Phenobarbital indirectly activates the constitutive active androstane receptor (CAR) by inhibition of epidermal growth factor receptor signaling
Mutoh, Shingo, Sobhany, Mack, Moore, Rick, Perera, Lalith, Pedersen, Lee, Sueyoshi, Tatsuya, Negishi, Masahiko
Published in Science signaling (07.05.2013)
Published in Science signaling (07.05.2013)
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CAR requires Gadd45β to promote phenobarbital-induced mouse liver tumors in early stage
Hori, Takeshi, Yokobori, Kosuke, Moore, Rick, Negishi, Masahiko, Sueyoshi, Tatsuya
Published in Frontiers in oncology (07.09.2023)
Published in Frontiers in oncology (07.09.2023)
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The roles of co-chaperone CCRP/DNAJC7 in Cyp2b10 gene activation and steatosis development in mouse livers
Ohno, Marumi, Kanayama, Tomohiko, Moore, Rick, Ray, Manas, Negishi, Masahiko
Published in PloS one (26.12.2014)
Published in PloS one (26.12.2014)
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Dephosphorylation of Threonine 38 Is Required for Nuclear Translocation and Activation of Human Xenobiotic Receptor CAR (NR1I3)
Mutoh, Shingo, Osabe, Makoto, Inoue, Kaoru, Moore, Rick, Pedersen, Lee, Perera, Lalith, Rebolloso, Yvette, Sueyoshi, Tatsuya, Negishi, Masahiko
Published in The Journal of biological chemistry (11.12.2009)
Published in The Journal of biological chemistry (11.12.2009)
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Relative Activation of Human Pregnane X Receptor versus Constitutive Androstane Receptor Defines Distinct Classes of CYP2B6 and CYP3A4 Inducers
Faucette, Stephanie R, Zhang, Tong-Cun, Moore, Rick, Sueyoshi, Tatsuya, Omiecinski, Curtis J, LeCluyse, Edward L, Negishi, Masahiko, Wang, Hongbing
Published in The Journal of pharmacology and experimental therapeutics (01.01.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2007)
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Flame retardant BDE-47 effectively activates nuclear receptor CAR in human primary hepatocytes
Sueyoshi, Tatsuya, Li, Linhao, Wang, Hongbing, Moore, Rick, Kodavanti, Prasada Rao S, Lehmler, Hans-Joachim, Negishi, Masahiko, Birnbaum, Linda S
Published in Toxicological sciences (01.02.2014)
Published in Toxicological sciences (01.02.2014)
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The orphan nuclear receptor constitutive active/androstane receptor is essential for liver tumor promotion by phenobarbital in mice
YAMAMOTO, Yukio, MOORE, Rick, GOLDSWORTHY, Thomas L, NEGISHI, Masahiko, MARONPOT, Robert R
Published in Cancer research (Chicago, Ill.) (15.10.2004)
Published in Cancer research (Chicago, Ill.) (15.10.2004)
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Estrogen receptor α phosphorylated at Ser216 confers inflammatory function to mouse microglia
Shindo, Sawako, Chen, Shih-Heng, Gotoh, Saki, Yokobori, Kosuke, Hu, Hao, Ray, Manas, Moore, Rick, Nagata, Kiyoshi, Martinez, Jennifer, Hong, Jau-Shyong, Negishi, Masahiko
Published in Cell communication and signaling (29.07.2020)
Published in Cell communication and signaling (29.07.2020)
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