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Applying label-free dynamic mass redistribution technology to frame signaling of G protein-coupled receptors noninvasively in living cells

Applying label-free dynamic mass redistribution technology to frame signaling of G protein-coupled receptors noninvasively in living cells

by Schröder, Ralf, Schmidt, Johannes, Blättermann, Stefanie, Peters, Lucas, Janssen, Nicole, Grundmann, Manuel, Seemann, Wiebke, Kaufel, Dorina, Merten, Nicole, Drewke, Christel, Gomeza, Jesus, Milligan, Graeme, Mohr, Klaus, Kostenis, Evi
Published in Nature protocols (01.11.2011)

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Deconvolution of complex G protein-coupled receptor signaling in live cells using dynamic mass redistribution measurements

Deconvolution of complex G protein-coupled receptor signaling in live cells using dynamic mass redistribution measurements

by Mohr, Klaus, Kostenis, Evi, Schröder, Ralf, Janssen, Nicole, Schmidt, Johannes, Kebig, Anna, Merten, Nicole, Hennen, Stephanie, Müller, Anke, Blättermann, Stefanie, Mohr-Andrä, Marion, Zahn, Sabine, Wenzel, Jörg, Smith, Nicola J, Gomeza, Jesús, Drewke, Christel, Milligan, Graeme
Published in Nature biotechnology (01.09.2010)

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The allosteric vestibule of a seven transmembrane helical receptor controls G-protein coupling

The allosteric vestibule of a seven transmembrane helical receptor controls G-protein coupling

by Bock, Andreas, Merten, Nicole, Schrage, Ramona, Dallanoce, Clelia, Bätz, Julia, Klöckner, Jessica, Schmitz, Jens, Matera, Carlo, Simon, Katharina, Kebig, Anna, Peters, Lucas, Müller, Anke, Schrobang-Ley, Jasmin, Tränkle, Christian, Hoffmann, Carsten, De Amici, Marco, Holzgrabe, Ulrike, Kostenis, Evi, Mohr, Klaus
Published in Nature communications (04.09.2012)

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Rational design of dualsteric GPCR ligands: quests and promise

Rational design of dualsteric GPCR ligands: quests and promise

by Mohr, Klaus, Tränkle, Christian, Kostenis, Evi, Barocelli, Elisabetta, De Amici, Marco, Holzgrabe, Ulrike
Published in British journal of pharmacology (01.03.2010)

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Repurposing HAMI3379 to Block GPR17 and Promote Rodent and Human Oligodendrocyte Differentiation

Repurposing HAMI3379 to Block GPR17 and Promote Rodent and Human Oligodendrocyte Differentiation

by Merten, Nicole, Fischer, Julia, Simon, Katharina, Zhang, Liguo, Schröder, Ralf, Peters, Lucas, Letombe, Anne-Gaelle, Hennen, Stephanie, Schrage, Ramona, Bödefeld, Theresa, Vermeiren, Celine, Gillard, Michel, Mohr, Klaus, Lu, Qing Richard, Brüstle, Oliver, Gomeza, Jesus, Kostenis, Evi
Published in Cell chemical biology (21.06.2018)

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Dynamic ligand binding dictates partial agonism at a G protein-coupled receptor

Dynamic ligand binding dictates partial agonism at a G protein-coupled receptor

by Bock, Andreas, Chirinda, Brian, Krebs, Fabian, Messerer, Regina, Bätz, Julia, Muth, Mathias, Dallanoce, Clelia, Klingenthal, Dominika, Tränkle, Christian, Hoffmann, Carsten, De Amici, Marco, Holzgrabe, Ulrike, Kostenis, Evi, Mohr, Klaus
Published in Nature chemical biology (01.01.2014)

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Rational Design of Partial Agonists for the Muscarinic M1 Acetylcholine Receptor

Rational Design of Partial Agonists for the Muscarinic M1 Acetylcholine Receptor

by Chen, Xinyu, Klöckner, Jessika, Holze, Janine, Zimmermann, Cornelia, Seemann, Wiebke K, Schrage, Ramona, Bock, Andreas, Mohr, Klaus, Tränkle, Christian, Holzgrabe, Ulrike, Decker, Michael
Published in Journal of medicinal chemistry (22.01.2015)

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Hybrid Molecules from Xanomeline and Tacrine: Enhanced Tacrine Actions on Cholinesterases and Muscarinic M1 Receptors

Hybrid Molecules from Xanomeline and Tacrine: Enhanced Tacrine Actions on Cholinesterases and Muscarinic M1 Receptors

by Fang, Lei, Jumpertz, Sabine, Zhang, Yihua, Appenroth, Dorothea, Fleck, Christian, Mohr, Klaus, Tränkle, Christian, Decker, Michael
Published in Journal of medicinal chemistry (11.03.2010)

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Ligand-Specific Allosteric Coupling Controls G‑Protein-Coupled Receptor Signaling

Ligand-Specific Allosteric Coupling Controls G‑Protein-Coupled Receptor Signaling

by Holze, Janine, Bermudez, Marcel, Pfeil, Eva Marie, Kauk, Michael, Bödefeld, Theresa, Irmen, Matthias, Matera, Carlo, Dallanoce, Clelia, De Amici, Marco, Holzgrabe, Ulrike, König, Gabriele Maria, Tränkle, Christian, Wolber, Gerhard, Schrage, Ramona, Mohr, Klaus, Hoffmann, Carsten, Kostenis, Evi, Bock, Andreas
Published in ACS pharmacology & translational science (09.10.2020)

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Allosteric Small Molecules Unveil a Role of an Extracellular E2/Transmembrane Helix 7 Junction for G Protein-coupled Receptor Activation

Allosteric Small Molecules Unveil a Role of an Extracellular E2/Transmembrane Helix 7 Junction for G Protein-coupled Receptor Activation

by Jäger, Dorothea, Schmalenbach, Caroline, Prilla, Stefanie, Schrobang, Jasmin, Kebig, Anna, Sennwitz, Matthias, Heller, Eberhard, Tränkle, Christian, Holzgrabe, Ulrike, Höltje, Hans-Dieter, Mohr, Klaus
Published in The Journal of biological chemistry (30.11.2007)

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Allosteric Site on Muscarinic Acetylcholine Receptors: Identification of Two Amino Acids in the Muscarinic M2 Receptor That Account Entirely for the M2/M5 Subtype Selectivities of Some Structurally Diverse Allosteric Ligands in N-Methylscopolamine-Occupied Receptors

Allosteric Site on Muscarinic Acetylcholine Receptors: Identification of Two Amino Acids in the Muscarinic M2 Receptor That Account Entirely for the M2/M5 Subtype Selectivities of Some Structurally Diverse Allosteric Ligands in N-Methylscopolamine-Occupied Receptors

by Voigtländer, Uta, Jöhren, Kirstin, Mohr, Marion, Raasch, Alexandra, Tränkle, Christian, Buller, Stefan, Ellis, John, Höltje, Hans-Dieter, Mohr, Klaus
Published in Molecular pharmacology (01.07.2003)

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An optical dynamic mass redistribution assay reveals biased signaling of dualsteric GPCR activators

An optical dynamic mass redistribution assay reveals biased signaling of dualsteric GPCR activators

by Kebig, Anna, Kostenis, Evi, Mohr, Klaus, Mohr-Andrä, Marion
Published in Journal of receptors and signal transduction (01.01.2009)

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Interactions of Orthosteric and Allosteric Ligands with [3H]Dimethyl-W84 at the Common Allosteric Site of Muscarinic M2 Receptors

Interactions of Orthosteric and Allosteric Ligands with [3H]Dimethyl-W84 at the Common Allosteric Site of Muscarinic M2 Receptors

by Tränkle, Christian, Weyand, Oliver, Voigtländer, Uta, Mynett, Anita, Lazareno, Sebastian, Birdsall, Nigel J M, Mohr, Klaus
Published in Molecular pharmacology (01.07.2003)

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A hydrazide linker strategy for heterobivalent compounds as ortho- and allosteric ligands of acetylcholine-binding proteins

A hydrazide linker strategy for heterobivalent compounds as ortho- and allosteric ligands of acetylcholine-binding proteins

by Elsinghorst, Paul W, Härtig, Wolfgang, Gündisch, Daniela, Mohr, Klaus, Tränkle, Christian, Gütschow, Michael
Published in Current topics in medicinal chemistry (01.11.2011)

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Allosteric modulators targeting CNS muscarinic receptors

Allosteric modulators targeting CNS muscarinic receptors

by Bock, Andreas, Schrage, Ramona, Mohr, Klaus
Published in Neuropharmacology (01.07.2018)

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Allosteric Site on Muscarinic Acetylcholine Receptors: A Single Amino Acid in Transmembrane Region 7 Is Critical to the Subtype Selectivities of Caracurine V Derivatives and Alkane-Bisammonium Ligands

Allosteric Site on Muscarinic Acetylcholine Receptors: A Single Amino Acid in Transmembrane Region 7 Is Critical to the Subtype Selectivities of Caracurine V Derivatives and Alkane-Bisammonium Ligands

by Buller, Stefan, Zlotos, Darius Paul, Mohr, Klaus, Ellis, John
Published in Molecular pharmacology (01.01.2002)

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Allosteric Modulation of Muscarinic Receptor Signaling: Alcuronium-Induced Conversion of Pilocarpine from an Agonist into an Antagonist

Allosteric Modulation of Muscarinic Receptor Signaling: Alcuronium-Induced Conversion of Pilocarpine from an Agonist into an Antagonist

by Katrin Zahn, Niels Eckstein, Christian TrÃ¤nkle, Wolfgang SadÃ©e, Klaus Mohr
Published in The Journal of pharmacology and experimental therapeutics (01.05.2002)

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Using a Radioalloster to Test Predictions of the Cooperativity Model for Gallamine Binding to the Allosteric Site of Muscarinic Acetylcholine M2 Receptors

Using a Radioalloster to Test Predictions of the Cooperativity Model for Gallamine Binding to the Allosteric Site of Muscarinic Acetylcholine M2 Receptors

by Christian TrÃ¤nkle, Oliver Weyand, Alexandra SchrÃ¶ter, Klaus Mohr
Published in Molecular pharmacology (01.11.1999)

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Divergent Modes of Action among Cationic Allosteric Modulators of Muscarinic M2 Receptors

Divergent Modes of Action among Cationic Allosteric Modulators of Muscarinic M2 Receptors

by Tränkle, C, Mohr, K
Published in Molecular pharmacology (01.04.1997)

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Structure−Activity Relationships in a Series of Bisquaternary Bisphthalimidine Derivatives Modulating the Muscarinic M2-Receptor Allosterically

Structure−Activity Relationships in a Series of Bisquaternary Bisphthalimidine Derivatives Modulating the Muscarinic M2-Receptor Allosterically

by Botero Cid, Hector M, Tränkle, Christian, Baumann, Knut, Pick, Rainer, Mies-Klomfass, Elisabeth, Kostenis, Evi, Mohr, Klaus, Holzgrabe, Ulrike
Published in Journal of medicinal chemistry (01.06.2000)

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