BCX-1812 (RWJ-270201): Discovery of a Novel, Highly Potent, Orally Active, and Selective Influenza Neuraminidase Inhibitor through Structure-Based Drug Design
Babu, Y. Sudhakar, Chand, Pooran, Bantia, Shanta, Kotian, Pravin, Dehghani, Ali, El-Kattan, Yahya, Lin, Tsu-Hsing, Hutchison, Tracy L, Elliott, Arthur J, Parker, Cynthia D, Ananth, Sandya L, Horn, LaShun L, Laver, Graeme W, Montgomery, John A
Published in Journal of medicinal chemistry (21.09.2000)
Published in Journal of medicinal chemistry (21.09.2000)
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Systematic Structure-Based Design and Stereoselective Synthesis of Novel Multisubstituted Cyclopentane Derivatives with Potent Antiinfluenza Activity
Chand, Pooran, Kotian, Pravin L, Dehghani, Ali, El-Kattan, Yahya, Lin, Tsu-Hsing, Hutchison, Tracy L, Babu, Y. Sudhakar, Bantia, Shanta, Elliott, Arthur J, Montgomery, John A
Published in Journal of medicinal chemistry (06.12.2001)
Published in Journal of medicinal chemistry (06.12.2001)
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Journal Article
Pseudoketogenesis in hepatectomized dogs
Des Rosiers, C, Montgomery, J A, Garneau, M, David, F, Mamer, O A, Daloze, P, Toffolo, G, Cobelli, C, Landau, B R, Brunengraber, H
Published in The American journal of physiology (01.03.1990)
Published in The American journal of physiology (01.03.1990)
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Comparison of the Anti-Influenza Virus Activity of RWJ-270201 with Those of Oseltamivir and Zanamivir
BANTIA, S, PARKER, C. D, HUTCHISON, T. L, MONTGOMERY, J. A, KELLOG, D. L, BABU, Y. S, ANANTH, S. L, HORN, L. L, ANDRIES, K, CHAND, P, KOTIAN, P. L, DEHGHANI, A, EL-KATTAN, Y, LIN, T
Published in Antimicrobial Agents and Chemotherapy (01.04.2001)
Published in Antimicrobial Agents and Chemotherapy (01.04.2001)
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Increased brain serotonin turnover correlates with the degree of shunting and hyperammonemia in rats following variable portal vein stenosis
Lozeva, Violina, Montgomery, Jane A, Tuomisto, Leena, Rocheleau, Bernard, Pannunzio, Marc, Huet, Pierre-Michel, Butterworth, Roger F
Published in Journal of hepatology (01.05.2004)
Published in Journal of hepatology (01.05.2004)
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Purine nucleoside phosphorylase inhibitor BCX-1777 (Immucillin-H)—a novel potent and orally active immunosuppressive agent
Bantia, Shanta, Miller, Patrick J, Parker, Cynthia D, Ananth, Sandya L, Horn, LaShun L, Kilpatrick, John M, Morris, Philip E, Hutchison, Tracy L, Montgomery, John A, Sandhu, Jasbir S
Published in International immunopharmacology (01.06.2001)
Published in International immunopharmacology (01.06.2001)
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Journal Article
Comparison of the Mechanism of Cytotoxicity of 2-Chloro-9-(2-deoxy-2-fluoro-β-d-arabinofuranosyl)adenine, 2-Chloro-9-(2-deoxy-2-fluoro-β-d-ribofuranosyl)adenine, and 2-Chloro-9-(2-deoxy-2,2-difluoro-β-d-ribofuranosyl)adenine in CEM Cells
Parker, W B, Shaddix, S C, Rose, L M, Shewach, D S, Hertel, L W, Secrist, 3rd, J A, Montgomery, J A, Bennett, Jr, L L
Published in Molecular pharmacology (01.03.1999)
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Published in Molecular pharmacology (01.03.1999)
Journal Article
Enhancement of Nucleoside Cytotoxicity through Nucleotide Prodrugs
Rose, Jerry D, Parker, William B, Someya, Hitoshi, Shaddix, Sue C, Montgomery, John A, Secrist, John A
Published in Journal of medicinal chemistry (26.09.2002)
Published in Journal of medicinal chemistry (26.09.2002)
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Journal Article
Potent Inhibition of Influenza Sialidase by a Benzoic Acid Containing a 2-Pyrrolidinone Substituent
Atigadda, Venkatram R, Brouillette, Wayne J, Duarte, Franco, Ali, Shoukath M, Babu, Yarlagadda S, Bantia, Shanta, Chand, Pooran, Chu, Naiming, Montgomery, John A, Walsh, David A, Sudbeck, Elise A, Finley, James, Luo, Ming, Air, Gillian M, Laver, Graeme W
Published in Journal of medicinal chemistry (01.07.1999)
Published in Journal of medicinal chemistry (01.07.1999)
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Journal Article
Design and Synthesis of Benzoic Acid Derivatives as Influenza Neuraminidase Inhibitors Using Structure-Based Drug Design
Chand, Pooran, Babu, Yarlagadda S, Bantia, Shanta, Chu, Naiming, Cole, L. Brent, Kotian, Pravin L, Laver, W. Graeme, Montgomery, John A, Pathak, Ved P, Petty, Sandra L, Shrout, David P, Walsh, David A, Walsh, Gerald M
Published in Journal of medicinal chemistry (05.12.1997)
Published in Journal of medicinal chemistry (05.12.1997)
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Journal Article
In vivo gene therapy of cancer with E. coli purine nucleoside phosphorylase
Parker, W B, King, S A, Allan, P W, Bennett, Jr, L L, Secrist, 3rd, J A, Montgomery, J A, Gilbert, K S, Waud, W R, Wells, A H, Gillespie, G Y, Sorscher, E J
Published in Human gene therapy (20.09.1997)
Published in Human gene therapy (20.09.1997)
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An overlap criterion for selection of core orbitals
Austin, Amy J., Frisch, Michael J., Montgomery, John A., Petersson, George A.
Published in Theoretical chemistry accounts (01.03.2002)
Published in Theoretical chemistry accounts (01.03.2002)
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Journal Article
Synthesis and biological activity of 4 '-thio-1-xylofuranosyl purine nucleosides
Tiwari, KN, Messini, L, Montgomery, JA, Secrist, JA
Published in Nucleosides, nucleotides & nucleic acids (01.01.2005)
Published in Nucleosides, nucleotides & nucleic acids (01.01.2005)
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Synthesis and biological activity of 2'-deoxy-4'-thio pyrimidine nucleosides
Secrist, John A, Tiwari, Kamal N, Riordan, James M, Montgomery, John A
Published in Journal of medicinal chemistry (01.08.1991)
Published in Journal of medicinal chemistry (01.08.1991)
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Journal Article
Hydrophobic benzoic acids as inhibitors of influenza neuraminidase
Atigadda, Venkatram R., Brouillette, Wayne J., Duarte, Franco, Babu, Yarlagadda S., Bantia, Shanta, Chand, Pooran, Chu, Naiming, Montgomery, John A., Walsh, David A., Sudbeck, Elise, Finley, James, Air, Gillian M., Luo, Ming, Laver, Graeme W.
Published in Bioorganic & medicinal chemistry (01.11.1999)
Published in Bioorganic & medicinal chemistry (01.11.1999)
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Journal Article
Structure-based design of inhibitors of purine nucleoside phosphorylase. 1. 9-(Arylmethyl) derivatives of 9-deazaguanine
Montgomery, John A., Niwas, Shri, Rose, Jerry D., Secrist, John A., Babu, Y. Sudhakar, Bugg, Charles E., Erion, Mark D., Guida, Wayne C., Ealick, Steven E.
Published in Journal of medicinal chemistry (1993)
Published in Journal of medicinal chemistry (1993)
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