Discovery of the pan-genotypic hepatitis C virus NS3/4A protease inhibitor voxilaprevir (GS-9857): A component of Vosevi
Taylor, James G., Zipfel, Sheila, Ramey, Kyla, Vivian, Randy, Schrier, Adam, Karki, Kapil K., Katana, Ashley, Kato, Darryl, Kobayashi, Tetsuya, Martinez, Ruben, Sangi, Michael, Siegel, Dustin, Tran, Chinh V., Yang, Zheng-Yu, Zablocki, Jeff, Yang, Cheng Y., Wang, Yujin, Wang, Kelly, Chan, Katie, Barauskas, Ona, Cheng, Guofeng, Jin, Debi, Schultz, Brian E., Appleby, Todd, Villaseñor, Armando G., Link, John O.
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
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Journal Article
Discovery of an Oral Respiratory Syncytial Virus (RSV) Fusion Inhibitor (GS-5806) and Clinical Proof of Concept in a Human RSV Challenge Study
Mackman, Richard L, Sangi, Michael, Sperandio, David, Parrish, Jay P, Eisenberg, Eugene, Perron, Michel, Hui, Hon, Zhang, Lijun, Siegel, Dustin, Yang, Hai, Saunders, Oliver, Boojamra, Constantine, Lee, Gary, Samuel, Dharmaraj, Babaoglu, Kerim, Carey, Anne, Gilbert, Brian E, Piedra, Pedro A, Strickley, Robert, Iwata, Quynh, Hayes, Jaclyn, Stray, Kirsten, Kinkade, April, Theodore, Dorothy, Jordan, Robert, Desai, Manoj, Cihlar, Tomas
Published in Journal of medicinal chemistry (26.02.2015)
Published in Journal of medicinal chemistry (26.02.2015)
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Discovery of N‑[4-[6-tert-Butyl-5-methoxy-8-(6-methoxy-2-oxo‑1H‑pyridin-3-yl)-3-quinolyl]phenyl]methanesulfonamide (RG7109), a Potent Inhibitor of the Hepatitis C Virus NS5B Polymerase
Talamas, Francisco X., Abbot, Sarah C., Anand, Shalini, Brameld, Ken A., Carter, David S., Chen, Jun, Davis, Dana, de Vicente, Javier, Fung, Amy D., Gong, Leyi, Harris, Seth F., Inbar, Petra, Labadie, Sharada S., Lee, Eun K., Lemoine, Remy, Le Pogam, Sophie, Leveque, Vincent, Li, Jim, McIntosh, Joel, Nájera, Isabel, Park, Jaehyeon, Railkar, Aruna, Rajyaguru, Sonal, Sangi, Michael, Schoenfeld, Ryan C., Staben, Leanna R., Tan, Yunchou, Taygerly, Joshua P., Villaseñor, Armando G., Weller, Paul E.
Published in Journal of medicinal chemistry (13.03.2014)
Published in Journal of medicinal chemistry (13.03.2014)
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GS-5806 Inhibits a Broad Range of Respiratory Syncytial Virus Clinical Isolates by Blocking the Virus-Cell Fusion Process
Perron, Michel, Stray, Kirsten, Kinkade, April, Theodore, Dorothy, Lee, Gary, Eisenberg, Eugene, Sangi, Michael, Gilbert, Brian E, Jordan, Robert, Piedra, Pedro A, Toms, Geoffery L, Mackman, Richard, Cihlar, Tomas
Published in Antimicrobial agents and chemotherapy (01.03.2016)
Published in Antimicrobial agents and chemotherapy (01.03.2016)
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Journal Article
Discovery of a Potent and Orally Bioavailable Cyclophilin Inhibitor Derived from the Sanglifehrin Macrocycle
Mackman, Richard L, Steadman, Victoria A, Dean, David K, Jansa, Petr, Poullennec, Karine G, Appleby, Todd, Austin, Carol, Blakemore, Caroline A, Cai, Ruby, Cannizzaro, Carina, Chin, Gregory, Chiva, Jean-Yves C, Dunbar, Neil A, Fliri, Hans, Highton, Adrian J, Hui, Hon, Ji, Mingzhe, Jin, Haolun, Karki, Kapil, Keats, Andrew J, Lazarides, Linos, Lee, Yu-Jen, Liclican, Albert, Mish, Michael, Murray, Bernard, Pettit, Simon B, Pyun, Peter, Sangi, Michael, Santos, Rex, Sanvoisin, Jonathan, Schmitz, Uli, Schrier, Adam, Siegel, Dustin, Sperandio, David, Stepan, George, Tian, Yang, Watt, Gregory M, Yang, Hai, Schultz, Brian E
Published in Journal of medicinal chemistry (08.11.2018)
Published in Journal of medicinal chemistry (08.11.2018)
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Journal Article
Discovery of a Novel Series of Potent Non-Nucleoside Inhibitors of Hepatitis C Virus NS5B
Schoenfeld, Ryan C, Bourdet, David L, Brameld, Ken A, Chin, Elbert, de Vicente, Javier, Fung, Amy, Harris, Seth F, Lee, Eun K, Le Pogam, Sophie, Leveque, Vincent, Li, Jim, Lui, Alfred S.-T, Najera, Isabel, Rajyaguru, Sonal, Sangi, Michael, Steiner, Sandra, Talamas, Francisco X, Taygerly, Joshua P, Zhao, Junping
Published in Journal of medicinal chemistry (24.10.2013)
Published in Journal of medicinal chemistry (24.10.2013)
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PYRAZOLO [1, 5-a] PYRIMIDINES AS ANTIVIRAL AGENTS
HUI HON CHUNG, YAN HAI, KERIM BABAOGLU, OLIVER L SAUNDERS, BOOJAMRA CONSTANTINE G, EISENBERG EUGENE J, JAY P PARRISH, MACKMAN RICHARD L, MICHAEL SANGI, DAVID SPERANDIO, DUSTIN SIEGEL
Year of Publication 16.04.2020
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Year of Publication 16.04.2020
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COMPOUNDS AND METHODS FOR ANTIVIRAL TREATMENT
HUI HON CHUNG, JAY P PARRISH, MACKMAN RICHARD L, MICHAEL SANGI, DAVID SPERANDIO, YANG HAI, DUSTIN SIEGEL
Year of Publication 21.06.2018
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Year of Publication 21.06.2018
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INHIBITORS OF HEPATITIS C VIRUS
KAPIL KUMAR KARKI, ZABLOCKI JEFF, JAMES G TAYLOR, YANG ZHENG-YU, VIVIAN RANDALL W, BARTON W PHILLIPS, KOBAYASHI TETSUYA, JEROMY J COTTELL, SHEILA ZIPFEL, DARRYL KATO, ASHLEY ANNE KATANA, JOHN O LINK, TERESA ALEJANDRA TREJO MARTIN, KYLA BJORNSON, RUBEN MARTINEZ, MICHAEL SANGI, EDA CANALES, HYUNG-JUNG PYUN, TRAN CHINH VIET, ADAM JAMES SCHRIER, DUSTIN SIEGEL
Year of Publication 10.09.2020
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Year of Publication 10.09.2020
Patent
COMPOUNDS AND METHODS FOR ANTIVIRAL TREATMENT
HUI HON CHUNG, JAY P PARRISH, MACKMAN RICHARD L, MICHAEL SANGI, DAVID SPERANDIO, YANG HAI, DUSTIN SIEGEL
Year of Publication 27.07.2017
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Year of Publication 27.07.2017
Patent
PYRAZOLO[1,5-A]PYRIMIDINE AS ANTIVIRAL AGENT
HUI HON CHUNG, BOOJAMRA CONSTANTINE G, JAY P PARRISH, PETR JANSA, MACKMAN RICHARD L, MICHAEL SANGI, DAVID SPERANDIO, YANG HAI, DUSTIN SIEGEL
Year of Publication 16.02.2017
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Year of Publication 16.02.2017
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PYRAZOLO[1,5-A]PYRIMIDINES AS ANTIVIRAL AGENT
HUI HON CHUNG, YAN HAI, KERIM BABAOGLU, OLIVER L SAUNDERS, BOOJAMRA CONSTANTINE G, EISENBERG EUGENE J, JAY P PARRISH, MACKMAN RICHARD L, MICHAEL SANGI, DAVID SPERANDIO, DUSTIN SIEGEL
Year of Publication 26.01.2017
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Year of Publication 26.01.2017
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HEPATITIS C VIRUS INHIBITOR
KAPIL KUMAR KARKI, ZABLOCKI JEFF, JAMES G TAYLOR, YANG ZHENG-YU, VIVIAN RANDALL W, BARTON W PHILLIPS, KOBAYASHI TETSUYA, JEROMY J COTTELL, SHEILA ZIPFEL, DARRYL KATO, ASHLEY ANNE KATANA, JOHN O LINK, TERESA ALEJANDRA TREJO MARTIN, KYLA BJORNSON, RUBEN MARTINEZ, MICHAEL SANGI, EDA CANALES, HYUNG-JUNG PYUN, TRAN CHINH VIET, ADAM JAMES SCHRIER, DUSTIN SIEGEL
Year of Publication 04.10.2018
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Year of Publication 04.10.2018
Patent
PYRAZOLO[1,5-A]PYRIMIDINES AS ANTIVIRAL AGENT
HUI HON CHUNG, YAN HAI, KERIM BABAOGLU, OLIVER L SAUNDERS, BOOJAMRA CONSTANTINE G, EISENBERG EUGENE J, JAY P PARRISH, MACKMAN RICHARD L, MICHAEL SANGI, DAVID SPERANDIO, DUSTIN SIEGEL
Year of Publication 07.12.2015
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Year of Publication 07.12.2015
Patent
INHIBITORS OF HEPATITIS C VIRUS
KAPIL KUMAR KARKI, ZABLOCKI JEFF, JAMES G TAYLOR, YANG ZHENG-YU, VIVIAN RANDALL W, BARTON W PHILLIPS, KOBAYASHI TETSUYA, JEROMY J COTTELL, SHEILA ZIPFEL, DARRYL KATO, ASHLEY ANNE KATANA, JOHN O LINK, TERESA ALEJANDRA TREJO MARTIN, KYLA BJORNSON, RUBEN MARTINEZ, MICHAEL SANGI, EDA CANALES, HYUNG-JUNG PYUN, TRAN CHINH VIET, ADAM JAMES SCHRIER, DUSTIN SIEGEL
Year of Publication 31.03.2016
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Year of Publication 31.03.2016
Patent
Sulfinylaminobenzamide and sulfonylaminobenzamide derivatives
Sangi, Michael, Sperandio, David, Notte, Gregory, Farand, Julie, Kaplan, Joshua A, Olen, Casey Lockwood
Year of Publication 01.08.2024
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Year of Publication 01.08.2024
Patent
Sulfinylaminobenzamide and sulfonylaminobenzamide derivatives
Sangi, Michael, Sperandio, David, Notte, Gregory, Farand, Julie, Kaplan, Joshua A, Olen, Casey Lockwood
Year of Publication 30.07.2024
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Year of Publication 30.07.2024
Patent
SULFONYLAMINOBENZAMIDE DERIVATIVES
FARAND, Julie, KAPLAN, Joshua A, SPERANDIO, David, OLEN, Casey Lockwood, SANGI, Michael, NOTTE, Gregory
Year of Publication 28.04.2024
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Year of Publication 28.04.2024
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