Enrichment Analysis for Discovering Biological Associations in Phenotypic Screens
Polyakov, Valery R, Moorcroft, Neil D, Drawid, Amar
Published in Journal of chemical information and modeling (24.02.2014)
Published in Journal of chemical information and modeling (24.02.2014)
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Design and synthesis of D1 agonist/D2 antagonist for treatment of schizophrenia
Giovanni, Andrew, Roehr, Joachim, Dwyer, Shannon, Neuenschwander, Kent, Scotese, Anthony, Moorcroft, Neil D., Davis, Larry, Gao, Zhongli
Published in Bioorganic & medicinal chemistry letters (01.03.2013)
Published in Bioorganic & medicinal chemistry letters (01.03.2013)
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Discovery of N-substituted 7-azaindoles as PIM1 kinase inhibitors – Part I
Barberis, Claude, Moorcroft, Neil, Arendt, Chris, Levit, Mikhail, Moreno-Mazza, Sandra, Batchelor, Joseph, Mechin, Ingrid, Majid, Tahir
Published in Bioorganic & medicinal chemistry letters (15.10.2017)
Published in Bioorganic & medicinal chemistry letters (15.10.2017)
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Discovery of N-substituted 7-azaindoles as Pan-PIM kinase inhibitors – Lead series identification – Part II
Barberis, Claude, Moorcroft, Neil, Pribish, James, Tserlin, Elina, Gross, Alexandre, Czekaj, Mark, Barrague, Matthieu, Erdman, Paul, Majid, Tahir, Batchelor, Joseph, Levit, Mikhail, Hebert, Andrew, Shen, Liduo, Moreno-Mazza, Sandra, Wang, Anlai
Published in Bioorganic & medicinal chemistry letters (15.10.2017)
Published in Bioorganic & medicinal chemistry letters (15.10.2017)
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Design and synthesis of D-1 agonist/D-2 antagonist for treatment of schizophrenia
Giovanni, Andrew, Roehr, Joachim, Dwyer, Shannon, Neuenschwander, Kent, Scotese, Anthony, Moorcroft, Neil D., Davis, Larry, Gao, Zhongli
Published in Bioorganic & medicinal chemistry letters (01.03.2013)
Published in Bioorganic & medicinal chemistry letters (01.03.2013)
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Mapping the kinase domain of janus kinase 3
Adams, Christopher, Aldous, David J., Amendola, Shelley, Bamborough, Paul, Bright, Colin, Crowe, Sarah, Eastwood, Paul, Fenton, Garry, Foster, Martyn, Harrison, Trevor K.P., King, Sue, Lai, Justine, Lawrence, Christopher, Letallec, Jean-Philippe, McCarthy, Clive, Moorcroft, Neil, Page, Kenneth, Rao, Sudha, Redford, Jane, Sadiq, Shazia, Smith, Keith, Souness, John E., Thurairatnam, Sukanthini, Vine, Mark, Wyman, Barry
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
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Journal Article
Mapping the kinase domain of Janus Kinase 3: Recent advances in the design of kinase inhibitors as novel therapeutic agents
ADAMS, Christopher, ALDOUS, David J, KING, Sue, LAI, Justine, LAWRENCE, Christopher, LETALLEC, Jean-Philippe, MCCARTHY, Clive, MOORCROFT, Neil, PAGE, Kenneth, RAO, Sudha, REDFORD, Jane, SADIQ, Shazia, AMENDOLA, Shelley, SMITH, Keith, SOUNESS, John E, THURAIRATNAM, Sukanthini, VINE, Mark, WYMAN, Barry, BAMBOROUGH, Paul, BRIGHT, Colin, CROWE, Sarah, EASTWOOD, Paul, FENTON, Garry, FOSTER, Martyn, HARRISON, Trevor K. P
Published in Bioorganic & medicinal chemistry letters (2003)
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Published in Bioorganic & medicinal chemistry letters (2003)
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derivados de azacarbolinas, a respectiva preparação e sua utilização terapêutica
Didier Babin, Ronghua Li, David Papin, Neil Moorcroft, Olivier Bedel, Serge Mignani, Thierry Gouyon, Mikhail Levit, Christopher Arendt
Year of Publication 15.01.2019
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Year of Publication 15.01.2019
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SUBSTITUTED PYRIDONES AS INHIBITORS OF POLY(ADP-RIBOSE) POLYMERASE (PARP)
MOORCROFT, NEIL, JIANG, JOHN, Z, EASTWOOD, PAUL, R, SCHWAHN, UWE, RUTTEN, HARTMUT, WEINTRAUB, PHILIP, M, MEHDI, SHUJAATH, STEFANY, DAVID, W, PEUKERT, STEFAN, MUSICK, KWON, YON, LIM, SUNGTAEK
Year of Publication 12.12.2012
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Year of Publication 12.12.2012
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AZACARBOLINE DERIVATIVES, PREPARATION METHOD THEREOF AND THERAPEUTIC USE OF SAME
ARENDT CHRISTOPHER, BEDEL OLIVIER, GOUYON THIERRY, LEVIT MIKHAIL, LI RONGHUA, MOORCROFT NEIL, PAPIN DAVID, BABIN DIDIER, MIGNANI SERGE
Year of Publication 21.07.2011
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Year of Publication 21.07.2011
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TETRAHYDROCARBOLINE DERIVATIVES AS EG5 INHIBITORS
MOORCROFT, NEIL DAVID, LI, RONGHUA, ZILBERSTEIN, ASHER, GROSS, ALEXANDRE, YU, KIN T, MAJID, TAHIR NADEEM
Year of Publication 14.07.2011
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Year of Publication 14.07.2011
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SUBSTITUTED PYRIDONES AS INHIBITORS OF POLY(ADP-RIBOSE) POLYMERASE (PARP)
JIANG JOHN Z, LIM SUNGTAEK, MUSICK KWON YON, MOORCROFT NEIL, PEUKERT STEFAN, STEFANY DAVID W, RUTTEN HARTMUT, SCHWAHN UWE, EASTWOOD PAUL R, MEHDI SHUJAATH, WEINTRAUB PHILIP M
Year of Publication 09.08.2012
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Year of Publication 09.08.2012
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