Chemoenzymatic Synthesis of Glycosylated Glucagon-like Peptide 1: Effect of Glycosylation on Proteolytic Resistance and in Vivo Blood Glucose-Lowering Activity
Ueda, Taichi, Tomita, Kazuyoshi, Notsu, Yoshihide, Ito, Takaomi, Fumoto, Masataka, Takakura, Tomoaki, Nagatome, Hirofumi, Takimoto, Akio, Mihara, Shin-Ichi, Togame, Hiroko, Kawamoto, Keiko, Iwasaki, Takanori, Asakura, Kenji, Oshima, Takeo, Hanasaki, Kohji, Nishimura, Shin-Ichiro, Kondo, Hirosato
Published in Journal of the American Chemical Society (06.05.2009)
Published in Journal of the American Chemical Society (06.05.2009)
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Structure−Activity Relationships of a Novel Class of Endothelin-A Receptor Antagonists and Discovery of Potent and Selective Receptor Antagonist, 2-(Benzo[1,3]dioxol-5-yl)-6-isopropyloxy-4-(4-methoxyphenyl)-2H-chromene-3- carboxylic Acid (S-1255). 1. Study on Structure−Activity Relationships and Basic Structure Crucial for ETA Antagonism
Ishizuka, Natsuki, Matsumura, Ken-ichi, Sakai, Katsunori, Fujimoto, Masafumi, Mihara, Shin-ichi, Yamamori, Teruo
Published in Journal of medicinal chemistry (09.05.2002)
Published in Journal of medicinal chemistry (09.05.2002)
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2 -Arylimino -5,6 -dihydro -4H-1,3 -thiazines as a new class of cannabinoid receptor agonists. Part 1 Discovery of CB2 receptor selective compounds
KAI, Hiroyuki, MORIOKA, Yasuhide, ARAI, Tohko, ABE, Kohji, OKABE, Hiroshi, BABA, Takahiko, YOSHIKAWA, Takayoshi, TAKENAKA, Hideyuki, MURASHI, Takami, MORITA, Koichi, SHINONOME, Satomi, NAKAZATO, Hitoshi, KAWAMOTO, Keiko, HANASAKI, Kohji, TAKAHASHI, Fumiyo, MIHARA, Shin-Ichi
Published in Bioorganic & medicinal chemistry letters (15.07.2007)
Published in Bioorganic & medicinal chemistry letters (15.07.2007)
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Synthesis and structure–activity relationships of potent and orally active sulfonamide ETB selective antagonists
Kanda, Yasuhiko, Kawanishi, Yasuyuki, Oda, Katsuo, Sakata, Teruo, Mihara, Shin-ichi, Asakura, Kenji, Kanemasa, Toshiyuki, Ninomiya, Mitsuyoshi, Fujimoto, Masafumi, Konoike, Toshiro
Published in Bioorganic & medicinal chemistry (01.04.2001)
Published in Bioorganic & medicinal chemistry (01.04.2001)
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1,3-Disubstituted Benzazepines as Novel, Potent, Selective Neuropeptide Y Y1 Receptor Antagonists
Murakami, Yasushi, Hara, Hirokazu, Okada, Tetsuo, Hashizume, Hiroshi, Kii, Makoto, Ishihara, Yasunobu, Ishikawa, Michio, Shimamura, Mayumi, Mihara, Shin-inchi, Kato, Goro, Hanasaki, Kohji, Hagishita, Sanji, Fujimoto, Masafumi
Published in Journal of medicinal chemistry (15.07.1999)
Published in Journal of medicinal chemistry (15.07.1999)
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A novel non-peptide endothelin antagonist isolated from bayberry, Myrica cerifera
Fujimoto, Masafumi, Mihara, Shin-ichi, Nakajima, Shigeyuki, Ueda, Motohiko, Nakamura, Miharu, Sakurai, Ken-suke
Published in FEBS letters (22.06.1992)
Published in FEBS letters (22.06.1992)
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