Mechanisms of ketamine and its metabolites as antidepressants
Hess, Evan M., Riggs, Lace M., Michaelides, Michael, Gould, Todd D.
Published in Biochemical pharmacology (01.03.2022)
Published in Biochemical pharmacology (01.03.2022)
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Chemogenetics revealed: DREADD occupancy and activation via converted clozapine
Gomez, Juan L., Bonaventura, Jordi, Lesniak, Wojciech, Mathews, William B., Sysa-Shah, Polina, Rodriguez, Lionel A., Ellis, Randall J., Richie, Christopher T., Harvey, Brandon K., Dannals, Robert F., Pomper, Martin G., Bonci, Antonello, Michaelides, Michael
Published in Science (American Association for the Advancement of Science) (04.08.2017)
Published in Science (American Association for the Advancement of Science) (04.08.2017)
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The Histone Methyltransferase Inhibitor A-366 Uncovers a Role for G9a/GLP in the Epigenetics of Leukemia
Pappano, William N, Guo, Jun, He, Yupeng, Ferguson, Debra, Jagadeeswaran, Sujatha, Osterling, Donald J, Gao, Wenqing, Spence, Julie K, Pliushchev, Marina, Sweis, Ramzi F, Buchanan, Fritz G, Michaelides, Michael R, Shoemaker, Alexander R, Tse, Chris, Chiang, Gary G
Published in PloS one (06.07.2015)
Published in PloS one (06.07.2015)
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Pharmacological and behavioral divergence of ketamine enantiomers: implications for abuse liability
Bonaventura, Jordi, Lam, Sherry, Carlton, Meghan, Boehm, Matthew A., Gomez, Juan L., Solís, Oscar, Sánchez-Soto, Marta, Morris, Patrick J., Fredriksson, Ida, Thomas, Craig J., Sibley, David R., Shaham, Yavin, Zarate, Carlos A., Michaelides, Michael
Published in Molecular psychiatry (01.11.2021)
Published in Molecular psychiatry (01.11.2021)
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Discovery of a selective catalytic p300/CBP inhibitor that targets lineage-specific tumours
Lasko, Loren M., Jakob, Clarissa G., Edalji, Rohinton P., Qiu, Wei, Montgomery, Debra, Digiammarino, Enrico L., Hansen, T. Matt, Risi, Roberto M., Frey, Robin, Manaves, Vlasios, Shaw, Bailin, Algire, Mikkel, Hessler, Paul, Lam, Lloyd T., Uziel, Tamar, Faivre, Emily, Ferguson, Debra, Buchanan, Fritz G., Martin, Ruth L., Torrent, Maricel, Chiang, Gary G., Karukurichi, Kannan, Langston, J. William, Weinert, Brian T., Choudhary, Chunaram, de Vries, Peter, Kluge, Arthur F., Patane, Michael A., Van Drie, John H., Wang, Ce, McElligott, David, Kesicki, Ed, Marmorstein, Ronen, Sun, Chaohong, Cole, Philip A., Rosenberg, Saul H., Michaelides, Michael R., Lai, Albert, Bromberg, Kenneth D.
Published in Nature (London) (05.10.2017)
Published in Nature (London) (05.10.2017)
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Ultrapotent chemogenetics for research and potential clinical applications
Magnus, Christopher J, Lee, Peter H, Bonaventura, Jordi, Zemla, Roland, Gomez, Juan L, Ramirez, Melissa H, Hu, Xing, Galvan, Adriana, Basu, Jayeeta, Michaelides, Michael, Sternson, Scott M
Published in Science (American Association for the Advancement of Science) (12.04.2019)
Published in Science (American Association for the Advancement of Science) (12.04.2019)
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High-potency ligands for DREADD imaging and activation in rodents and monkeys
Bonaventura, Jordi, Eldridge, Mark A. G., Hu, Feng, Gomez, Juan L., Sanchez-Soto, Marta, Abramyan, Ara M., Lam, Sherry, Boehm, Matthew A., Ruiz, Christina, Farrell, Mitchell R., Moreno, Andrea, Galal Faress, Islam Mustafa, Andersen, Niels, Lin, John Y., Moaddel, Ruin, Morris, Patrick J., Shi, Lei, Sibley, David R., Mahler, Stephen V., Nabavi, Sadegh, Pomper, Martin G., Bonci, Antonello, Horti, Andrew G., Richmond, Barry J., Michaelides, Michael
Published in Nature communications (11.10.2019)
Published in Nature communications (11.10.2019)
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The SUV4-20 inhibitor A-196 verifies a role for epigenetics in genomic integrity
Bromberg, Kenneth D, Mitchell, Taylor R H, Upadhyay, Anup K, Jakob, Clarissa G, Jhala, Manisha A, Comess, Kenneth M, Lasko, Loren M, Li, Conglei, Tuzon, Creighton T, Dai, Yujia, Li, Fengling, Eram, Mohammad S, Nuber, Alexander, Soni, Niru B, Manaves, Vlasios, Algire, Mikkel A, Sweis, Ramzi F, Torrent, Maricel, Schotta, Gunnar, Sun, Chaohong, Michaelides, Michael R, Shoemaker, Alex R, Arrowsmith, Cheryl H, Brown, Peter J, Santhakumar, Vijayaratnam, Martin, Alberto, Rice, Judd C, Chiang, Gary G, Vedadi, Masoud, Barsyte-Lovejoy, Dalia, Pappano, William N
Published in Nature chemical biology (01.03.2017)
Published in Nature chemical biology (01.03.2017)
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Progress towards a public chemogenomic set for protein kinases and a call for contributions
Drewry, David H, Wells, Carrow I, Andrews, David M, Angell, Richard, Al-Ali, Hassan, Axtman, Alison D, Capuzzi, Stephen J, Elkins, Jonathan M, Ettmayer, Peter, Frederiksen, Mathias, Gileadi, Opher, Gray, Nathanael, Hooper, Alice, Knapp, Stefan, Laufer, Stefan, Luecking, Ulrich, Michaelides, Michael, Müller, Susanne, Muratov, Eugene, Denny, R Aldrin, Saikatendu, Kumar S, Treiber, Daniel K, Zuercher, William J, Willson, Timothy M
Published in PloS one (02.08.2017)
Published in PloS one (02.08.2017)
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Elucidation of The Behavioral Program and Neuronal Network Encoded by Dorsal Raphe Serotonergic Neurons
Urban, Daniel J, Zhu, Hu, Marcinkiewcz, Catherine A, Michaelides, Michael, Oshibuchi, Hidehiro, Rhea, Darren, Aryal, Dipendra K, Farrell, Martilias S, Lowery-Gionta, Emily, Olsen, Reid H J, Wetsel, William C, Kash, Thomas L, Hurd, Yasmin L, Tecott, Laurence H, Roth, Bryan L
Published in Neuropsychopharmacology (New York, N.Y.) (01.04.2016)
Published in Neuropsychopharmacology (New York, N.Y.) (01.04.2016)
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Target deconvolution studies of (2R,6R)-hydroxynorketamine: an elusive search
Bonaventura, Jordi, Gomez, Juan L., Carlton, Meghan L., Lam, Sherry, Sanchez-Soto, Marta, Morris, Patrick J., Moaddel, Ruin, Kang, Hye Jin, Zanos, Panos, Gould, Todd D., Thomas, Craig J., Sibley, David R., Zarate, Carlos A., Michaelides, Michael
Published in Molecular psychiatry (01.10.2022)
Published in Molecular psychiatry (01.10.2022)
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The Kinase Chemogenomic Set (KCGS): An Open Science Resource for Kinase Vulnerability Identification
Wells, Carrow I, Al-Ali, Hassan, Andrews, David M, Asquith, Christopher R M, Axtman, Alison D, Dikic, Ivan, Ebner, Daniel, Ettmayer, Peter, Fischer, Christian, Frederiksen, Mathias, Futrell, Robert E, Gray, Nathanael S, Hatch, Stephanie B, Knapp, Stefan, Lücking, Ulrich, Michaelides, Michael, Mills, Caitlin E, Müller, Susanne, Owen, Dafydd, Picado, Alfredo, Saikatendu, Kumar S, Schröder, Martin, Stolz, Alexandra, Tellechea, Mariana, Turunen, Brandon J, Vilar, Santiago, Wang, Jinhua, Zuercher, William J, Willson, Timothy M, Drewry, David H
Published in International journal of molecular sciences (08.01.2021)
Published in International journal of molecular sciences (08.01.2021)
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Discovery and Development of Potent and Selective Inhibitors of Histone Methyltransferase G9a
Sweis, Ramzi F, Pliushchev, Marina, Brown, Peter J, Guo, Jun, Li, Fengling, Maag, David, Petros, Andrew M, Soni, Nirupama B, Tse, Chris, Vedadi, Masoud, Michaelides, Michael R, Chiang, Gary G, Pappano, William N
Published in ACS medicinal chemistry letters (13.02.2014)
Published in ACS medicinal chemistry letters (13.02.2014)
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Discovery of Potent Azetidine-Benzoxazole MerTK Inhibitors with In Vivo Target Engagement
Frey, Robin R., Jana, Navendu, Gorman, Jacob V., Wang, Jin, Smith, Heath A., Bromberg, Kenneth D., Thakur, Ashish, Doktor, Stella Z., Indulkar, Anura S., Jakob, Clarissa G., Upadhyay, Anup K., Qiu, Wei, Manaves, Vlasios, Gambino, Frank, Valentino, Stephen A., Montgomery, Debra, Zhou, Yebin, Li, Tao, Buchanan, Fritz G., Ferguson, Debra C., Kurnick, Matthew D., Kapecki, Nicolas, Lai, Albert, Michaelides, Michael R., Penning, Thomas D.
Published in Journal of medicinal chemistry (10.10.2024)
Published in Journal of medicinal chemistry (10.10.2024)
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A non-canonical striatopallidal Go pathway that supports motor control
Labouesse, Marie A., Torres-Herraez, Arturo, Chohan, Muhammad O., Villarin, Joseph M., Greenwald, Julia, Sun, Xiaoxiao, Zahran, Mysarah, Tang, Alice, Lam, Sherry, Veenstra-VanderWeele, Jeremy, Lacefield, Clay O., Bonaventura, Jordi, Michaelides, Michael, Chan, C. Savio, Yizhar, Ofer, Kellendonk, Christoph
Published in Nature communications (23.10.2023)
Published in Nature communications (23.10.2023)
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Motivational valence is determined by striatal melanocortin 4 receptors
Klawonn, Anna Mathia, Fritz, Michael, Nilsson, Anna, Bonaventura, Jordi, Shionoya, Kiseko, Mirrasekhian, Elahe, Karlsson, Urban, Jaarola, Maarit, Granseth, Björn, Blomqvist, Anders, Michaelides, Michael, Engblom, David
Published in The Journal of clinical investigation (01.07.2018)
Published in The Journal of clinical investigation (01.07.2018)
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Discovery of A‑910, a Highly Potent and Orally Bioavailable Dual MerTK/Axl-Selective Tyrosine Kinase Inhibitor
Yu, Yiyun, Jang, Miyeon, Miyashiro, Julie, Clark, Richard F., Zhu, Gui-Dong, Gong, Jane, Dai, Yujia, Frey, Robin R., Penning, Thomas D., Kim, Hadong, Lee, Hyung Ki, Kim, Jin Kwan, Ryu, Ki Moon, Park, Seong Jin, Yoon, Taeyoung, Li, Tao, Kurnick, Matthew D., Kapecki, Nicolas J., Li, Leiming, Gorman, Jacob V., Montgomery, Debra A., Manaves, Vlasios, Bromberg, Kenneth D., Doktor, Stella Z., Thakur, Ashish, Wang, Jin, Smith, Heath A., Buchanan, Fritz G., Ferguson, Debra C., Torrent, Maricel, Jakob, Clarissa G., Qiu, Wei, Upadhyay, Anup K., Martin, Ruth L., Lai, Albert, Michaelides, Michael R.
Published in Journal of medicinal chemistry (10.10.2024)
Published in Journal of medicinal chemistry (10.10.2024)
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Enabling, Decagram-Scale Synthesis of Macrocyclic MCL‑1 Inhibitor ABBV-467
Brady, Patrick B., Sorensen, Bryan K., Risi, Roberto M., Curtin, Michael L., Mantei, Robert A., Florjancic, Alan S., Mastracchio, Anthony, Ji, Cheng, Kunzer, Aaron R., Lai, Chunqiu, Storer, Gregory E., Chan, Vincent S., Henry, Rodger F., Souers, Andrew J., Michaelides, Michael R., Judd, Andrew S., Hansen, T. Matthew
Published in Journal of organic chemistry (17.11.2023)
Published in Journal of organic chemistry (17.11.2023)
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