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Nayagam, Vasantha M, Wang, Xukun, Tan, Yong Cheng, Poulsen, Anders, Goh, Kee Chuan, Ng, Tony, Wang, Haishan, Song, Hong Yan, Ni, Binhui, Entzeroth, Michael, Stünkel, Walter
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Differential scanning fluorimetry as secondary screening platform for small molecule inhibitors of Bcl-XL
Wan, Kah Fei, Wang, Sifang, Brown, Christopher J., Yu, Victor C., Entzeroth, Michael, Lane, David P., Lee, May Ann
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Published in Cell cycle (Georgetown, Tex.) (01.12.2009)
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Entzeroth, Michael, Flotow, Horst, Condron, Peter
Published in Current protocols in pharmacology (01.03.2009)
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The first highly potent and selective non-peptide neuropeptide Y Y1 receptor antagonist : BIBP3226
RUDOLF, K, EBERLEIN, W, ENGEL, W, WIELAND, H. A, WILLIM, K. D, ENTZEROTH, M, WIENEN, W, BECK-SICKINGER, A. G, DOODS, H. N
Published in European journal of pharmacology (27.12.1994)
Published in European journal of pharmacology (27.12.1994)
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BIBP 3226, the first selective neuropeptide Y1 receptor antagonist: A review of its pharmacological properties
Doods, Henri N., Wieland, Heike A., Engel, Wolfhard, Eberlein, Wolfgang, Willim, Klaus-Dieter, Entzeroth, Michael, Wienen, Wolfgang, Rudolf, Klaus
Published in Regulatory peptides (27.08.1996)
Published in Regulatory peptides (27.08.1996)
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Function of the SIRT1 protein deacetylase in cancer
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Published in Biotechnology journal (01.11.2007)
Published in Biotechnology journal (01.11.2007)
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Characterization of muscarinic receptors in guinea-pig uterus
Doods, Henri N., Willim, Klaus D., Boddeke, Hendrikus W.G.M., Entzeroth, Michael
Published in European journal of pharmacology (07.12.1993)
Published in European journal of pharmacology (07.12.1993)
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Differential scanning fluorimetry as secondary screening platform for small molecule inhibitors of Bcl-X L
Wan, Kah Fei, Wang, Sifang, Brown, Christopher J., Yu, Victor C., Entzeroth, Michael, Lane, David P., Lee, May Ann
Published in Cell cycle (Georgetown, Tex.) (01.12.2009)
Published in Cell cycle (Georgetown, Tex.) (01.12.2009)
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Development of Human Calcitonin Gene-Related Peptide (CGRP) Receptor Antagonists. 1. Potent and Selective Small Molecule CGRP Antagonists. 1-[N 2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1- piperidinyl]carbonyl]-d-tyrosyl]-l-lysyl]-4-(4-pyridinyl)piperazine: The First CGRP Antagonist for Clinical Trials in Acute Migraine
Rudolf, Klaus, Eberlein, Wolfgang, Engel, Wolfhard, Pieper, Helmut, Entzeroth, Michael, Hallermayer, Gerhard, Doods, Henri
Published in Journal of medicinal chemistry (22.09.2005)
Published in Journal of medicinal chemistry (22.09.2005)
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A Review on Telmisartan: A Novel, Long‐Acting Angiotensin II‐Receptor Antagonist
Wienen, Wolfgang, Entzeroth, Michael, Meel, Jacobus C. A., Stangier, Joachim, Busch, Ulrich, Ebner, Thomas, Schmid, Jochen, Lehmann, Horst, Matzek, Kandace, Kempthorne‐Rawson, Joan, Gladigau, Volker, Hauel, Norbert H.
Published in Cardiovascular drug reviews (01.06.2000)
Published in Cardiovascular drug reviews (01.06.2000)
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N-Hydroxy-1,2-disubstituted-1H-benzimidazol-5-yl acrylamides as novel histone deacetylase inhibitors: design, synthesis, SAR studies, and in vivo antitumor activity
Wang, Haishan, Yu, Niefang, Song, Hongyan, Chen, Dizhong, Zou, Yong, Deng, Weiping, Lye, Pek Ling, Chang, Joyce, Ng, Melvin, Sun, Eric T, Sangthongpitag, Kanda, Wang, Xukun, Wu, Xiaofeng, Khng, Hwee Hoon, Fang, Lijuan, Goh, Siok Kun, Ong, Wai Chung, Bonday, Zahid, Stünkel, Walter, Poulsen, Anders, Entzeroth, Michael
Published in Bioorganic & medicinal chemistry letters (01.03.2009)
Published in Bioorganic & medicinal chemistry letters (01.03.2009)
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