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Published in Proceedings of the National Academy of Sciences - PNAS (01.09.2020)
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Human serotonin1B receptor expression in Sf9 cells: Phosphorylation, palmitoylation, and adenylyl cyclase inhibition
Ng, Gordon YK, George, Susan R., Zastawny, Roman L., Caron, Mireille, Bouvier, Michel, Dennis, Michael, O'Dowd, Brian F.
Published in Biochemistry (Easton) (02.11.1993)
Published in Biochemistry (Easton) (02.11.1993)
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Distinct conformations of GPCR–β-arrestin complexes mediate desensitization, signaling, and endocytosis
Cahill, Thomas J., Thomsen, Alex R. B., Tarrasch, Jeffrey T., Plouffe, Bianca, Nguyen, Anthony H., Yang, Fan, Huang, Li-Yin, Kahsai, Alem W., Bassoni, Daniel L., Gavino, Bryant J., Lamerdin, Jane E., Triest, Sarah, Shukla, Arun K., Berger, Benjamin, Little, John, Antar, Albert, Blanc, Adi, Qu, Chang-Xiu, Chen, Xin, Kawakami, Kouki, Inoue, Asuka, Aoki, Junken, Steyaert, Jan, Sun, Jin-Peng, Bouvier, Michel, Skiniotis, Georgios, Lefkowitz, Robert J.
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Published in Proceedings of the National Academy of Sciences - PNAS (07.03.2017)
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Abstract C111: Characterization of kisspeptin receptor signaling pathways in cervical cancer: Unveiling novel mechanisms and therapeutic potentials
Rodríguez-Sarmiento, Deisy Y., Scarpelli-Pereira, Pedro H., Bouvier, Michel
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Manifold roles of β-arrestins in GPCR signaling elucidated with siRNA and CRISPR/Cas9
Luttrell, Louis M, Wang, Jialu, Plouffe, Bianca, Smith, Jeffrey S, Yamani, Lama, Kaur, Suneet, Jean-Charles, Pierre-Yves, Gauthier, Christophe, Lee, Mi-Hye, Pani, Biswaranjan, Kim, Jihee, Ahn, Seungkirl, Rajagopal, Sudarshan, Reiter, Eric, Bouvier, Michel, Shenoy, Sudha K, Laporte, Stéphane A, Rockman, Howard A, Lefkowitz, Robert J
Published in Science signaling (25.09.2018)
Published in Science signaling (25.09.2018)
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Structural insights into binding specificity, efficacy and bias of a β2AR partial agonist
Masureel, Matthieu, Zou, Yaozhong, Picard, Louis-Philippe, van der Westhuizen, Emma, Mahoney, Jacob P., Rodrigues, João P. G. L. M., Mildorf, Thomas J., Dror, Ron O., Shaw, David E., Bouvier, Michel, Pardon, Els, Steyaert, Jan, Sunahara, Roger K., Weis, William I., Zhang, Cheng, Kobilka, Brian K.
Published in Nature chemical biology (01.11.2018)
Published in Nature chemical biology (01.11.2018)
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Structure-based discovery of nonopioid analgesics acting through the α2A-adrenergic receptor
Fink, Elissa A, Xu, Jun, Hübner, Harald, Braz, Joao M, Seemann, Philipp, Avet, Charlotte, Craik, Veronica, Weikert, Dorothee, Schmidt, Maximilian F, Webb, Chase M, Tolmachova, Nataliya A, Moroz, Yurii S, Xi-Ping Huang, Kalyanaraman, Chakrapani, Gahbauer, Stefan, Chen, Geng, Liu, Zheng, Jacobson, Matthew P, Irwin, John J, Bouvier, Michel, Du, Yang, Shoichet, Brian K, Basbaum, Allan I, Gmeiner, Peter
Published in Science (American Association for the Advancement of Science) (30.09.2022)
Published in Science (American Association for the Advancement of Science) (30.09.2022)
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Inhibitors that stabilize a closed RAF kinase domain conformation induce dimerization
Lavoie, Hugo, Thevakumaran, Neroshan, Gavory, Gwenaëlle, Li, John J, Padeganeh, Abbas, Guiral, Sébastien, Duchaine, Jean, Mao, Daniel Y L, Bouvier, Michel, Sicheri, Frank, Therrien, Marc
Published in Nature chemical biology (01.07.2013)
Published in Nature chemical biology (01.07.2013)
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Translating biased signaling in the ghrelin receptor system into differential in vivo functions
Mende, Franziska, Hundahl, Cecilie, Plouffe, Bianca, Skov, Louise Julie, Sivertsen, Bjørn, Madsen, Andreas Nygaard, Lückmann, Michael, Diep, Thi Ai, Offermanns, Stefan, Frimurer, Thomas Michael, Bouvier, Michel, Holst, Birgitte
Published in Proceedings of the National Academy of Sciences - PNAS (23.10.2018)
Published in Proceedings of the National Academy of Sciences - PNAS (23.10.2018)
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G protein selectivity profile of GPR56/ADGRG1 and its effect on downstream effectors
Jallouli, Raida, Moreno-Salinas, Ana L., Laniel, Andréanne, Holleran, Brian, Avet, Charlotte, Jacob, Joan, Hoang, Trang, Lavoie, Christine, Carmon, Kendra S., Bouvier, Michel, Leduc, Richard
Published in Cellular and molecular life sciences : CMLS (01.12.2024)
Published in Cellular and molecular life sciences : CMLS (01.12.2024)
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KCTD Hetero-oligomers Confer Unique Kinetic Properties on Hippocampal GABAB Receptor-Induced K+ Currents
Fritzius, Thorsten, Turecek, Rostislav, Seddik, Riad, Kobayashi, Hiroyuki, Tiao, Jim, Rem, Pascal D, Metz, Michaela, Kralikova, Michaela, Bouvier, Michel, Gassmann, Martin, Bettler, Bernhard
Published in The Journal of neuroscience (01.02.2017)
Published in The Journal of neuroscience (01.02.2017)
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Differential β-arrestin-dependent conformational signaling and cellular responses revealed by angiotensin analogs
Zimmerman, Brandon, Beautrait, Alexandre, Aguila, Benjamin, Charles, Ricardo, Escher, Emanuel, Claing, Audrey, Bouvier, Michel, Laporte, Stéphane A
Published in Science signaling (24.04.2012)
Published in Science signaling (24.04.2012)
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BRET-based effector membrane translocation assay monitors GPCR-promoted and endocytosis-mediated Gq activation at early endosomes
Wright, Shane C., Lukasheva, Viktoriya, Le Gouill, Christian, Kobayashi, Hiroyuki, Breton, Billy, Mailhot-Larouche, Samuel, Blondel-Tepaz, Élodie, Vieira, Nichelle Antunes, Costa-Neto, Claudio, Héroux, Madeleine, Lambert, Nevin A., Parreiras-e-Silva, Lucas Tabajara, Bouvier, Michel
Published in Proceedings of the National Academy of Sciences - PNAS (18.05.2021)
Published in Proceedings of the National Academy of Sciences - PNAS (18.05.2021)
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Apelin protects against abdominal aortic aneurysm and the therapeutic role of neutral endopeptidase resistant apelin analogs
Wang, Wang, Shen, Mengcheng, Fischer, Conrad, Basu, Ratnadeep, Hazra, Saugata, Couvineau, Pierre, Paul, Manish, Wang, Faqi, Toth, Sandra, Mix, Doran S., Poglitsch, Marko, Gerard, Norma P., Bouvier, Michel, Vederas, John C., Penninger, Josef M., Kassiri, Zamaneh, Oudit, Gavin Y.
Published in Proceedings of the National Academy of Sciences - PNAS (25.06.2019)
Published in Proceedings of the National Academy of Sciences - PNAS (25.06.2019)
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BRET analysis of GPCR oligomerization: newer does not mean better
Bouvier, Michel, Heveker, Nikolaus, Jockers, Ralf, Marullo, Stefano, Milligan, Graeme
Published in Nature methods (01.01.2007)
Published in Nature methods (01.01.2007)
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Biased Signaling Favoring Gi over β-Arrestin Promoted by an Apelin Fragment Lacking the C-terminal Phenylalanine
Ceraudo, Emilie, Galanth, Cécile, Carpentier, Eric, Banegas-Font, Inmaculada, Schonegge, Anne-Marie, Alvear-Perez, Rodrigo, Iturrioz, Xavier, Bouvier, Michel, Llorens-Cortes, Catherine
Published in The Journal of biological chemistry (01.08.2014)
Published in The Journal of biological chemistry (01.08.2014)
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