An efficient and convenient synthesis of tetrahydrocycloheptapyridines: New precursors for CNS agents
Yoshizumi, T, Miyazoe, H, Sugimoto, Y, Takahashi, H, Okamoto, O
Published in Synthesis (Stuttgart) (01.07.2005)
Published in Synthesis (Stuttgart) (01.07.2005)
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Journal Article
Design, synthesis and evaluation of a novel cyclohexanamine class of neuropeptide Y Y1 receptor antagonists
Cho, Kaimei, Ando, Makoto, Kobayashi, Kensuke, Miyazoe, Hiroshi, Tsujino, Toshiaki, Ito, Sayaka, Suzuki, Tomoki, Tanaka, Takeshi, Tokita, Shigeru, Sato, Nagaaki
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
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Journal Article
Design, synthesis, and structure–activity relationship study of a novel class of ORL1 receptor antagonists based on N-biarylmethyl spiropiperidine
Yoshizumi, Takashi, Miyazoe, Hiroshi, Ito, Hirokatsu, Tsujita, Tomohiro, Takahashi, Hirobumi, Asai, Masanori, Ozaki, Satoshi, Ohta, Hisashi, Okamoto, Osamu
Published in Bioorganic & medicinal chemistry (01.07.2008)
Published in Bioorganic & medicinal chemistry (01.07.2008)
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A Novel Class of Cycloalkano[b]pyridines as Potent and Orally Active Opioid Receptor-like 1 Antagonists with Minimal Binding Affinity to the hERG K+ Channel
Yoshizumi, Takashi, Takahashi, Hirobumi, Miyazoe, Hiroshi, Sugimoto, Yuichi, Tsujita, Tomohiro, Kato, Tetsuya, Ito, Hirokatsu, Kawamoto, Hiroshi, Hirayama, Mioko, Ichikawa, Daisuke, Azuma-Kanoh, Tomoko, Ozaki, Satoshi, Shibata, Yoshihiro, Tani, Takeshi, Chiba, Masato, Ishii, Yasuyuki, Okuda, Shoki, Tadano, Kiyoshi, Fukuroda, Takahiro, Okamoto, Osamu, Ohta, Hisashi
Published in Journal of medicinal chemistry (10.07.2008)
Published in Journal of medicinal chemistry (10.07.2008)
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Journal Article
Synthetic and Theoretical Studies on Group-Transfer Imidoylation of Organotellurium Compounds. Remarkable Reactivity of Isonitriles in Comparison with Carbon Monoxide in Radical-Mediated Reactions
Yamago, Shigeru, Miyazoe, Hiroshi, Goto, Ryuta, Hashidume, Masahiro, Sawazaki, Takashi, Yoshida, Jun-ichi
Published in Journal of the American Chemical Society (25.04.2001)
Published in Journal of the American Chemical Society (25.04.2001)
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Optimization of a series of 2,4-diaminopyridines as neuropeptide Y Y1 receptor antagonists with reduced hERG activity
Kameda, Minoru, Kobayashi, Kensuke, Ito, Hirokatsu, Miyazoe, Hiroshi, Tsujino, Toshiaki, Nakama, Chisato, Kawamoto, Hiroshi, Ando, Makoto, Ito, Sayaka, Suzuki, Tomoki, Kanno, Tetsuya, Tanaka, Takeshi, Tahara, Yoshio, Tani, Takeshi, Tanaka, Sachiko, Tokita, Shigeru, Sato, Nagaaki
Published in Bioorganic & medicinal chemistry letters (01.08.2009)
Published in Bioorganic & medicinal chemistry letters (01.08.2009)
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Journal Article
A Diversity-Oriented Synthesis of α-Amino Acid Derivatives by a Silyltelluride-Mediated Radical Coupling Reaction of Imines and Isonitriles
Yamago, Shigeru, Miyazoe, Hiroshi, Nakayama, Takeyoshi, Miyoshi, Masaki, Yoshida, Junichi
Published in Angewandte Chemie (International ed.) (03.01.2003)
Published in Angewandte Chemie (International ed.) (03.01.2003)
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Journal Article
Discovery of novel arylpyrazole series as potent and selective opioid receptor-like 1 (ORL1) antagonists
Kobayashi, Kensuke, Uchiyama, Minaho, Ito, Hirokatsu, Takahashi, Hirobumi, Yoshizumi, Takashi, Sakoh, Hiroki, Nagatomi, Yasushi, Asai, Masanori, Miyazoe, Hiroshi, Tsujita, Tomohiro, Hirayama, Mioko, Ozaki, Satoshi, Tani, Takeshi, Ishii, Yasuyuki, Ohta, Hisashi, Okamoto, Osamu
Published in Bioorganic & medicinal chemistry letters (01.07.2009)
Published in Bioorganic & medicinal chemistry letters (01.07.2009)
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Journal Article
2-Cyclohexylcarbonylbenzimidazoles as potent, orally available and brain-penetrable opioid receptor-like 1 (ORL1) antagonists
Kobayashi, Kensuke, Uchiyama, Minaho, Takahashi, Hirobumi, Kawamoto, Hiroshi, Ito, Satoru, Yoshizumi, Takashi, Nakashima, Hiroshi, Kato, Tetsuya, Shimizu, Atsushi, Yamamoto, Izumi, Asai, Masanori, Miyazoe, Hiroshi, Ohno, Akio, Hirayama, Mioko, Ozaki, Satoshi, Tani, Takeshi, Ishii, Yasuyuki, Tanaka, Takeshi, Mochidome, Takanobu, Tadano, Kiyoshi, Fukuroda, Takahiro, Ohta, Hisashi, Okamoto, Osamu
Published in Bioorganic & medicinal chemistry letters (01.06.2009)
Published in Bioorganic & medicinal chemistry letters (01.06.2009)
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Journal Article
DIARYL KETIMINE DERIVATIVE HAVING ANTAGONISTIC ACTIVITY ON MELANIN-CONCENTRATING HORMONE RECEPTOR
HIROSE, ETSUKO, KAMEDA, MINORU, MORIYA, MINORU, SUZUKI, TAKAO, ANDO, MAKOTO, MIYAZOE, HIROSHI
Year of Publication 02.04.2009
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Year of Publication 02.04.2009
Patent
Discovery of novel diarylketoxime derivatives as selective and orally active melanin-concentrating hormone 1 receptor antagonists
Suzuki, Takao, Kameda, Minoru, Ando, Makoto, Miyazoe, Hiroshi, Sekino, Etsuko, Ito, Satoru, Masutani, Kouta, Kamijo, Kaori, Takezawa, Akihiro, Moriya, Minoru, Ito, Masahiko, Ito, Junko, Nakase, Kazuho, Matsushita, Hiroko, Ishihara, Akane, Takenaga, Norihiro, Tokita, Shigeru, Kanatani, Akio, Sato, Nagaaki, Fukami, Takehiro
Published in Bioorganic & medicinal chemistry letters (15.09.2009)
Published in Bioorganic & medicinal chemistry letters (15.09.2009)
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Journal Article
DIARYL KETIMINE DERIVATIVE
KAMEDA, MINORU, MORIYA, MINORU, SUZUKI, TAKAO, ANDO, MAKOTO, MIYAZOE, HIROSHI, SEKINO, ETSUKO
Year of Publication 24.04.2008
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Year of Publication 24.04.2008
Patent
DIARYL KETIMINE DERIVATIVE
KAMEDA, MINORU, MORIYA, MINORU, SUZUKI, TAKAO, ANDO, MAKOTO, MIYAZOE, HIROSHI, SEKINO, ETSUKO
Year of Publication 03.04.2008
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Year of Publication 03.04.2008
Patent
ALKYLAMINOPYRIDINE DERIVATIVE
KAMEDA, MINORU, KAWAMOTO, HIROSHI, KOBAYASHI, KENSUKE, ANDO, MAKOTO, ITO, HIROKATSU, TSUJINO, TOSHIAKI, MIYAZOE, HIROSHI, NAKAMA, CHISATO, SATO, NAGAAKI
Year of Publication 11.09.2009
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Year of Publication 11.09.2009
Patent