NOVEL CHIRAL N-ACYL-5,6,7,(8-SUBSTITUTED)-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-A]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS AND CHIRAL SYNTHESIS THEREOF
BATT, FRÉDÉRIC, HOVEYDA, HAMID, ROY, MARIE-ODILE, EL BOUSMAQUI, MOHAMED, DUTHEUIL, GUILLAUME, FRASER, GRAEME
Year of Publication 08.06.2016
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Year of Publication 08.06.2016
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HIDTIL UKENDTE CHIRALE N-ACYL-5,6,7,(8-SUBSTITUERET)-TETRAHYDRO-[1,2,4]TRIAZOL[4,3-A]PYRAZINER SOM SELEKTIVE NK-3-RECEPTORANTAGONISTER, FARMACEUTISK SAMMENSÆTNING OG FREMGANGSMÅDER TIL ANVENDELSE VED NK-3-RECEPTORMEDIEREDE SYGDOMME
BATT, FRÉDÉRIC, ROY, MARIE-ODILE, EL BOUSMAQUI, MOHAMED, FRASER, GRAEME, DUTHEUIL, GUILLAUME, HOVEYEDA, HAMID
Year of Publication 25.04.2016
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Year of Publication 25.04.2016
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NOVEL CHIRAL N-ACYL-5,6,7,(8-SUBSTITUTED)-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-A]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, AND METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS
BATT, FRÉDÉRIC, ROY, MARIE-ODILE, EL BOUSMAQUI, MOHAMED, DUTHEUIL, GUILLAUME, FRASER, GRAEME, HOVEYEDA, HAMID
Year of Publication 06.04.2016
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Year of Publication 06.04.2016
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Novel chiral n-acyl-5,6,7,(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines as selective nk-3 receptor antagonists, pharmaceutical composition, methods for use in nk-3 receptor mediated disorders and chiral synthesis thereof
DUTHEUIL GUILLAUME, ROY MARIE-ODILE, FRASER GRAEME, EL BOUSMAQUI MOHAMED, BATT FREDERIC, HOVEYDA HAMID
Year of Publication 23.12.2015
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Year of Publication 23.12.2015
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NOVEL CHIRAL N-ACYL-5,6,7,(8-SUBSTITUTED)-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-A]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, AND METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS
BATT, FRÉDÉRIC, ROY, MARIE-ODILE, EL BOUSMAQUI, MOHAMED, DUTHEUIL, GUILLAUME, FRASER, GRAEME, HOVEYEDA, HAMID
Year of Publication 13.08.2014
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Year of Publication 13.08.2014
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Novel chiral N-acyl-5,6,7,(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor mediated disorders and chiral synthesis thereof
HOVEYDA, HAMID, ROY, MARIE-ODILE, EL BOUSMAQUI, MOHAMED, DUTHEUIL, GUILLAUME, FRASER, GRAEME, BATT, FREDERIC
Year of Publication 10.04.2014
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Year of Publication 10.04.2014
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NOVEL CHIRAL N-ACYL-5,6,7,(8-SUBSTITUTED)-TETRAHYDRO-[1,2,4]TRIAZ OLO[4,3-a]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS AND CHIRAL SYNTHESIS THEREOF
Frédéric BATT, Mohamed EL BOUSMAQUI, Graeme FRASER, Guillaume DUTHEUIL, Hamid HOVEYDA, Marie-Odile ROY
Year of Publication 04.09.2019
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Year of Publication 04.09.2019
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NOVEL CHIRAL N-ACYL-5,6,7(8-SUBSTITUTED)-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-a]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS AND CHIRAL SYNTHESIS THEREOF
DUTHEUIL GUILLAUME, HOVEYDA HAMID R, FRASER GRAEME L, ROY MARIE-ODILE, EL BOUSMAQUI MOHAMED, BATT FREDERIC
Year of Publication 18.09.2014
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Year of Publication 18.09.2014
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NOVEL CHIRAL N-ACYL-5,6,7,(8-SUBSTITUTED)-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-a]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS AND CHIRAL SYNTHESIS THEREOF
HOVEYDA, HAMID, ROY, MARIE-ODILE, EL BOUSMAQUI, MOHAMED, DUTHEUIL, GUILLAUME, FRASER, GRAEME, BATT, FREDERIC
Year of Publication 11.04.2013
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Year of Publication 11.04.2013
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NOVEL CHIRAL N-ACYL-5,6,7,(8-SUBSTITUTED)-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-A]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS AND CHIRAL SYNTHESIS THEREOF
HOVEYDA, HAMID, ROY, MARIE-ODILE, EL BOUSMAQUI, MOHAMED, DUTHEUIL, GUILLAUME, FRASER, GRAEME, BATT, FREDERIC
Year of Publication 11.04.2013
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Year of Publication 11.04.2013
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INTERMEDIATE FOR PREPARING NEUROKININ-3 RECEPTOR ANTAGONISTS
HOVEYDA Hamid, ROY Marie-Odile, FRASER Graeme, EL BOUSMAQUI Mohamed, BATT Frederic, DUTHEUIL Guillaume
Year of Publication 31.08.2018
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Year of Publication 31.08.2018
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CHIRAL N-ACYL-5,6,7-(8-SUBSTITUTED)TETRAHYDRO[1,2,4]TRIAZOLO[4,3-a]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS AND CHIRAL SYNTHESIS THEREOF
ROY Marie-Odile, FRASER Graeme, EL BOUSMAQUI Mohamed, BATT Frederic, HOVEYEDA Hamid, DUTHEUIL Guillaume
Year of Publication 30.03.2018
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Year of Publication 30.03.2018
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n-acil-5,6,7, (8-substituído) - tetraidro-[1,2,4] triazolo [4,3 -a] pirazinas quirais inovadoras como antagonistas de receptor de nk-3 seletivos, composição farmacêutica, métodos para usar em distúrbios mediados por receptor de nk-3 e síntese quiral dos mesmos
HAMID HOVEYDA, MARIE-ODILE ROY, FRÉDÉRIC BATT, GRAEME FRASER, GUILLAUME DUTHEUIL, MOHAMED EL BOUSMAQUI
Year of Publication 23.01.2018
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Year of Publication 23.01.2018
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NOVEL COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS FOR USE IN TREATING METABOLIC DISORDERS
BERNARD, JEROME, HOVEYDA, HAMID, EL BOUSMAQUI, MOHAMED, DUTHEUIL, GUILLAUME
Year of Publication 08.12.2011
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Year of Publication 08.12.2011
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ΝΕΕΣ ΧΕΙΡΙΚΕΣ Ν-ΑΚΥΛ-5,6,7,8-ΥΠΟΚΑΤΕΣΤΗΜΕΝΕΣ)-ΤΕΤΡΑΫΔΡΟ-[1,2,4]ΤΡΙΑΖΟΛΟ[4,3-A]ΠΥΡΑΖΙΝΕΣ ΩΣ ΕΠΙΛΕΚΤΙΚΟΙ ΑΝΤΑΓΩΝΙΣΤΕΣ ΤΟΥ ΥΠΟΔΟΧΕΑ ΝΚ-3, ΦΑΡΜΑΚΕΥΤΙΚΗ ΣΥΝΘΕΣΗ ΚΑΙ ΜΕΘΟΔΟΙ ΓΙΑ ΤΗ ΧΡΗΣΗ ΣΕ ΔΙΑΤΑΡΑΧΕΣ ΜΕΣΟΛΑΒΟΥΜΕΝΕΣ ΑΠΟ ΤΟΝ ΥΠΟΔΟΧΕΑ ΝΚ-3
BATT Frédéric, ROY Marie-Odile, FRASER Graeme, EL BOUSMAQUI Mohamed, HOVEYEDA Hamid, DUTHEUIL Guillaume
Year of Publication 17.05.2017
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Year of Publication 17.05.2017
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n-acil-5,6,7, (8-substituído) - tetraidro-[1,2,4] triazolo [4,3 -a] pirazinas quirais inovadoras como antagonistas de receptor de nk-3 seletivos, composição farmacêutica, métodos para usar em distúrbios mediados por receptor de nk-3 e síntese quiral dos mesmos
HAMID HOVEYDA, MARIE-ODILE ROY, FRÉDÉRIC BATT, GRAEME FRASER, GUILLAUME DUTHEUIL, MOHAMED EL BOUSMAQUI
Year of Publication 11.04.2017
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Year of Publication 11.04.2017
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NOVEL CHIRAL N-ACYL-5,6,7,(8-SUBSTITUTED)-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-A]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, AND METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS
BATT, FRÉDÉRIC, ROY, MARIE-ODILE, EL BOUSMAQUI, MOHAMED, DUTHEUIL, GUILLAUME, FRASER, GRAEME, HOVEYEDA, HAMID
Year of Publication 31.10.2016
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Year of Publication 31.10.2016
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Nuevas N-acil-5,6,7,(8-sustituido)-tetrahidro-[1,2,4]triazolo[4,3a]pirazinas quirales, como antagonistas selectivas del receptor de NK-3, composición farmacéutica y métodos para uso en trastornos mediados por el receptor de NK-3
DUTHEUIL, Guillaume, EL BOUSMAQUI, Mohamed, BATT, Frédéric, ROY, Marie-Odile, HOVEYEDA, Hamid, FRASER, Graeme
Year of Publication 01.06.2016
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Year of Publication 01.06.2016
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NOVEL CHIRAL N-ACYL-5,6,7,(8-SUBSTITUTED)-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3- A]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, AND METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS NK-3 N--567(8-)--[12 4][43-A] NK-3
DUTHEUIL, Guillaume, EL BOUSMAQUI, Mohamed, BATT, Frdric, ROY, Marie-Odile, HOVEYEDA, Hamid, FRASER, Graeme
Year of Publication 06.02.2015
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Year of Publication 06.02.2015
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NOVEL CHIRAL N-ACYL-5,6,7,(8-SUBSTITUTED)-TETRAHYDRO-[1,2,4]TRIAZ OLO[4,3-a]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS AND CHIRAL SYNTHESIS THEREOF
HAMID HOVEYDA, MARIE-ODILE ROY, FRÉDÉRIC BATT, GRAEME FRASER, GUILLAUME DUTHEUIL, MOHAMED EL BOUSMAQUI
Year of Publication 22.08.2014
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Year of Publication 22.08.2014
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