Selective mono- and polymethylene homologations of copper reagents using (iodomethyl)zinc iodide
Sidduri, AchyuthaRao, Rozema, Michael J, Knochel, Paul
Published in Journal of organic chemistry (01.05.1993)
Published in Journal of organic chemistry (01.05.1993)
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Safe Scale-Up of a Hydrazine Condensation by the Addition of a Base
Wang, Zhe, Richter, Steven M, Gandarilla, Jorge, Kruger, Albert W, Rozema, Michael J
Published in Organic process research & development (20.12.2013)
Published in Organic process research & development (20.12.2013)
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The Discovery and Development of a Safe, Practical Synthesis of ABT-869
Kruger, Albert W, Rozema, Michael J, Chu-Kung, Alexander, Gandarilla, Jorge, Haight, Anthony R, Kotecki, Brian J, Richter, Steven M, Schwartz, Albert M, Wang, Zhe
Published in Organic process research & development (20.11.2009)
Published in Organic process research & development (20.11.2009)
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Journal Article
Preparation and reactions of zinc and copper organometallics bearing acidic hydrogens
Knoess, H. Peter, Furlong, Michael T, Rozema, Michael J, Knochel, Paul
Published in Journal of organic chemistry (01.10.1991)
Published in Journal of organic chemistry (01.10.1991)
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Development of a Scalable Synthesis of Dipeptidyl Peptidase-4 Inhibitor ABT-279
McDermott, Todd S, Bhagavatula, Lakshmi, Borchardt, Thomas B, Engstrom, Kenneth M, Gandarilla, Jorge, Kotecki, Brian J, Kruger, Albert W, Rozema, Michael J, Sheikh, Ahmad Y, Wagaw, Seble H, Wittenberger, Steven J
Published in Organic process research & development (20.11.2009)
Published in Organic process research & development (20.11.2009)
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PROCESSES FOR PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-a]PYRROLO[2,3-e]-PYRAZIN-8-YL)-N-(2,2,2-TRIFLUOROETHYL)PYRROLIDINE-1-CARBOXAMIDE AND SOLID STATE FORMS THEREOF
AHMAD Y SHEIKH, MICHAEL J ROZEMA, THOMAS B BORCHARDT, PETER T MAYER, BEN KLUENDER, MATHEW M MULHERN, AYMAN ALLIAN, MOHAMED-ESLAM F MOHAMED, LAKSHMI BHAGAVATULA, JAYANTHY JAYANTH, AHMED A OTHMAN, PATRICK J MARROUM, FREDRIK LARS NORDSTROM
Year of Publication 29.05.2024
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Year of Publication 29.05.2024
Patent
Zinc and copper carbenoids as efficient and selective a1/d1 multicoupling reagents. 1
Knochel, Paul, Jeong, Nakcheol, Rozema, Michael J, Yeh, Ming Chang P
Published in Journal of the American Chemical Society (01.08.1989)
Published in Journal of the American Chemical Society (01.08.1989)
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METHODS FOR PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-a]PYRROLO[2,3-e]-PYRAZIN-8-YL)-N-(2,2,2-TRIFLUOROETHYL)PYRROLIDINE-1-CARBOXAMIDE AND SOLID STATE FORMS THEREOF
AHMAD Y SHEIKH, MICHAEL J ROZEMA, THOMAS B BORCHARDT, PETER T MAYER, BEN KLUENDER, MATHEW M MULHERN, AYMAN ALLIAN, MOHAMED-ESLAM F MOHAMED, LAKSHMI BHAGAVATULA, JAYANTHY JAYANTH, AHMED A OTHMAN, PATRICK J MARROUM, FREDRIK LARS NORDSTROM
Year of Publication 16.08.2023
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Year of Publication 16.08.2023
Patent
PROCESSES FOR PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-a]PYRROLO[2,3-e]-PYRAZIN-8-YL)-N-(2,2,2-TRIFLUOROETHYL)PYRROLIDINE-1-CARBOXAMIDE AND SOLID STATE FORMS THEREOF
AHMAD Y SHEIKH, MICHAEL J ROZEMA, THOMAS B BORCHARDT, PETER T MAYER, BEN KLUENDER, MATHEW M MULHERN, AYMAN ALLIAN, MOHAMED-ESLAM F MOHAMED, LAKSHMI BHAGAVATULA, JAYANTHY JAYANTH, AHMED A OTHMAN, PATRICK J MARROUM, FREDRIK LARS NORDSTROM
Year of Publication 18.02.2021
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Year of Publication 18.02.2021
Patent
Enantioselective preparation of polyfunctional secondary allylic alcohols using functionalized dialkylzincs prepared by a copper(I) catalyzed iodine-zinc exchange reaction
Rozema, Michael J., Eisenberg, Christina, Lütjens, Henning, Ostwald, Roswitha, Belyk, Kevin, Knochell, Paul
Published in Tetrahedron letters (07.05.1993)
Published in Tetrahedron letters (07.05.1993)
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Development of a Scalable Enantioselective Synthesis of JAK Inhibitor Upadacitinib
Rozema, Michael J., Bhagavatula, Lakshmi, Christesen, Alan, Dunn, Travis B., Ickes, Andrew, Kotecki, Brian J., Marek, James C., Moschetta, Eric, Morrill, Westin H., Mulhern, Mathew, Rasmussen, Michael, Reynolds, Troy, Yu, Su
Published in Organic process research & development (18.03.2022)
Published in Organic process research & development (18.03.2022)
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Journal Article
Nucleophilic reactivity of zinc and copper carbenoids. Part II
Knochel, Paul, Chou, Tso Sheng, Chen, Huai Gu, Yeh, Ming Chang P, Rozema, Michael J
Published in Journal of organic chemistry (01.10.1989)
Published in Journal of organic chemistry (01.10.1989)
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Identification and Preliminary Characterization of a Potent, Safe, and Orally Efficacious Inhibitor of Acyl-CoA:Diacylglycerol Acyltransferase 1
Yeh, Vince S. C, Beno, David W. A, Brodjian, Sevan, Brune, Michael E, Cullen, Steven C, Dayton, Brian D, Dhaon, Madhup K, Falls, Hugh D, Gao, Ju, Grihalde, Nelson, Hajduk, Philip, Hansen, T. Matthew, Judd, Andrew S, King, Andrew J, Klix, Russel C, Larson, Kelly J, Lau, Yau Y, Marsh, Kennan C, Mittelstadt, Scott W, Plata, Dan, Rozema, Michael J, Segreti, Jason A, Stoner, Eric J, Voorbach, Martin J, Wang, Xiaojun, Xin, Xili, Zhao, Gang, Collins, Christine A, Cox, Bryan F, Reilly, Regina M, Kym, Philip R, Souers, Andrew J
Published in Journal of medicinal chemistry (23.02.2012)
Published in Journal of medicinal chemistry (23.02.2012)
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Enantioselective synthesis of the farnesyltransferase inhibitor, A-345665.0
Rozema, Michael J., Fickes, Michael, McLaughlin, Maureen, Rohde, Bridget, McDermott, Todd
Published in Tetrahedron letters (04.12.2006)
Published in Tetrahedron letters (04.12.2006)
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Synthesis of a novel farnesyl transferase inhibitor, ABT-100; selective preparation of a stereogenic tertiary carbinol
Rozema, Michael J., Kruger, Albert W., Rohde, Bridget D., Shelat, Bhadra, Bhagavatula, Lakshmi, Tien, James J., Zhang, Weijiang, Henry, Rodger F.
Published in Tetrahedron (02.05.2005)
Published in Tetrahedron (02.05.2005)
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