu, McConnell, Darryl B., Fesik, Stephen W.
Published in Journal of medicinal chemistry (05.08.2024)
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Structure-based discovery of potent WD repeat domain 5 inhibitors that demonstrate efficacy and safety in preclinical animal models
Teuscher, Kevin B, Chowdhury, Somenath, Meyers, Kenneth M, Tian, Jianhua, Sai, Jiqing, Van Meveren, Mayme, South, Taylor M, Sensintaffar, John L, Rietz, Tyson A, Goswami, Soumita, Wang, Jing, Grieb, Brian C, Lorey, Shelly L, Howard, Gregory C, Liu, Qi, Moore, William J, Stott, Gordon M, Tansey, William P, Lee, Taekyu, Fesik, Stephen W
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Rohde, Jason M, Karavadhi, Surendra, Pragani, Rajan, Liu, Li, Fang, Yuhong, Zhang, Weihe, McIver, Andrew, Zheng, Hongchao, Liu, Qingyang, Davis, Mindy I, Urban, Daniel J, Lee, Tobie D, Cheff, Dorian M, Hollingshead, Melinda, Henderson, Mark J, Martinez, Natalia J, Brimacombe, Kyle R, Yasgar, Adam, Zhao, Wei, Klumpp-Thomas, Carleen, Michael, Sam, Covey, Joseph, Moore, William J, Stott, Gordon M, Li, Zhuyin, Simeonov, Anton, Jadhav, Ajit, Frye, Stephen, Hall, Matthew D, Shen, Min, Wang, Xiaodong, Patnaik, Samarjit, Boxer, Matthew B
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O'Donoghue, Seán I, Baldi, Benedetta Frida, Clark, Susan J, Darling, Aaron E, Hogan, James M, Kaur, Sandeep, Maier-Hein, Lena, McCarthy, Davis J, Moore, William J, Stenau, Esther, Swedlow, Jason R, Vuong, Jenny, Procter, James B
Published in Annual review of biomedical data science (20.07.2018)
Published in Annual review of biomedical data science (20.07.2018)
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Discovery and Optimization of 2 H -1λ 2 -Pyridin-2-one Inhibitors of Mutant Isocitrate Dehydrogenase 1 for the Treatment of Cancer
Rohde, Jason M, Karavadhi, Surendra, Pragani, Rajan, Liu, Li, Fang, Yuhong, Zhang, Weihe, McIver, Andrew, Zheng, Hongchao, Liu, Qingyang, Davis, Mindy I, Urban, Daniel J, Lee, Tobie D, Cheff, Dorian M, Hollingshead, Melinda, Henderson, Mark J, Martinez, Natalia J, Brimacombe, Kyle R, Yasgar, Adam, Zhao, Wei, Klumpp-Thomas, Carleen, Michael, Sam, Covey, Joseph, Moore, William J, Stott, Gordon M, Li, Zhuyin, Simeonov, Anton, Jadhav, Ajit, Frye, Stephen, Hall, Matthew D, Shen, Min, Wang, Xiaodong, Patnaik, Samarjit, Boxer, Matthew B
Published in Journal of medicinal chemistry (22.04.2021)
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Metadata management for high content screening in OMERO
Li, Simon, Besson, Sébastien, Blackburn, Colin, Carroll, Mark, Ferguson, Richard K., Flynn, Helen, Gillen, Kenneth, Leigh, Roger, Lindner, Dominik, Linkert, Melissa, Moore, William J., Ramalingam, Balaji, Rozbicki, Emil, Rustici, Gabriella, Tarkowska, Aleksandra, Walczysko, Petr, Williams, Eleanor, Allan, Chris, Burel, Jean-Marie, Moore, Josh, Swedlow, Jason R.
Published in Methods (San Diego, Calif.) (01.03.2016)
Published in Methods (San Diego, Calif.) (01.03.2016)
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Mitotic mechanics: the auroras come into view
Andrews, Paul D, Knatko, Elena, Moore, William J, Swedlow, Jason R
Published in Current opinion in cell biology (01.12.2003)
Published in Current opinion in cell biology (01.12.2003)
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Optimization of ether and aniline based inhibitors of lactate dehydrogenase
Christov, Plamen P., Kim, Kwangho, Jana, Somnath, Romaine, Ian M., Rai, Ganesha, Mott, Bryan T., Allweil, Alexander A., Lamers, Alexander, Brimacombe, Kyle R., Urban, Daniel J., Lee, Tobie D., Hu, Xin, Lukacs, Christine M., Davies, Douglas R., Jadhav, Ajit, Hall, Matthew D., Green, Neal, Moore, William J., Stott, Gordon M., Flint, Andrew J., Maloney, David J., Sulikowski, Gary A., Waterson, Alex G.
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
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