Search Results - "MITKIN OLEG" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Non-rigid Diarylmethyl Analogs of Baloxavir as Cap-Dependent Endonuclease Inhibitors of Influenza Viruses

Non-rigid Diarylmethyl Analogs of Baloxavir as Cap-Dependent Endonuclease Inhibitors of Influenza Viruses

by Ivashchenko, Andrei A, Mitkin, Oleg D, Jones, Jeremy C, Nikitin, Alexander V, Koryakova, Angela G, Ryakhovskiy, Alexey, Karapetian, Ruben N, Kravchenko, Dmitry V, Aladinskiy, Vladimir, Leneva, Irina A, Falynskova, Irina N, Glubokova, Ekaterina A, Govorkova, Elena A, Ivachtchenko, Alexandre V
Published in Journal of medicinal chemistry (10.09.2020)

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Synthesis and Structure–Activity Relationship (SAR) of (5,7-Disubstituted 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidin-2-yl)-methylamines as Potent Serotonin 5-HT6 Receptor (5-HT6R) Antagonists

Synthesis and Structure–Activity Relationship (SAR) of (5,7-Disubstituted 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidin-2-yl)-methylamines as Potent Serotonin 5-HT6 Receptor (5-HT6R) Antagonists

by Ivachtchenko, Alexandre V, Golovina, Elena S, Kadieva, Madina G, Kysil, Volodymyr M, Mitkin, Oleg D, Tkachenko, Sergey E, Okun, Ilya M
Published in Journal of medicinal chemistry (08.12.2011)

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Synthesis, inhibitory activity and oral dosing formulation of AV5124, the structural analogue of influenza virus endonuclease inhibitor baloxavir

Synthesis, inhibitory activity and oral dosing formulation of AV5124, the structural analogue of influenza virus endonuclease inhibitor baloxavir

by Ivashchenko, Andrei A, Mitkin, Oleg D, Jones, Jeremy C, Nikitin, Alexander V, Koryakova, Angela G, Karapetian, Ruben N, Kravchenko, Dmitry V, Mochalov, Stephan V, Ryakhovskiy, Alexey A, Aladinskiy, Vladimir, Leneva, Irina A, Falynskova, Irina N, Glubokova, Ekaterina A, Govorkova, Elena A, Ivachtchenko, Alexandre V
Published in Journal of antimicrobial chemotherapy (12.03.2021)

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Synthesis, biological evaluation and in silico modeling of novel pan-genotypic NS5A inhibitors

Synthesis, biological evaluation and in silico modeling of novel pan-genotypic NS5A inhibitors

by Ivashchenko, Andrey A., Ivanenkov, Yan A., Aladinskiy, Vladimir A., Karapetian, Ruben N., Koryakova, Angela G., Ryakhovskiy, Alexey A., Mitkin, Oleg D., Kravchenko, Dmitry V., Savchuk, Nikolai P., Zagribelnyy, Bogdan A., Ivashchenko, Alexander V.
Published in Bioorganic & medicinal chemistry (15.10.2020)

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Synthesis, biological evaluation and in silico modeling of novel integrase strand transfer inhibitors (INSTIs)

Synthesis, biological evaluation and in silico modeling of novel integrase strand transfer inhibitors (INSTIs)

by Ivashchenko, Andrey A., Ivanenkov, Yan A., Koryakova, Angela G., Karapetian, Ruben N., Mitkin, Oleg D., Aladinskiy, Vladimir A., Kravchenko, Dmitry V., Savchuk, Nikolai P., Ivashchenko, Alexander V.
Published in European journal of medicinal chemistry (01.03.2020)

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Safety and efficacy of aviandr in patients with generalized anxiety disorder: A multicenter, randomized, double-blind, placebo-controlled, dose-finding, pilot study

Safety and efficacy of aviandr in patients with generalized anxiety disorder: A multicenter, randomized, double-blind, placebo-controlled, dose-finding, pilot study

by Ivashchenko, Andrey A., Morozova, Margarita A., Vostokova, Natalia V., Beniashvily, Allan G., Bukhanovskaya, Olga A., Burminskiy, Denis S., Egorova, Alina N., Gluskina, Lubov Y., Gorchakov, Dmitriy S., Karapetian, Ruben N., Kasimova, Lala N., Kravchenko, Dmitry V., Lepilkina, Taissia A., Merkulova, Elena A., Mitkin, Oleg D., Penchul, Nataliya A., Potanin, Sergey S., Rupchev, George E., Ivachtchenko, Alexandre V.
Published in Journal of psychiatric research (01.11.2021)

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(3-Phenylsulfonylcycloalkano[e and d]pyrazolo[1,5-a]pyrimidin-2-yl)amines: Potent and Selective Antagonists of the Serotonin 5-HT6 Receptor

(3-Phenylsulfonylcycloalkano[e and d]pyrazolo[1,5-a]pyrimidin-2-yl)amines: Potent and Selective Antagonists of the Serotonin 5-HT6 Receptor

by Ivachtchenko, Alexandre V, Dmitriev, Dmitri E, Golovina, Elena S, Kadieva, Madina G, Koryakova, Angela G, Kysil, Volodymyr M, Mitkin, Oleg D, Okun, Ilya M, Tkachenko, Sergey E, Vorobiev, Anton A
Published in Journal of medicinal chemistry (22.07.2010)

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Design, synthesis and biological evaluation of novel 5-oxo-2-thioxoimidazolidine derivatives as potent androgen receptor antagonists

Design, synthesis and biological evaluation of novel 5-oxo-2-thioxoimidazolidine derivatives as potent androgen receptor antagonists

by Ivachtchenko, Alexandre V., Ivanenkov, Yan A., Mitkin, Oleg D., Vorobiev, Anton A., Kuznetsova, Irina V., Shevkun, Natalia A., Koryakova, Angela G., Karapetian, Ruben N., Trifelenkov, Andrey S., Kravchenko, Dmitry V., Veselov, Mark S., Chufarova, Nina V.
Published in European journal of medicinal chemistry (24.06.2015)

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Synthesis, X-Ray Crystal Structure, Hirshfeld Surface Analysis, and Molecular Docking Study of Novel Hepatitis B (HBV) Inhibitor: 8-Fluoro-5-(4-fluorobenzyl)-3-(2-methoxybenzyl)-3,5-dihydro-4H-pyrimido[5,4-b]indol-4-one

Synthesis, X-Ray Crystal Structure, Hirshfeld Surface Analysis, and Molecular Docking Study of Novel Hepatitis B (HBV) Inhibitor: 8-Fluoro-5-(4-fluorobenzyl)-3-(2-methoxybenzyl)-3,5-dihydro-4H-pyrimido[5,4-b]indol-4-one

by Ivashchenko, Aleksandr V., Mitkin, Oleg D., Kravchenko, Dmitry V., Kuznetsova, Irina V., Kovalenko, Sergiy M., Bunyatyan, Natalya D., Langer, Thierry
Published in Crystals (Basel) (01.08.2019)

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Synthesis and SAR of 3-arylsulfonyl-pyrazolo[1,5-a]pyrimidines as potent serotonin 5-HT6 receptor antagonists

Synthesis and SAR of 3-arylsulfonyl-pyrazolo[1,5-a]pyrimidines as potent serotonin 5-HT6 receptor antagonists

by Ivachtchenko, Alexandre V., Golovina, Elena S., Kadieva, Madina G., Kysil, Volodymyr M., Mitkin, Oleg D., Tkachenko, Sergey E., Okun, Ilya
Published in Bioorganic & medicinal chemistry (15.02.2011)

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Novel oral anti-influenza drug candidate AV5080

Novel oral anti-influenza drug candidate AV5080

by Ivachtchenko, Alexandre V, Ivanenkov, Yan A, Mitkin, Oleg D, Yamanushkin, Pavel M, Bichko, Vadim V, Shevkun, Natalia A, Karapetian, Ruben N, Leneva, Irina A, Borisova, Olga V, Veselov, Mark S
Published in Journal of antimicrobial chemotherapy (01.07.2014)

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Antagonists of 5-HT6 receptors. Substituted 3-(phenylsulfonyl)pyrazolo[1,5-a]pyrido[3,4-e]pyrimidines and 3-(phenylsulfonyl)pyrazolo[1,5-a]pyrido[4,3-d]pyrimidines—Synthesis and ‘structure–activity’ relationship

Antagonists of 5-HT6 receptors. Substituted 3-(phenylsulfonyl)pyrazolo[1,5-a]pyrido[3,4-e]pyrimidines and 3-(phenylsulfonyl)pyrazolo[1,5-a]pyrido[4,3-d]pyrimidines—Synthesis and ‘structure–activity’ relationship

by Ivachtchenko, Alexandre V., Golovina, Elena S., Kadieva, Madina G., Kysil, Volodymyr M., Mitkin, Oleg D., Vorobiev, Anton A., Okun, Ilya
Published in Bioorganic & medicinal chemistry letters (01.07.2012)

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Novel One-Pot Synthesis of Methyl 4-Hydroxy-2-thioxo-1,2-dihydroquinoline-3-carboxylate: Synthetic and Crystallographic Studies

Novel One-Pot Synthesis of Methyl 4-Hydroxy-2-thioxo-1,2-dihydroquinoline-3-carboxylate: Synthetic and Crystallographic Studies

by Kovalenko, Sergiy M., Drushlyak, Oleksandr G., Konovalova, Irina S., Mariutsa, Illia O., Kravchenko, Dmitry V., Ivachtchenko, Alexandre V., Mitkin, Oleg D.
Published in MolBank (01.12.2019)

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Synthesis, X-ray crystal structure, Hirshfeld surface analysis, and molecular docking study of novel inhibitor of hepatitis B: methyl 4-fluoro-3-(morpholinosulfonyl)benzo[b]thiophene-2-carboxylate

Synthesis, X-ray crystal structure, Hirshfeld surface analysis, and molecular docking study of novel inhibitor of hepatitis B: methyl 4-fluoro-3-(morpholinosulfonyl)benzo[b]thiophene-2-carboxylate

by Ivachtchenko, Alexandre V., Mitkin, Oleg D., Kravchenko, Dmitry V., Kovalenko, Sergiy M., Shishkina, Svitlana V., Bunyatyan, Natalya D., Konovalova, Irina S., Dmitrieva, Irina G., Ivanov, Vladimir V., Langer, Thierry
Published in Heliyon (01.11.2019)

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Discovery of Novel Highly Potent Hepatitis C Virus NS5A Inhibitor (AV4025)

Discovery of Novel Highly Potent Hepatitis C Virus NS5A Inhibitor (AV4025)

by Ivachtchenko, Alexandre V, Mitkin, Oleg D, Yamanushkin, Pavel M, Kuznetsova, Irina V, Bulanova, Elena A, Shevkun, Natalia A, Koryakova, Angela G, Karapetian, Ruben N, Bichko, Vadim V, Trifelenkov, Andrey S, Kravchenko, Dmitry V, Vostokova, Natalia V, Veselov, Mark S, Chufarova, Nina V, Ivanenkov, Yan A
Published in Journal of medicinal chemistry (25.09.2014)

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2-Substituted 5,6-dimethyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines: New series of highly potent and specific serotonin 5-HT6 receptor antagonists

2-Substituted 5,6-dimethyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines: New series of highly potent and specific serotonin 5-HT6 receptor antagonists

by Ivachtchenko, Alexandre V., Golovina, Elena S., Kadieva, Madina G., Koryakova, Angela G., Mitkin, Oleg D., Tkachenko, Sergey E., Kysil, Volodymyr M., Okun, Ilya
Published in European journal of medicinal chemistry (01.04.2011)

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Journal Article

Crystal structure, Hirshfeld analysis and a mol-ecular docking study of a new inhibitor of the Hepatitis B virus (HBV): ethyl 5-methyl-1,1-dioxo-2-{[5-(pentan-3-yl)-1,2,4-oxa-diazol-3-yl]meth-yl}-2H-1,2,6-thia-diazine-4-carboxyl-ate

Crystal structure, Hirshfeld analysis and a mol-ecular docking study of a new inhibitor of the Hepatitis B virus (HBV): ethyl 5-methyl-1,1-dioxo-2-{[5-(pentan-3-yl)-1,2,4-oxa-diazol-3-yl]meth-yl}-2H-1,2,6-thia-diazine-4-carboxyl-ate

by Ivachtchenko, Alexandre V, Kovalenko, Sergiy M, Kravchenko, Dmitry V, Mitkin, Oleg D, Ivanov, Vladimir V, Langer, Thierry
Published in Acta crystallographica. Section E, Crystallographic communications (01.01.2020)

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A novel influenza virus neuraminidase inhibitor AV5027

A novel influenza virus neuraminidase inhibitor AV5027

by Ivachtchenko, Alexandre V., Ivanenkov, Yan A., Mitkin, Oleg D., Yamanushkin, Pavel M., Bichko, Vadim V., Leneva, Irina A., Borisova, Olga V.
Published in Antiviral research (01.12.2013)

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Synthesis, Single Crystal X-Ray Analysis, Prediction and Study of Pharmacological Activity of 4-(1H-Benzo[d]imidazol-2-yl)-1-Phenyl-1H-1,2,3-triazol-5-Amine and Its Solvates

Synthesis, Single Crystal X-Ray Analysis, Prediction and Study of Pharmacological Activity of 4-(1H-Benzo[d]imidazol-2-yl)-1-Phenyl-1H-1,2,3-triazol-5-Amine and Its Solvates

by Ivachtchenko, Alexandre V., Mitkin, Oleg D., Kravchenko, Dmitry V., Kovalenko, Sergiy M., Shishkina, Svitlana V., Bunyatyan, Natalya D., Konovalova, Irina S., Ivanov, Vladimir V., Konovalova, Olena D., Langer, Thierry
Published in Crystals (Basel) (05.12.2019)

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Synthesis and biological evaluation of novel γ-carboline analogues of Dimebon as potent 5-HT6 receptor antagonists

Synthesis and biological evaluation of novel γ-carboline analogues of Dimebon as potent 5-HT6 receptor antagonists

by IVACHTCHENKO, Alexandre V, FROLOV, Eugene B, MITKIN, Oleg D, KYSIL, Volodymyr M, KHVAT, Alexander V, OKUN, Ilya M, TLCACHENKO, Sergey E
Published in Bioorganic & medicinal chemistry letters (15.06.2009)

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