Potent, Selective, Water Soluble, Brain-Permeable EP2 Receptor Antagonist for Use in Central Nervous System Disease Models
Amaradhi, Radhika, Banik, Avijit, Mohammed, Shabber, Patro, Vidyavathi, Rojas, Asheebo, Wang, Wenyi, Motati, Damoder Reddy, Dingledine, Ray, Ganesh, Thota
Published in Journal of medicinal chemistry (13.02.2020)
Published in Journal of medicinal chemistry (13.02.2020)
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Journal Article
Combinatorial targeting of glutamine metabolism and lysosomal-based lipid metabolism effectively suppresses glioblastoma
Zhong, Yaogang, Geng, Feng, Mazik, Logan, Yin, Xinmin, Becker, Aline Paixao, Mohammed, Shabber, Su, Huali, Xing, Enming, Kou, Yongjun, Chiang, Cheng-Yao, Fan, Yunzhou, Guo, Yongchen, Wang, Qiang, Li, Pui-Kai, Mo, Xiaokui, Lefai, Etienne, He, Liqing, Cheng, Xiaolin, Zhang, Xiang, Chakravarti, Arnab, Guo, Deliang
Published in Cell reports. Medicine (17.09.2024)
Published in Cell reports. Medicine (17.09.2024)
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Journal Article
Discovery of Quinazolin-4(3H)‑ones as NLRP3 Inflammasome Inhibitors: Computational Design, Metal-Free Synthesis, and in Vitro Biological Evaluation
Abdullaha, Mohd, Mohammed, Shabber, Ali, Mehboob, Kumar, Ajay, Vishwakarma, Ram A, Bharate, Sandip B
Published in Journal of organic chemistry (03.05.2019)
Published in Journal of organic chemistry (03.05.2019)
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Journal Article
GAC inhibitors with a 4-hydroxypiperidine spacer: Requirements for potency
McDermott, Lee, Koes, David, Mohammed, Shabber, Iyer, Prema, Boby, Melissa, Balasubramanian, Venkatakrishnan, Geedy, Mackenzie, Katt, William, Cerione, Richard
Published in Bioorganic & medicinal chemistry letters (01.10.2019)
Published in Bioorganic & medicinal chemistry letters (01.10.2019)
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Journal Article
LX1 Targets Androgen Receptor Variants and AKR1C3 to overcome Therapy Resistance in Advanced Prostate Cancer
Ning, Shu, Armstrong, Cameron M, Xing, Enming, Leslie, Amy R, Gao, Richard Y, Sharifi, Masuda, Schaaf, Zachary A, Lou, Wei, Han, Xiangrui, Xu, Desiree H, Yang, Rui, Cheng, Jeffrey, Mohammed, Shabber, Mitsiades, Nicholas, Liu, Chengfei, Lombard, Alan P, Wu, Chun-Yi, Cheng, Xiolin, Li, Pui-Kai, Gao, Allen C
Published in Cancer research (Chicago, Ill.) (01.08.2024)
Published in Cancer research (Chicago, Ill.) (01.08.2024)
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Journal Article
Abstract 3106: Design, synthesis, and screening of niclosamide analogs as androgen receptor degraders for hepatocellular carcinoma
Cheng, Jeffrey, Xing, Enming, Mohammed, Shabber, Montgomery, Emma, Granchie, Lauren, Coss, Christopher, Li, Pui-Kai
Published in Cancer research (Chicago, Ill.) (04.04.2023)
Published in Cancer research (Chicago, Ill.) (04.04.2023)
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Journal Article
Second-Generation Prostaglandin Receptor EP2 Antagonist, TG8-260, with High Potency, Selectivity, Oral Bioavailability, and Anti-Inflammatory Properties
Amaradhi, Radhika, Mohammed, Shabber, Banik, Avijit, Franklin, Ronald, Dingledine, Raymond, Ganesh, Thota
Published in ACS pharmacology & translational science (11.02.2022)
Published in ACS pharmacology & translational science (11.02.2022)
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Journal Article
Synthesis, antileishmanial and antitrypanosomal activities of N-substituted tetrahydro-beta-carbolines
Manda, Sudhakar, Khan, Shabana I., Jain, Surendra K., Mohammed, Shabber, Tekwani, Babu L., Khan, Ikhlas A., Vishwakarma, Ram A., Bharate, Sandip B.
Published in Bioorganic & medicinal chemistry letters (01.08.2014)
Published in Bioorganic & medicinal chemistry letters (01.08.2014)
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Journal Article
PROSTAGLANDIN RECEPTOR EP2 ANTAGONISTS, DERIVATIVES, AND USES RELATED THERETO
GANESH, Thota, DINGLEDINE, Raymond J, AMARADAHI, Radhika, MOHAMMED, Shabber
Year of Publication 23.11.2022
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Year of Publication 23.11.2022
Patent
PROSTAGLANDIN RECEPTOR EP2 ANTAGONISTS, DERIVATIVES, AND USES RELATED THERETO
GANESH, Thota, DINGLEDINE, Raymond J, AMARADAHI, Radhika, MOHAMMED, Shabber
Year of Publication 26.05.2022
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Year of Publication 26.05.2022
Patent