Search Results - "MICHAEL VAN ZANDT" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Discovery of N‑Substituted 3‑Amino-4-(3-boronopropyl)pyrrolidine-3-carboxylic Acids as Highly Potent Third-Generation Inhibitors of Human Arginase I and II

Discovery of N‑Substituted 3‑Amino-4-(3-boronopropyl)pyrrolidine-3-carboxylic Acids as Highly Potent Third-Generation Inhibitors of Human Arginase I and II

by Van Zandt, Michael C, Jagdmann, G. Erik, Whitehouse, Darren L, Ji, Minkoo, Savoy, Jennifer, Potapova, Olga, Cousido-Siah, Alexandra, Mitschler, Andre, Howard, Eduardo I, Pyle, Anna Marie, Podjarny, Alberto D
Published in Journal of medicinal chemistry (12.09.2019)

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Journal Article

Chemical Synthesis and Characterization of Epicatechin Glucuronides and Sulfates: Bioanalytical Standards for Epicatechin Metabolite Identification

Chemical Synthesis and Characterization of Epicatechin Glucuronides and Sulfates: Bioanalytical Standards for Epicatechin Metabolite Identification

by Zhang, Mingbao, Jagdmann, G. Erik, Van Zandt, Michael, Sheeler, Ryan, Beckett, Paul, Schroeter, Hagen
Published in Journal of natural products (Washington, D.C.) (22.02.2013)

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Journal Article

The antimalarial activity of the pantothenamide α-PanAm is via inhibition of pantothenate phosphorylation

The antimalarial activity of the pantothenamide α-PanAm is via inhibition of pantothenate phosphorylation

by Chiu, Joy E., Thekkiniath, Jose, Choi, Jae-Yeon, Perrin, Benjamin A., Lawres, Lauren, Plummer, Mark, Virji, Azan Z., Abraham, Amanah, Toh, Justin Y., Zandt, Michael Van, Aly, Ahmed S. I., Voelker, Dennis R., Mamoun, Choukri Ben
Published in Scientific reports (27.10.2017)

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Discovery of (R)‑2-Amino-6-borono-2-(2-(piperidin-1-yl)ethyl)hexanoic Acid and Congeners As Highly Potent Inhibitors of Human Arginases I and II for Treatment of Myocardial Reperfusion Injury

Discovery of (R)‑2-Amino-6-borono-2-(2-(piperidin-1-yl)ethyl)hexanoic Acid and Congeners As Highly Potent Inhibitors of Human Arginases I and II for Treatment of Myocardial Reperfusion Injury

by Van Zandt, Michael C, Whitehouse, Darren L, Golebiowski, Adam, Ji, Min Koo, Zhang, Mingbao, Beckett, R. Paul, Jagdmann, G. Erik, Ryder, Todd R, Sheeler, Ryan, Andreoli, Monica, Conway, Bruce, Mahboubi, Keyvan, D’Angelo, Gerard, Mitschler, Andre, Cousido-Siah, Alexandra, Ruiz, Francesc X, Howard, Eduardo I, Podjarny, Alberto D, Schroeter, Hagen
Published in Journal of medicinal chemistry (28.03.2013)

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Discovery of 3-[(4,5,7-Trifluorobenzothiazol-2-yl)methyl]indole-N-acetic Acid (Lidorestat) and Congeners as Highly Potent and Selective Inhibitors of Aldose Reductase for Treatment of Chronic Diabetic Complications

Discovery of 3-[(4,5,7-Trifluorobenzothiazol-2-yl)methyl]indole-N-acetic Acid (Lidorestat) and Congeners as Highly Potent and Selective Inhibitors of Aldose Reductase for Treatment of Chronic Diabetic Complications

by Van Zandt, Michael C, Jones, Michael L, Gunn, David E, Geraci, Leo S, Jones, J. Howard, Sawicki, Diane R, Sredy, Janet, Jacot, Jorge L, DiCioccio, A. Thomas, Petrova, Tatiana, Mitschler, Andre, Podjarny, Alberto D
Published in Journal of medicinal chemistry (05.05.2005)

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Journal Article

Small molecules that target group II introns are potent antifungal agents

Small molecules that target group II introns are potent antifungal agents

by Fedorova, Olga, Jagdmann, G. Erik, Adams, Rebecca L., Yuan, Lin, Van Zandt, Michael C., Pyle, Anna Marie
Published in Nature chemical biology (01.12.2018)

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Journal Article

Editing N-Glycan Site Occupancy with Small-Molecule Oligosaccharyltransferase Inhibitors

Editing N-Glycan Site Occupancy with Small-Molecule Oligosaccharyltransferase Inhibitors

by Rinis, Natalia, Golden, Jennifer E, Marceau, Caleb D, Carette, Jan E, Van Zandt, Michael C, Gilmore, Reid, Contessa, Joseph N
Published in Cell chemical biology (18.10.2018)

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Discovery of [3-(4,5,7-trifluoro-benzothiazol-2-ylmethyl)-pyrrolo[2,3-b] pyridin-1-yl]acetic acids as highly potent and selective inhibitors of aldose reductase for treatment of chronic diabetic complications

Discovery of [3-(4,5,7-trifluoro-benzothiazol-2-ylmethyl)-pyrrolo[2,3-b] pyridin-1-yl]acetic acids as highly potent and selective inhibitors of aldose reductase for treatment of chronic diabetic complications

by VAN ZANDT, Michael C, DOAN, Brian, SAWICKI, Diane R, SREDY, Janet, PODJARNY, Alberto D
Published in Bioorganic & medicinal chemistry letters (01.04.2009)

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Journal Article

Topical application of aminoglycoside antibiotics enhances host resistance to viral infections in a microbiota-independent manner

Topical application of aminoglycoside antibiotics enhances host resistance to viral infections in a microbiota-independent manner

by Gopinath, Smita, Kim, Myoungjoo V., Rakib, Tasfia, Wong, Patrick W., van Zandt, Michael, Barry, Natasha A., Kaisho, Tsuneyasu, Goodman, Andrew L., Iwasaki, Akiko
Published in Nature microbiology (01.05.2018)

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Journal Article

Crystal Structure of Schistosoma mansoni Arginase, a Potential Drug Target for the Treatment of Schistosomiasis

Crystal Structure of Schistosoma mansoni Arginase, a Potential Drug Target for the Treatment of Schistosomiasis

by Hai, Yang, Edwards, Jennifer E, Van Zandt, Michael C, Hoffmann, Karl F, Christianson, David W
Published in Biochemistry (Easton) (22.07.2014)

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Journal Article

Enantioselective synthesis of orthogonally protected (2R,3R)-(−)-epicatechin derivatives, key intermediates in the de novo chemical synthesis of (−)-epicatechin glucuronides and sulfates

Enantioselective synthesis of orthogonally protected (2R,3R)-(−)-epicatechin derivatives, key intermediates in the de novo chemical synthesis of (−)-epicatechin glucuronides and sulfates

by Zhang, Mingbao, Erik Jagdmann, G., Van Zandt, Michael, Beckett, Paul, Schroeter, Hagen
Published in Tetrahedron: asymmetry (15.04.2013)

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Journal Article

Design and synthesis of highly potent and selective (2-arylcarbamoyl-phenoxy)-acetic acid inhibitors of aldose reductase for treatment of chronic diabetic complications

Design and synthesis of highly potent and selective (2-arylcarbamoyl-phenoxy)-acetic acid inhibitors of aldose reductase for treatment of chronic diabetic complications

by Van Zandt, Michael C., Sibley, Evelyn O., McCann, Erin E., Combs, Kerry J., Flam, Brenda, Sawicki, Diane R., Sabetta, Al, Carrington, Anne, Sredy, Janet, Howard, Eduardo, Mitschler, Andre, Podjarny, Alberto D.
Published in Bioorganic & medicinal chemistry (01.11.2004)

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Journal Article

COMPOSITIONS AND METHODS FOR INHIBITING ARGINASE ACTIVITY

COMPOSITIONS AND METHODS FOR INHIBITING ARGINASE ACTIVITY

by ERIC B SJOGREN, DARREN WHITEHOUSE, MICHAEL VAN ZANDT, JIM LI
Year of Publication 20.05.2021

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Patent

Discovery of a Series of Potent, Selective, and Orally Bioavailable Nucleoside Inhibitors of CD73 That Demonstrates In Vivo Antitumor Activity

Discovery of a Series of Potent, Selective, and Orally Bioavailable Nucleoside Inhibitors of CD73 That Demonstrates In Vivo Antitumor Activity

by Li, Jim, Chen, Lijing, Billedeau, Roland J., Stanton, Timothy F., Chiang, John T. P., Lee, Clarissa C., Li, Weiqun, Steggerda, Susanne, Emberley, Ethan, Gross, Matthew, Bhupathi, Deepthi, Che, Xiaoying, Chen, Jason, Dang, Rosalyn, Huang, Tony, Ma, Yong, MacKinnon, Andrew, Makkouk, Amani, Marguier, Gisele, Neou, Silinda, Sotirovska, Natalija, Spurlock, Sandra, Zhang, Jing, Zhang, Winter, van Zandt, Michael, Yuan, Lin, Savoy, Jennifer, Parlati, Francesco, Sjogren, Eric B.
Published in Journal of medicinal chemistry (12.01.2023)

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Journal Article

Synthesis of quaternary α-amino acid-based arginase inhibitors via the Ugi reaction

Synthesis of quaternary α-amino acid-based arginase inhibitors via the Ugi reaction

by Golebiowski, Adam, Whitehouse, Darren, Beckett, R. Paul, Van Zandt, Michael, Ji, Min Koo, Ryder, Todd R., Jagdmann, Erik, Andreoli, Monica, Lee, Yung, Sheeler, Ryan, Conway, Bruce, Olczak, Jacek, Mazur, Marzena, Czestkowski, Wojciech, Piotrowska, Wieslawa, Cousido-Siah, Alexandra, Ruiz, Francesc X., Mitschler, Andre, Podjarny, Alberto, Schroeter, Hagen
Published in Bioorganic & medicinal chemistry letters (01.09.2013)

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Journal Article

A versatile approach to the regioselective synthesis of diverse (−)-epicatechin-β-d-glucuronides

A versatile approach to the regioselective synthesis of diverse (−)-epicatechin-β-d-glucuronides

by Mull, Eric S., Van Zandt, Michael, Golebiowski, Adam, Beckett, R. Paul, Sharma, Pradeep K., Schroeter, Hagen
Published in Tetrahedron letters (21.03.2012)

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Journal Article

2-Substituted-2-amino-6-boronohexanoic acids as arginase inhibitors

2-Substituted-2-amino-6-boronohexanoic acids as arginase inhibitors

by Golebiowski, Adam, Paul Beckett, R., Van Zandt, Michael, Ji, Min Koo, Whitehouse, Darren, Ryder, Todd R., Jagdmann, Erik, Andreoli, Monica, Mazur, Adam, Padmanilayam, Manyian, Cousido-Siah, Alexandra, Mitschler, Andre, Ruiz, Francesc X., Podjarny, Alberto, Schroeter, Hagen
Published in Bioorganic & medicinal chemistry letters (01.04.2013)

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Journal Article

Chemoenzymic Synthesis of 4-Substituted Riboses. S-(4'-Methyladenosyl)-L-homocysteine

Chemoenzymic Synthesis of 4-Substituted Riboses. S-(4'-Methyladenosyl)-L-homocysteine

by Johnson, Carl R, Esker, John L, Van Zandt, Michael C
Published in Journal of organic chemistry (01.10.1994)

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Journal Article

How to Avoid Title Fraud on Your Property

How to Avoid Title Fraud on Your Property

by Van Zandt, Michael J
Published in The Voice of Experience (01.10.2022)

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Newsletter

Discovery of [3-(4,5,7-trifluoro-benzothiazol-2-ylmethyl)-pyrrolo[2,3-b]pyridin -1-yl]ace tic acids as highly potent and selective inhibitors of aldose reductase for treatment of chronic diabetic complications

Discovery of [3-(4,5,7-trifluoro-benzothiazol-2-ylmethyl)-pyrrolo[2,3-b]pyridin -1-yl]ace tic acids as highly potent and selective inhibitors of aldose reductase for treatment of chronic diabetic complications

by Van Zandt, Michael C, Doan, Brian, Sawicki, Diane R, Sredy, Janet, Podjarny, Alberto D
Published in Bioorganic & medicinal chemistry letters (01.04.2009)

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