Discovery of 2‑(((1r,4r)‑4-(((4-Chlorophenyl)(phenyl)carbamoyl)oxy)methyl)cyclohexyl)methoxy)acetate (Ralinepag): An Orally Active Prostacyclin Receptor Agonist for the Treatment of Pulmonary Arterial Hypertension
Tran, Thuy-Anh, Kramer, Bryan, Shin, Young-Jun, Vallar, Pureza, Boatman, P. Douglas, Zou, Ning, Sage, Carleton R, Gharbaoui, Tawfik, Krishnan, Ashwin, Pal, Biman, Shakya, Sagar R, Garrido Montalban, Antonio, Adams, John W, Ramirez, Juan, Behan, Dominic P, Shifrina, Anna, Blackburn, Anthony, Leakakos, Tina, Shi, Yunqing, Morgan, Michael, Sadeque, Abu, Chen, Weichao, Unett, David J, Gaidarov, Ibragim, Chen, Xiaohua, Chang, Steve, Shu, Hsin-Hui, Tung, Shiu-Feng, Semple, Graeme
Published in Journal of medicinal chemistry (09.02.2017)
Published in Journal of medicinal chemistry (09.02.2017)
Get full text
Journal Article
An Efficient Scale-Up Process for the Preparation of the APD334 Precursor 4‑Chloromethyl-1-cyclopentyl-2-(trifluoromethyl)benzene
Sengupta, Dipanjan, Gharbaoui, Tawfik, Krishnan, Ashwin, Buzard, Daniel J, Jones, Robert M, Ma, You-An, Burda, Robert, Garrido Montalban, Antonio, Semple, Graeme
Published in Organic process research & development (19.06.2015)
Published in Organic process research & development (19.06.2015)
Get full text
Journal Article
Optimization of α-ketoamide based p38 inhibitors through modifications to the region that binds to the allosteric site
Montalban, Antonio Garrido, Boman, Erik, Chang, Chau-Dung, Ceide, Susana Conde, Dahl, Russell, Dalesandro, David, Delaet, Nancy G.J., Erb, Eric, Ernst, Justin T., Gibbs, Andrew, Kahl, Jeffrey, Kessler, Linda, Kucharski, Jeff, Lum, Christopher, Lundström, Jan, Miller, Stephen, Nakanishi, Hiroshi, Roberts, Edward, Saiah, Eddine, Sullivan, Robert, Urban, Jan, Wang, Zhijun, Larson, Christopher J.
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
Get full text
Journal Article
KR-003048, a potent, orally active inhibitor of p38 mitogen-activated protein kinase
Montalban, Antonio Garrido, Boman, Erik, Chang, Chau-Dung, Ceide, Susana Conde, Dahl, Russell, Dalesandro, David, Delaet, Nancy G.J., Erb, Eric, Ernst, Justin, Gibbs, Andrew, Kahl, Jeffrey, Kessler, Linda, Lundström, Jan, Miller, Stephen, Nakanishi, Hiroshi, Roberts, Edward, Saiah, Eddine, Sullivan, Robert, Wang, Zhijun, Larson, Christopher J.
Published in European journal of pharmacology (25.04.2010)
Published in European journal of pharmacology (25.04.2010)
Get full text
Journal Article
The design and synthesis of novel α-ketoamide-based p38 MAP kinase inhibitors
Montalban, Antonio Garrido, Boman, Erik, Chang, Chau-Dung, Ceide, Susana Conde, Dahl, Russell, Dalesandro, David, Delaet, Nancy G.J., Erb, Eric, Ernst, Justin T., Gibbs, Andrew, Kahl, Jeffrey, Kessler, Linda, Lundström, Jan, Miller, Stephen, Nakanishi, Hiroshi, Roberts, Edward, Saiah, Eddine, Sullivan, Robert, Wang, Zhijun, Larson, Christopher J.
Published in Bioorganic & medicinal chemistry letters (15.03.2008)
Published in Bioorganic & medicinal chemistry letters (15.03.2008)
Get full text
Journal Article
Synthesis of porphyrazine-octaamine, hexamine and diamine derivatives
Fuchter, Matthew J., Beall, L. Scott, Baum, Sven M., Montalban, Antonio Garrido, Sakellariou, Efstathia G., Mani, Neelakandha S., Miller, Todd, Vesper, Benjamin J., White, Andrew J.P., Williams, David J., Barrett, Anthony G.M., Hoffman, Brian M.
Published in Tetrahedron (20.06.2005)
Published in Tetrahedron (20.06.2005)
Get full text
Journal Article
‘Reverse’ α-ketoamide-based p38 MAP kinase inhibitors
Montalban, Antonio Garrido, Boman, Erik, Chang, Chau-Dung, Ceide, Susana Conde, Dahl, Russell, Dalesandro, David, Delaet, Nancy G.J., Erb, Eric, Gibbs, Andrew, Kahl, Jeff, Kessler, Linda, Lundström, Jan, Miller, Stephen, Nakanishi, Hiroshi, Roberts, Ed, Saiah, Eddine, Sullivan, Robert, Wang, Zhijun, Larson, Christopher J.
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
Get full text
Journal Article
11 - -2-7-4--3--1234--[]-3- 1 - CRYSTALLINE L-ARGININE SALT OF R-2-7-4-CYCLOPENTYL-3-TRIFLUOROMETHYLBENZYLOXY-1234-TETRAHYDROCYCLO-PENTA[B]INDOL-3-YLACETIC ACIDCOMPOUND1 FOR USE IN SIPI RECEPTOR-ASSOCIATED DISORDERS
MONTALBAN ANTONIO GARRIDO, SELVEY LEE ALANI, HADD MARK A, RUETER JAIMIE KARYN, BLACKBURN ANTHONY C, CASTRO RYAN O, MA YOU AN, CARLOS MARLON, SHAKYA SAGAR RAJ
Year of Publication 24.11.2023
Get full text
Year of Publication 24.11.2023
Patent
EPR Spectra from “EPR-Silent” Species: High-Field EPR Spectroscopy of Manganese(III) Porphyrins
Goldberg, David P, Telser, Joshua, Krzystek, J, Montalban, Antonio Garrido, Brunel, Louis-Claude, Barrett, Anthony G. M, Hoffman, Brian M
Published in Journal of the American Chemical Society (17.09.1997)
Published in Journal of the American Chemical Society (17.09.1997)
Get full text
Journal Article
Novel peripherally functionalized seco-porphyrazines: synthesis, characterization and spectroscopic evaluation
Sakellariou, Efstathia G, Montalban, Antonio Garrido, Beall, Scott L, Henderson, David, Meunier, Hubert G, Phillips, David, Suhling, Klaus, Barrett, Anthony G.M, Hoffman, Brian M
Published in Tetrahedron (10.11.2003)
Published in Tetrahedron (10.11.2003)
Get full text
Journal Article
Peripherally Metalated Secoporphyrazines: A New Generation of Photoactive Pigments
Sakellariou, Efstathia G, Montalban, Antonio Garrido, Meunier, Hubert G, Rumbles, Garry, Phillips, David, Ostler, Richard B, Suhling, Klaus, Barrett, Anthony G. M, Hoffman, Brian M
Published in Inorganic chemistry (22.04.2002)
Published in Inorganic chemistry (22.04.2002)
Get full text
Journal Article
A Facile and Regioselective Synthesis of Trans-Heterofunctionalized Porphyrazine Derivatives
Forsyth, Timothy P, Williams, D. Bradley G, Montalban, Antonio Garrido, Stern, Charlotte L, Barrett, Anthony G. M, Hoffman, Brian M
Published in Journal of organic chemistry (23.01.1998)
Published in Journal of organic chemistry (23.01.1998)
Get full text
Journal Article
Bis(dimethylamino)porphyrazines: Synthetic, Structural, and Spectroscopic Investigations
Montalban, Antonio Garrido, Jarrell, Wade, Riguet, Eric, McCubbin, Quentin J, Anderson, Mairin E, White, Andrew J. P, Williams, David J, Barrett, Anthony G. M, Hoffman, Brian M
Published in Journal of organic chemistry (21.04.2000)
Published in Journal of organic chemistry (21.04.2000)
Get full text
Journal Article
Seco-Porphyrazines: Synthetic, Structural, and Spectroscopic Investigations
Montalban, Antonio Garrido, Lange, Steven J, Beall, L. Scott, Mani, Neelakandha S, Williams, David J, White, Andrew J. P, Barrett, Anthony G. M, Hoffman, Brian M
Published in Journal of organic chemistry (26.12.1997)
Published in Journal of organic chemistry (26.12.1997)
Get full text
Journal Article
Porphyrazinediols: Synthesis, Characterization, and Complexation to Group IVB Metallocenes
Bellec, Nathalie, Garrido Montalban, Antonio, Williams, D. Bradley G, Cook, Andrew S, Anderson, Mairin E, Feng, Xidong, Barrett, Anthony G. M, Hoffman, Brian M
Published in Journal of organic chemistry (24.03.2000)
Published in Journal of organic chemistry (24.03.2000)
Get full text
Journal Article
Metal Ion Binding to Octakis(dimethylamino)porphyrazine: Core Coordination of Mn(III) and Peripheral Coordination of Pd(II)
Goldberg, David P, Montalban, Antonio Garrido, White, Andrew J. P, Williams, David J, Barrett, Anthony G. M, Hoffman, Brian M
Published in Inorganic chemistry (15.06.1998)
Published in Inorganic chemistry (15.06.1998)
Get full text
Journal Article
Synthesis and photophysical properties of peripherally metallated bis(dimethylamino)porphyrazines
Sakellariou, Efstathia G, Montalban, Antonio Garrido, Meunier, Hubert G, Ostler, Richard B, Rumbles, Garry, Barrett, Anthony G.M, Hoffman, Brian M
Published in Journal of photochemistry and photobiology. A, Chemistry. (29.09.2000)
Published in Journal of photochemistry and photobiology. A, Chemistry. (29.09.2000)
Get full text
Journal Article
Ｓ1Ｐ1 수용체-관련 장애에서의 사용을 위한 의 결정성 Ｌ-아르기닌 염
MONTALBAN ANTONIO GARRIDO, SELVEY LEE ALANI, HADD MARK A, RUETER JAIMIE KARYN, BLACKBURN ANTHONY C, CASTRO RYAN O, MA YOU AN, CARLOS MARLON, SHAKYA SAGAR RAJ
Year of Publication 12.02.2018
Get full text
Year of Publication 12.02.2018
Patent