Recombinant irisin induces weight loss in high fat DIO mice through increase in energy consumption and thermogenesis
Niranjan, Sanjay B., Belwalkar, Shraddha Vijay, Tambe, Suhas, Venkataraman, Krishnan, Mookhtiar, Kasim A.
Published in Biochemical and biophysical research communications (05.11.2019)
Published in Biochemical and biophysical research communications (05.11.2019)
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Journal Article
Regulation of RIPK1 activation by TAK1-mediated phosphorylation dictates apoptosis and necroptosis
Geng, Jiefei, Ito, Yasushi, Shi, Linyu, Amin, Palak, Chu, Jiachen, Ouchida, Amanda Tomie, Mookhtiar, Adnan Kasim, Zhao, Heng, Xu, Daichao, Shan, Bing, Najafov, Ayaz, Gao, Guangping, Akira, Shizuo, Yuan, Junying
Published in Nature communications (25.08.2017)
Published in Nature communications (25.08.2017)
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Journal Article
RIPK1 mediates axonal degeneration by promoting inflammation and necroptosis in ALS
Ito, Yasushi, Ofengeim, Dimitry, Najafov, Ayaz, Das, Sudeshna, Saberi, Shahram, Li, Ying, Hitomi, Junichi, Zhu, Hong, Chen, Hongbo, Mayo, Lior, Geng, Jiefei, Amin, Palak, DeWitt, Judy Park, Mookhtiar, Adnan Kasim, Florez, Marcus, Ouchida, Amanda Tomie, Fan, Jian-bing, Pasparakis, Manolis, Kelliher, Michelle A., Ravits, John, Yuan, Junying
Published in Science (American Association for the Advancement of Science) (05.08.2016)
Published in Science (American Association for the Advancement of Science) (05.08.2016)
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Journal Article
Design and synthesis of novel xanthine derivatives as potent and selective A2B adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases
Basu, Sujay, Barawkar, Dinesh A., Ramdas, Vidya, Patel, Meena, Waman, Yogesh, Panmand, Anil, Kumar, Santosh, Thorat, Sachin, Naykodi, Minakshi, Goswami, Arnab, Reddy, B. Srinivasa, Prasad, Vandna, Chaturvedi, Sandhya, Quraishi, Azfar, Menon, Suraj, Paliwal, Shalini, Kulkarni, Abhay, Karande, Vikas, Ghosh, Indraneel, Mustafa, Syed, De, Siddhartha, Jain, Vaibhav, Banerjee, Ena Ray, Rouduri, Sreekanth R., Palle, Venkata P., Chugh, Anita, Mookhtiar, Kasim A.
Published in European journal of medicinal chemistry (07.07.2017)
Published in European journal of medicinal chemistry (07.07.2017)
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Journal Article
Discovery and evaluation of novel FAAH inhibitors in neuropathic pain model
Bhuniya, Debnath, Kharul, Rajendra K., Hajare, Atul, Shaikh, Nadim, Bhosale, Sandeep, Balwe, Sandip, Begum, Fouzia, De, Siddhartha, Athavankar, Sonalee, Joshi, Dhananjay, Madgula, Vamsi, Joshi, Kaushal, Raje, Amol A., Meru, Ashwinkumar V., Magdum, Amol, Mookhtiar, Kasim A., Barbhaiya, Rashmi
Published in Bioorganic & medicinal chemistry letters (15.01.2019)
Published in Bioorganic & medicinal chemistry letters (15.01.2019)
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Journal Article
Discovery and pharmacological evaluation of indole derivatives as potent and selective RORγt inverse agonist for multiple autoimmune conditions
Shaikh, Nadim S., Iyer, Jitesh P., Munot, Yogesh S., Mukhopadhyay, Partha P., Raje, Amol A., Nagaraj, Ranganayaki, Jamdar, Vijay, Gavhane, Ravindra, Lohote, Mahendra, Sherkar, Prasad, Bala, Madhu, Petla, Rajkanth, Meru, Ashwinkumar, Umrani, Dhananjay, Rouduri, Sreekanth, Joshi, Sachin, Reddy, Satyanarayan, Kandikere, Vishwottam, Bhuniya, Debnath, Kulkarni, Bheemashankar, Mookhtiar, Kasim A.
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
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Journal Article
Modifications of flexible nonyl chain and nucleobase head group of (+)-erythro-9-(2′s-hydroxy-3′s-nonyl)adenine [(+)-EHNA] as adenosine deaminase inhibitors
Kandalkar, Sachin R., Ramaiah, Parimi Atchuta, Joshi, Manoj, Wavhal, Atul, Waman, Yogesh, Raje, Amol A., Tambe, Ashwini, Ansari, Shariq, De, Siddhartha, Palle, Venkata P., Mookhtiar, Kasim A., Deshpande, Anil M., Barawkar, Dinesh A.
Published in Bioorganic & medicinal chemistry (15.10.2017)
Published in Bioorganic & medicinal chemistry (15.10.2017)
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Journal Article
Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A2A Receptor Antagonists and Their Biological Evaluation
Basu, Sujay, Barawkar, Dinesh A, Thorat, Sachin, Shejul, Yogesh D, Patel, Meena, Naykodi, Minakshi, Jain, Vaibhav, Salve, Yogesh, Prasad, Vandna, Chaudhary, Sumit, Ghosh, Indraneel, Bhat, Ganesh, Quraishi, Azfar, Patil, Harish, Ansari, Shariq, Menon, Suraj, Unadkat, Vishal, Thakare, Rhishikesh, Seervi, Madhav S, Meru, Ashwinkumar V, De, Siddhartha, Bhamidipati, Ravi K, Rouduri, Sreekanth R, Palle, Venkata P, Chug, Anita, Mookhtiar, Kasim A
Published in Journal of medicinal chemistry (26.01.2017)
Published in Journal of medicinal chemistry (26.01.2017)
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Journal Article
257 Combination of adenosine antagonists A2AR (TT-10) and A2BR (TT-4) with checkpoint inhibitors demonstrate anti-tumor activity in CT-26 murine colon tumor allograft model
Pastore, Desa Rae, Kumar, Sushant, Schwartz, Brian, Mookhtiar, Kasim, Reddy, Vijay
Published in Journal for immunotherapy of cancer (01.11.2021)
Published in Journal for immunotherapy of cancer (01.11.2021)
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Journal Article
Discovery of a potent and selective small molecule hGPR91 antagonist
Bhuniya, Debnath, Umrani, Dhananjay, Dave, Bhavesh, Salunke, Deepak, Kukreja, Gagan, Gundu, Jayasagar, Naykodi, Minakshi, Shaikh, Nadim S., Shitole, Prasad, Kurhade, Santosh, De, Siddhartha, Majumdar, Sreemita, Reddy, Srinivasa B., Tambe, Suhas, Shejul, Yogesh, Chugh, Anita, Palle, Venkata P., Mookhtiar, Kasim A., Cully, Doris, Vacca, Joseph, Chakravarty, Prasun K., Nargund, Ravi P., Wright, Samuel D., Graziano, Michael P., Singh, Sheo B., Roy, Sophie, Cai, Tian-Quan
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
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Journal Article
Evaluation of separate role of intestine and liver in first pass metabolism of budesonide in rat
Raje, Amol A., Deshpande, Radni D., Pathade, Vishal V., Mahajan, Vallabh, Joshi, Kaushal, Tambe, Ashwini, Jinugu, Ramana, Madgula, Vamsi L. M., Gaur, Ashwani, Kandikere, Vishwottam, Patil, Chandragouda R., Mookhtiar, Kasim A.
Published in Xenobiotica (02.12.2018)
Published in Xenobiotica (02.12.2018)
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Journal Article
Discovery of liver-directed glucokinase activator having anti-hyperglycemic effect without hypoglycemia
Deshpande, Anil M., Bhuniya, Debnath, De, Siddhartha, Dave, Bhavesh, Vyavahare, Vinod P., Kurhade, Santosh H., Kandalkar, Sachin R., Naik, Keshav P., Kobal, Balasaheb S., Kaduskar, Rahul D., Basu, Sujay, Jain, Vaibhav, Patil, Pratima, Chaturvedi Joshi, Sandhya, Bhat, Ganesh, Raje, Amol A., Reddy, Satyanarayana, Gundu, Jayasagar, Madgula, Vamsi, Tambe, Suhas, Shitole, Prasad, Umrani, Dhananjay, Chugh, Anita, Palle, Venkata P., Mookhtiar, Kasim A.
Published in European journal of medicinal chemistry (16.06.2017)
Published in European journal of medicinal chemistry (16.06.2017)
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Journal Article
Discovery and evaluation of 1H-pyrrolo[2,3-b]pyridine based selective and reversible small molecule BTK inhibitors for the treatment of rheumatoid arthritis
Thakkar, Mahesh, Bhuniya, Debnath, Kaduskar, Rahul, Mengawade, Tanaji, Naik, Keshav, Salunkhe, Videsh, Bhalerao, Amit, Kurhade, Santosh, Mavinahalli, Jagadeesh, Jain, Vaibhav, Petla, Rajkanth, Avaragolla, Satheesh, Ray, Swagatam, Rouduri, Sreekanth, Dhanave, Avinash, De, Siddhartha, Pathade, Vishal, Tambe, Ashwini, Raje, Amol A., Madgula, Vamsi, Joshi, Sachin, Nadeem, Ahmed, bala, Madhu, Umrani, Dhananjay, Hariharan, Narayanan, Kulkarni, Bheemashankar, Mookhtiar, Kasim A.
Published in Bioorganic & medicinal chemistry letters (15.04.2017)
Published in Bioorganic & medicinal chemistry letters (15.04.2017)
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Journal Article
759 ADPORT-601 (TT-10–101): first-in-human study of adenosine 2A (A2A) and adenosine 2B (A2B) receptor antagonists in participants with selected advanced solid tumors
Subudhi, Sumit, Falchook, Gerald S, Salkeni, Mohamad A, El-Khoueiry, Anthony, Grewal, Jaspreet, Tester, William, Pachynski, Russell, Upadhaya, Samik, Saez Ibanez, Ana Rosa, Kumar, Sushant, Mookhtiar, Kasim, Stanton-Pastore, Desa Rae, Kramer, Robert, Fairchild, Justin, Walters, Ian, Fong, Lawrence
Published in Journal for immunotherapy of cancer (01.11.2023)
Published in Journal for immunotherapy of cancer (01.11.2023)
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Journal Article
Pharmacological and X-Ray Structural Characterization of a Novel Selective Androgen Receptor Modulator: Potent Hyperanabolic Stimulation of Skeletal Muscle with Hypostimulation of Prostate in Rats
Ostrowski, Jacek, Kuhns, Joyce E, Lupisella, John A, Manfredi, Mark C, Beehler, Blake C, Krystek, Stanley R, Bi, Yingzhi, Sun, Chongqing, Seethala, Ramakrishna, Golla, Rajasree, Sleph, Paul G, Fura, Aberra, An, Yongmi, Kish, Kevin F, Sack, John S, Mookhtiar, Kasim A, Grover, Gary J, Hamann, Lawrence G
Published in Endocrinology (Philadelphia) (01.01.2007)
Published in Endocrinology (Philadelphia) (01.01.2007)
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Journal Article
Design and synthesis of novel xanthine derivatives as potent and selective A 2B adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases
Basu, Sujay, Barawkar, Dinesh A, Ramdas, Vidya, Patel, Meena, Waman, Yogesh, Panmand, Anil, Kumar, Santosh, Thorat, Sachin, Naykodi, Minakshi, Goswami, Arnab, Reddy, B Srinivasa, Prasad, Vandna, Chaturvedi, Sandhya, Quraishi, Azfar, Menon, Suraj, Paliwal, Shalini, Kulkarni, Abhay, Karande, Vikas, Ghosh, Indraneel, Mustafa, Syed, De, Siddhartha, Jain, Vaibhav, Banerjee, Ena Ray, Rouduri, Sreekanth R, Palle, Venkata P, Chugh, Anita, Mookhtiar, Kasim A
Published in European journal of medicinal chemistry (07.07.2017)
Published in European journal of medicinal chemistry (07.07.2017)
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Journal Article
Design and synthesis of novel, potent and selective hypoxanthine analogs as adenosine A 1 receptor antagonists and their biological evaluation
Koul, Summon, Ramdas, Vidya, Barawkar, Dinesh A, Waman, Yogesh B, Prasad, Neela, Madadi, Santosh Kumar, Shejul, Yogesh D, Bonagiri, Rajesh, Basu, Sujay, Menon, Suraj, Reddy, Srinivasa B, Chaturvedi, Sandhya, Chennamaneni, Srinivas Rao, Bedse, Gaurav, Thakare, Rhishikesh, Gundu, Jayasagar, Chaudhary, Sumit, De, Siddhartha, Meru, Ashwinkumar V, Palle, Venkata, Chugh, Anita, Mookhtiar, Kasim A
Published in Bioorganic & medicinal chemistry (15.03.2017)
Published in Bioorganic & medicinal chemistry (15.03.2017)
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Journal Article
Design and synthesis of novel, potent and selective hypoxanthine analogs as adenosine A1 receptor antagonists and their biological evaluation
Koul, Summon, Ramdas, Vidya, Barawkar, Dinesh A., Waman, Yogesh B., Prasad, Neela, Madadi, Santosh Kumar, Shejul, Yogesh D., Bonagiri, Rajesh, Basu, Sujay, Menon, Suraj, Reddy, Srinivasa B., Chaturvedi, Sandhya, Chennamaneni, Srinivas Rao, Bedse, Gaurav, Thakare, Rhishikesh, Gundu, Jayasagar, Chaudhary, Sumit, De, Siddhartha, Meru, Ashwinkumar V., Palle, Venkata, Chugh, Anita, Mookhtiar, Kasim A.
Published in Bioorganic & medicinal chemistry (15.03.2017)
Published in Bioorganic & medicinal chemistry (15.03.2017)
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Journal Article
Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A 2A Receptor Antagonists and Their Biological Evaluation
Basu, Sujay, Barawkar, Dinesh A, Thorat, Sachin, Shejul, Yogesh D, Patel, Meena, Naykodi, Minakshi, Jain, Vaibhav, Salve, Yogesh, Prasad, Vandna, Chaudhary, Sumit, Ghosh, Indraneel, Bhat, Ganesh, Quraishi, Azfar, Patil, Harish, Ansari, Shariq, Menon, Suraj, Unadkat, Vishal, Thakare, Rhishikesh, Seervi, Madhav S, Meru, Ashwinkumar V, De, Siddhartha, Bhamidipati, Ravi K, Rouduri, Sreekanth R, Palle, Venkata P, Chug, Anita, Mookhtiar, Kasim A
Published in Journal of medicinal chemistry (26.01.2017)
Published in Journal of medicinal chemistry (26.01.2017)
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Journal Article
A 2B adenosine receptor antagonists: Design, synthesis and biological evaluation of novel xanthine derivatives
Basu, Sujay, Barawkar, Dinesh A, Ramdas, Vidya, Waman, Yogesh, Patel, Meena, Panmand, Anil, Kumar, Santosh, Thorat, Sachin, Bonagiri, Rajesh, Jadhav, Dilip, Mukhopadhyay, Partha, Prasad, Vandna, Reddy, B Srinivasa, Goswami, Arnab, Chaturvedi, Sandhya, Menon, Suraj, Quraishi, Azfar, Ghosh, Indraneel, Dusange, Sushant, Paliwal, Shalini, Kulkarni, Abhay, Karande, Vikas, Thakre, Rhishikesh, Bedse, Gaurav, Rouduri, Sreekanth, Gundu, Jayasagar, Palle, Venkata P, Chugh, Anita, Mookhtiar, Kasim A
Published in European journal of medicinal chemistry (15.02.2017)
Published in European journal of medicinal chemistry (15.02.2017)
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Journal Article