c-Myc Modulation and Acetylation Is a Key HDAC Inhibitor Target in Cancer
Nebbioso, Angela, Carafa, Vincenzo, Conte, Mariarosaria, Tambaro, Francesco Paolo, Abbondanza, Ciro, Martens, Joost, Nees, Matthias, Benedetti, Rosaria, Pallavicini, Isabella, Minucci, Saverio, Garcia-Manero, Guillermo, Iovino, Francesco, Lania, Gabriella, Ingenito, Concetta, Belsito Petrizzi, Valeria, Stunnenberg, Hendrik G, Altucci, Lucia
Published in Clinical cancer research (15.05.2017)
Published in Clinical cancer research (15.05.2017)
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Sex-Based Dimorphism of Anticancer Immune Response and Molecular Mechanisms of Immune Evasion
Conforti, Fabio, Pala, Laura, Pagan, Eleonora, Bagnardi, Vincenzo, De Pas, Tommaso, Queirolo, Paola, Pennacchioli, Elisabetta, Catania, Chiara, Cocorocchio, Emilia, Ferrucci, Pier Francesco, Saponara, Maristella, Orsolini, Gianmarco, Zagami, Paola, Nicoló, Eleonora, De Marinis, Filippo, Tortora, Giampaolo, Bria, Emilio, Minucci, Saverio, Joffe, Hadine, Veronesi, Paolo, Wargo, Jennifer, Rosenthal, Rachel, Swanton, Charles, Mantovani, Alberto, Gelber, Richard D, Viale, Giuseppe, Goldhirsch, Aron, Giaccone, Giuseppe
Published in Clinical cancer research (01.08.2021)
Published in Clinical cancer research (01.08.2021)
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Journal Article
Pharmacological inhibition of LSD1 triggers myeloid differentiation by targeting GSE1 oncogenic functions in AML
Nicosia, Luciano, Boffo, Francesca Ludovica, Ceccacci, Elena, Conforti, Fabio, Pallavicini, Isabella, Bedin, Fabio, Ravasio, Roberto, Massignani, Enrico, Somervaille, Tim C P, Minucci, Saverio, Bonaldi, Tiziana
Published in Oncogene (04.02.2022)
Published in Oncogene (04.02.2022)
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Journal Article
Tuning mTORC1 activity dictates the response of acute myeloid leukemia to LSD1 inhibition
Abdel-Aziz, Amal Kamal, Pallavicini, Isabella, Ceccacci, Elena, Meroni, Giuseppe, Saadeldin, Mona Kamal, Varasi, Mario, Minucci, Saverio
Published in Haematologica (Roma) (01.08.2020)
Published in Haematologica (Roma) (01.08.2020)
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Journal Article
Self-renewal of tumor cells: epigenetic determinants of the cancer stem cell phenotype
Ravasio, Roberto, Ceccacci, Elena, Minucci, Saverio
Published in Current opinion in genetics & development (01.02.2016)
Published in Current opinion in genetics & development (01.02.2016)
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Journal Article
Co-targeting leukemia-initiating cells and leukemia bulk leads to disease eradication
Moretti, Simona, Abdel-Aziz, Amal Kamal, Ceccacci, Elena, Pallavicini, Isabella, Santoro, Fabio, de Thé, Hugues, Minucci, Saverio
Published in Leukemia (01.05.2022)
Published in Leukemia (01.05.2022)
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Journal Article
Interplay between oncogene-induced DNA damage response and heterochromatin in senescence and cancer
Mercurio, Ciro, dal Zuffo, Roberto, Liontos, Michalis, d'Ario, Giovanni, Hahn, William C, Gorgoulis, Vassilis, Dobreva, Miryana, Minucci, Saverio, Sulli, Gabriele, Montani, Erica, d'Adda di Fagagna, Fabrizio, Matti, Valentina, Gargiulo, Gaetano, Di Micco, Raffaella, Botrugno, Oronza A
Published in Nature cell biology (01.03.2011)
Published in Nature cell biology (01.03.2011)
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Journal Article
Surmounting the resistance against EGFR inhibitors through the development of thieno[2,3-d]pyrimidine-based dual EGFR/HER2 inhibitors
Milik, Sandra N., Abdel-Aziz, Amal Kamal, Lasheen, Deena S., Serya, Rabah A.T., Minucci, Saverio, Abouzid, Khaled A.M.
Published in European journal of medicinal chemistry (15.07.2018)
Published in European journal of medicinal chemistry (15.07.2018)
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Journal Article
The Polycomb group proteins bind throughout the INK4A-ARF locus and are disassociated in senescent cells
Bracken, Adrian P, Kleine-Kohlbrecher, Daniela, Dietrich, Nikolaj, Pasini, Diego, Gargiulo, Gaetano, Beekman, Chantal, Theilgaard-Mönch, Kim, Minucci, Saverio, Porse, Bo T, Marine, Jean-Christophe, Hansen, Klaus H, Helin, Kristian
Published in Genes & development (01.03.2007)
Published in Genes & development (01.03.2007)
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Journal Article
Long non‐coding RNA TINCR suppresses metastatic melanoma dissemination by preventing ATF4 translation
Melixetian, Marine, Bossi, Daniela, Mihailovich, Marija, Punzi, Simona, Barozzi, Iros, Marocchi, Federica, Cuomo, Alessandro, Bonaldi, Tiziana, Testa, Giuseppe, Marine, Jean‐Christophe, Leucci, Eleonora, Minucci, Saverio, Pelicci, Pier Giuseppe, Lanfrancone, Luisa
Published in EMBO reports (03.03.2021)
Published in EMBO reports (03.03.2021)
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Journal Article
Differential epigenetic reprogramming in response to specific endocrine therapies promotes cholesterol biosynthesis and cellular invasion
Nguyen, Van T M, Barozzi, Iros, Faronato, Monica, Lombardo, Ylenia, Steel, Jennifer H, Patel, Naina, Darbre, Philippa, Castellano, Leandro, Győrffy, Balázs, Woodley, Laura, Meira, Alba, Patten, Darren K, Vircillo, Valentina, Periyasamy, Manikandan, Ali, Simak, Frige, Gianmaria, Minucci, Saverio, Coombes, R Charles, Magnani, Luca
Published in Nature communications (27.11.2015)
Published in Nature communications (27.11.2015)
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Journal Article
Biochemical, Structural, and Biological Evaluation of Tranylcypromine Derivatives as Inhibitors of Histone Demethylases LSD1 and LSD2
Binda, Claudia, Valente, Sergio, Romanenghi, Mauro, Pilotto, Simona, Cirilli, Roberto, Karytinos, Aristotele, Ciossani, Giuseppe, Botrugno, Oronza A, Forneris, Federico, Tardugno, Maria, Edmondson, Dale E, Minucci, Saverio, Mattevi, Andrea, Mai, Antonello
Published in Journal of the American Chemical Society (19.05.2010)
Published in Journal of the American Chemical Society (19.05.2010)
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Journal Article
Chromatin immunoprecipitation and high-throughput sequencing from paraffin-embedded pathology tissue
Fanelli, Mirco, Amatori, Stefano, Barozzi, Iros, Minucci, Saverio
Published in Nature protocols (01.12.2011)
Published in Nature protocols (01.12.2011)
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Journal Article
Longitudinal single-cell transcriptomics reveals distinct patterns of recurrence in acute myeloid leukemia
Zhai, Yanan, Singh, Prashant, Dolnik, Anna, Brazda, Peter, Atlasy, Nader, del Gaudio, Nunzio, Döhner, Konstanze, Döhner, Hartmut, Minucci, Saverio, Martens, Joost, Altucci, Lucia, Megchelenbrink, Wout, Bullinger, Lars, Stunnenberg, Hendrik G
Published in Molecular cancer (19.08.2022)
Published in Molecular cancer (19.08.2022)
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Journal Article
HDAC-regulated myomiRs control BAF60 variant exchange and direct the functional phenotype of fibro-adipogenic progenitors in dystrophic muscles
Saccone, Valentina, Consalvi, Silvia, Giordani, Lorenzo, Mozzetta, Chiara, Barozzi, Iros, Sandoná, Martina, Ryan, Tammy, Rojas-Muñoz, Agustin, Madaro, Luca, Fasanaro, Pasquale, Borsellino, Giovanna, De Bardi, Marco, Frigè, Gianmaria, Termanini, Alberto, Sun, Xin, Rossant, Janet, Bruneau, Benoit G, Mercola, Mark, Minucci, Saverio, Puri, Pier Lorenzo
Published in Genes & development (15.04.2014)
Published in Genes & development (15.04.2014)
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Journal Article
Discovery of a Novel Inhibitor of Histone Lysine-Specific Demethylase 1A (KDM1A/LSD1) as Orally Active Antitumor Agent
Vianello, Paola, Botrugno, Oronza A, Cappa, Anna, Dal Zuffo, Roberto, Dessanti, Paola, Mai, Antonello, Marrocco, Biagina, Mattevi, Andrea, Meroni, Giuseppe, Minucci, Saverio, Stazi, Giulia, Thaler, Florian, Trifiró, Paolo, Valente, Sergio, Villa, Manuela, Varasi, Mario, Mercurio, Ciro
Published in Journal of medicinal chemistry (25.02.2016)
Published in Journal of medicinal chemistry (25.02.2016)
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