Design and Synthesis of Novel α1 a Adrenoceptor-Selective Antagonists. 3. Approaches To Eliminate Opioid Agonist Metabolites by Using Substituted Phenylpiperazine Side Chains
Lagu, Bharat, Tian, Dake, Nagarathnam, Dhanapalan, Marzabadi, Mohammad R, Wong, Wai C, Miao, Shou W, Zhang, Fengqi, Sun, Wanying, Chiu, George, Fang, James, Forray, Carlos, Chang, Raymond S. L, Ransom, Richard W, Chen, Tsing B, O'Malley, Stacey, Zhang, Kanyin, Vyas, Kamlesh P, Gluchowski, Charles
Published in Journal of medicinal chemistry (18.11.1999)
Published in Journal of medicinal chemistry (18.11.1999)
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Design and Synthesis of Novel α1 a Adrenoceptor-Selective Antagonists. 4. Structure−Activity Relationship in the Dihydropyrimidine Series
Wong, Wai C, Sun, Wanying, Lagu, Bharat, Tian, Dake, Marzabadi, Mohammad R, Zhang, Fengqi, Nagarathnam, Dhanapalan, Miao, Shou W, Wetzel, John M, Peng, Jian, Forray, Carlos, Chang, Raymond S. L, Chen, Tsing B, Ransom, Richard, O'Malley, Stacey, Broten, Theodore P, Kling, Paul, Vyas, Kamlesh P, Zhang, Kanyin, Gluchowski, Charles
Published in Journal of medicinal chemistry (18.11.1999)
Published in Journal of medicinal chemistry (18.11.1999)
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Journal Article
Design and synthesis of novel alpha(1a) adrenoceptor-selective antagonists. 3. Approaches to eliminate opioid agonist metabolites by using substituted phenylpiperazine side chains
Lagu, B, Tian, D, Nagarathnam, D, Marzabadi, MR, Wong, WC, Miao, SW, Zhang, FQ, Sun, WY, Chiu, G, Fang, J, Forray, C, Chang, RSL, Ransom, RW, Chen, TB, O'Malley, S, Zhang, KY, Vyas, KP, Gluchowski, C
Published in Journal of medicinal chemistry (18.11.1999)
Published in Journal of medicinal chemistry (18.11.1999)
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Journal Article
Design and synthesis of novel alpha(1a) adrenoceptor-selective antagonists. 4. Structure-activity relationship in the dihydropyrimidine series
Wong, WC, Sun, WY, Lagu, B, Tian, D, Marzabadi, MR, Zhang, FQ, Nagarathnam, D, Miao, SW, Wetzel, JM, Peng, J, Forray, C, Chang, RSL, Chen, TB, Ransom, R, O'Malley, S, Broten, TP, Kling, P, Vyas, KP, Zhang, KY, Gluchowski, C
Published in Journal of medicinal chemistry (18.11.1999)
Published in Journal of medicinal chemistry (18.11.1999)
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In vitro studies on L-771,688 (SNAP 6383), a new potent and selective α1A-adrenoceptor antagonist
CHANG, Raymond S. L, CHEN, Tsing-Bau, QUANRONG SHEN, LAGU, Bharat, MURALI DHAR, T. G, TYAGARAJAN, Sriram, MARZABADI, Mohammad R, WONG, Wai C, GLUCHOWSKI, Charles, FORRAY, Carlos, O'MALLEY, Stacey S, PETTIBONE, Douglas J, DISALVO, Jerry, FRANCIS, Barbara, BOCK, Mark G, FREIDINGER, Roger, NAGARATHNAM, Dhanapalan, MIAO, Shou W
Published in European journal of pharmacology (01.12.2000)
Published in European journal of pharmacology (01.12.2000)
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Journal Article
Design and Synthesis of Novel α 1 a Adrenoceptor-Selective Antagonists. 4. Structure−Activity Relationship in the Dihydropyrimidine Series
Wong, Wai C., Sun, Wanying, Lagu, Bharat, Tian, Dake, Marzabadi, Mohammad R., Zhang, Fengqi, Nagarathnam, Dhanapalan, Miao, Shou W., Wetzel, John M., Peng, Jian, Forray, Carlos, Chang, Raymond S. L., Chen, Tsing B., Ransom, Richard, O'Malley, Stacey, Broten, Theodore P., Kling, Paul, Vyas, Kamlesh P., Zhang, Kanyin, Gluchowski, Charles
Published in Journal of medicinal chemistry (01.11.1999)
Published in Journal of medicinal chemistry (01.11.1999)
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Journal Article
Design and Synthesis of Novel α 1 a Adrenoceptor-Selective Antagonists. 3. Approaches To Eliminate Opioid Agonist Metabolites by Using Substituted Phenylpiperazine Side Chains
Lagu, Bharat, Tian, Dake, Nagarathnam, Dhanapalan, Marzabadi, Mohammad R., Wong, Wai C., Miao, Shou W., Zhang, Fengqi, Sun, Wanying, Chiu, George, Fang, James, Forray, Carlos, Chang, Raymond S. L., Ransom, Richard W., Chen, Tsing B., O'Malley, Stacey, Zhang, Kanyin, Vyas, Kamlesh P., Gluchowski, Charles
Published in Journal of medicinal chemistry (01.11.1999)
Published in Journal of medicinal chemistry (01.11.1999)
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Journal Article
In vitro studies on L-771,688 (SNAP 6383), a new potent and selective α 1A-adrenoceptor antagonist
Chang, Raymond S.L, Chen, Tsing-Bau, O'Malley, Stacey S, Pettibone, Douglas J, DiSalvo, Jerry, Francis, Barbara, Bock, Mark G, Freidinger, Roger, Nagarathnam, Dhanapalan, Miao, Shou W, Shen, Quanrong, Lagu, Bharat, Murali Dhar, T.G, Tyagarajan, Sriram, Marzabadi, Mohammad R, Wong, Wai C, Gluchowski, Charles, Forray, Carlos
Published in European journal of pharmacology (2000)
Published in European journal of pharmacology (2000)
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Soluble guanylate cyclase stimulators
SMITH, CAMERON J, FU, JIANMIN, CHEN, YI-HENG, LI, HONG, WHITEHEAD, ALAN, STELMACH, JOHN, JIANG, FA-LONG, ZHANG, YONG, MIAO, SHOU-WU, LI, GUO-QING, BERGER, RAPHAELLE, GARFUNKLE, JOIE, JI, GANG, ZHANG, RUI, RAGHAVAN, SUBHAREKHA
Year of Publication 01.10.2017
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Year of Publication 01.10.2017
Patent
Design and Synthesis of Novel α1 a Adrenoceptor-Selective Antagonists. 2. Approaches To Eliminate Opioid Agonist Metabolites via Modification of Linker and 4-Methoxycarbonyl-4-phenylpiperidine Moiety
Murali Dhar, T. G, Nagarathnam, Dhanapalan, Marzabadi, Mohammad R, Lagu, Bharat, Wong, Wai C, Chiu, George, Tyagarajan, Sriram, Miao, Shou Wu, Zhang, Fengqi, Sun, Wanying, Tian, Dake, Shen, Quanrong, Zhang, Jack, Wetzel, John M, Forray, Carlos, Chang, Raymond S. L, Broten, Theodore P, Schorn, Terry W, Chen, Tsing Bao, O'Malley, Stacy, Ransom, Richard, Schneck, Kathryn, Bendesky, Robert, Harrell, Charles M, Vyas, Kamlesh P, Zhang, Kanyin, Gilbert, John, Pettibone, Douglas J, Patane, Michael A, Bock, Mark G, Freidinger, Roger M, Gluchowski, Charles
Published in Journal of medicinal chemistry (18.11.1999)
Published in Journal of medicinal chemistry (18.11.1999)
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Journal Article
Design and Synthesis of Novel α1 a Adrenoceptor-Selective Antagonists. 1. Structure−Activity Relationship in Dihydropyrimidinones
Nagarathnam, Dhanapalan, Miao, Shou Wu, Lagu, Bharat, Chiu, George, Fang, James, Murali Dhar, T. G, Zhang, Jack, Tyagarajan, Sriram, Marzabadi, Mohammad R, Zhang, Fengqi, Wong, Wai C, Sun, Wanying, Tian, Dake, Wetzel, John M, Forray, Carlos, Chang, Raymond S. L, Broten, Theodore P, Ransom, Richard W, Schorn, Terry W, Chen, Tsing B, O'Malley, Stacey, Kling, Paul, Schneck, Kathryn, Bendesky, Robert, Harrell, Charles M, Vyas, Kamlesh P, Gluchowski, Charles
Published in Journal of medicinal chemistry (18.11.1999)
Published in Journal of medicinal chemistry (18.11.1999)
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Journal Article
Identification of a Dihydropyridine as a Potent α1a Adrenoceptor-Selective Antagonist That Inhibits Phenylephrine-Induced Contraction of the Human Prostate
Wong, Wai C, Chiu, George, Wetzel, John M, Marzabadi, Mohammad R, Nagarathnam, Dhanapalan, Wang, Diana, Fang, James, Miao, Shou Wu, Hong, Xingfang, Forray, Carlos, Vaysse, Pierre J.-J, Branchek, Theresa A, Gluchowski, Charles, Tang, Rui, Lepor, Herbert
Published in Journal of medicinal chemistry (02.07.1998)
Published in Journal of medicinal chemistry (02.07.1998)
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DIHYDROPYRIMDINES AND USES THEREOF
CHIU, GEORGE, LADU, BHARAT, NAGARATHNAM, DHANAPALAN, MIAO, SHOU W, DHAR, MURALI T, WONG, WAI C, MARZABADI, MOHAMMAD R, GLUCHOWSKI, CHARLES
Year of Publication 27.02.1998
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Year of Publication 27.02.1998
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Dihydropyrimidines and uses thereof
GLUCHOWSKI CHARLES, PATANE MICHAEL A, MIAO SHOU WU, WONG WAI C, NAGARATHNAM DHANAPALAN
Year of Publication 08.05.2001
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Year of Publication 08.05.2001
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Dihydropyrimidines and uses thereof
GLUCHOWSKI CHARLES, PATANE MICHAEL A, MIAO SHOU WU, WONG WAI C, NAGARATHNAM DHANAPALAN
Year of Publication 09.01.2001
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Year of Publication 09.01.2001
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DIHYDROPYRIMIDINES AND USES THEREOF
DHAR, T.G. MURALI, CHIU, GEORGE, NAGARATHNAM, DHANAPALAN, MIAO, SHOU WU, LAGU, BHARAT, WONG, WAI C, MARZABADI, MOHAMMAD R, GLUCHOWSKI, CHARLES
Year of Publication 29.06.2004
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Year of Publication 29.06.2004
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5-(heterocyclic alkyl)-6-aryl-dihydropyrimidines
CHIU GEORGE, GLUCHOWSKI CHARLES, DHAR T. G. MURALI, MIAO SHOU WU, LAGU BHARAT, WONG WAI C, NAGARATHNAM DHANAPALAN, MARZABADI MOHAMMAD R
Year of Publication 27.04.2004
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Year of Publication 27.04.2004
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DIHYDROPYRIMIDINES AND USES THEREOF
PATANE, MICHAEL, A, NAGARATHNAM, DHANAPALAN, WONG, WAI, C, GLUCHOWSKI, CHARLES, MIAO, SHOU, WU
Year of Publication 06.05.1999
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Year of Publication 06.05.1999
Patent