Characterization of Pharmacologic and Pharmacokinetic Properties of CCX168, a Potent and Selective Orally Administered Complement 5a Receptor Inhibitor, Based on Preclinical Evaluation and Randomized Phase 1 Clinical Study
Bekker, Pirow, Dairaghi, Daniel, Seitz, Lisa, Leleti, Manmohan, Wang, Yu, Ertl, Linda, Baumgart, Trageen, Shugarts, Sarah, Lohr, Lisa, Dang, Ton, Miao, Shichang, Zeng, Yibin, Fan, Pingchen, Zhang, Penglie, Johnson, Daniel, Powers, Jay, Jaen, Juan, Charo, Israel, Schall, Thomas J
Published in PloS one (21.10.2016)
Published in PloS one (21.10.2016)
Get full text
Journal Article
A phase I thorough QT/QTc study evaluating therapeutic and supratherapeutic doses of avacopan in healthy participants
Miao, Shichang, Staehr, Peter, Tai, Ezra, Darpo, Borje, Xue, Hongqi, Armas, Danielle, Webster, Kenneth, Oberoi, Rajneet K.
Published in Clinical and translational science (01.07.2024)
Published in Clinical and translational science (01.07.2024)
Get full text
Journal Article
Transcription Factor KLF7 Promotes Osteoclast Differentiation by Suppressing HO-1
Chen, Changhong, Hu, Fei, Miao, Shichang, Sun, Liping, Jiao, Yajun, Xu, Mingwei, Huang, Xin, Yang, Ying, Zhou, Rongkui
Published in Frontiers in genetics (28.03.2022)
Published in Frontiers in genetics (28.03.2022)
Get full text
Journal Article
CCX559 is a potent, orally-administered small molecule PD-L1 inhibitor that induces anti-tumor immunity
Sullivan, Kathleen M C, Vilalta, Marta, Ertl, Linda S, Wang, Yu, Dunlap, Carolyn, Ebsworth, Karen, Zhao, Bin N, Li, Shijie, Zeng, Yibin, Miao, Zhenhua, Fan, Pingchen, Mali, Venkat, Lange, Christopher, McMurtrie, Darren, Yang, Ju, Lui, Rebecca, Scamp, Ryan, Chhina, Vicky, Kumamoto, Alice, Yau, Simon, Dang, Ton, Easterday, Ashton, Liu, Shirley, Miao, Shichang, Charo, Israel, Schall, Thomas J, Zhang, Penglie
Published in PloS one (07.06.2023)
Published in PloS one (07.06.2023)
Get full text
Journal Article
CCR1 blockade reduces tumor burden and osteolysis in vivo in a mouse model of myeloma bone disease
Dairaghi, Daniel J., Oyajobi, Babatunde O., Gupta, Anjana, McCluskey, Brandon, Miao, Shichang, Powers, Jay P., Seitz, Lisa C., Wang, Yu, Zeng, Yibin, Zhang, Penglie, Schall, Thomas J., Jaen, Juan C.
Published in Blood (16.08.2012)
Published in Blood (16.08.2012)
Get full text
Journal Article
CCR2 antagonism leads to marked reduction in proteinuria and glomerular injury in murine models of focal segmental glomerulosclerosis (FSGS)
Miao, Zhenhua, Ertl, Linda S, Newland, Dale, Zhao, Bin, Wang, Yu, Zang, Xiaoping, Campbell, James J, Liu, Xiaoli, Dang, Ton, Miao, Shichang, Krasinski, Antoni, Punna, Sreenivas, Zeng, Yibin, McMahon, Jeffrey, Zhang, Penglie, Charo, Israel F, Schall, Thomas J, Singh, Rajinder
Published in PloS one (21.03.2018)
Published in PloS one (21.03.2018)
Get full text
Journal Article
Correction: Characterization of Pharmacologic and Pharmacokinetic Properties of CCX168, a Potent and Selective Orally Administered Complement 5a Receptor Inhibitor, Based on Preclinical Evaluation and Randomized Phase 1 Clinical Study
Bekker, Pirow, Dairaghi, Daniel, Seitz, Lisa, Leleti, Manmohan, Wang, Yu, Ertl, Linda, Baumgart, Trageen, Shugarts, Sarah, Lohr, Lisa, Dang, Ton, Miao, Shichang, Zeng, Yibin, Fan, Pingchen, Zhang, Penglie, Johnson, Daniel, Powers, Jay, Jaen, Juan, Charo, Israel, Schall, Thomas J
Published in PloS one (04.01.2019)
Published in PloS one (04.01.2019)
Get full text
Journal Article
A fully automated plasma protein precipitation sample preparation method for LC–MS/MS bioanalysis
Ma, Ji, Shi, Jianxia, Le, Hoa, Cho, Robert, Huang, Judy Chi-jou, Miao, Shichang, Wong, Bradley K.
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.02.2008)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.02.2008)
Get full text
Journal Article
Tetrahydroquinoline derivatives as CRTH2 antagonists
Liu, Jiwen, Wang, Yingcai, Sun, Ying, Marshall, Derek, Miao, Shichang, Tonn, George, Anders, Penny, Tocker, Joel, Tang, H. Lucy, Medina, Julio
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
Get full text
Journal Article
Orally administered CCR2 selective inhibitor CCX872-b clinical trial in pancreatic cancer
Noel, Marcus Smith, Hezel, Aram F., Linehan, David, Wang-Gillam, Andrea, Eskens, Ferry, Sleijfer, Stefan, Desar, Ingrid, Erdkamp, Frans, Wilmink, Johanna, Diehl, Janet, Potarca, Antonia, Zhao, Niky, Deng, Jun, Lohr, Lisa, Miao, Shichang, Charo, Israel, Singh, Rajinder, Schall, Thomas J., Bekker, Pirow
Published in Journal of clinical oncology (01.02.2017)
Published in Journal of clinical oncology (01.02.2017)
Get full text
Journal Article
Discovery and optimization of a series of quinazolinone-derived antagonists of CXCR3
Johnson, Michael, Li, An-Rong, Liu, Jiwen, Fu, Zice, Zhu, Liusheng, Miao, Shichang, Wang, Xuemei, Xu, Qingge, Huang, Alan, Marcus, Andrew, Xu, Feng, Ebsworth, Karen, Sablan, Emmanuel, Danao, Jay, Kumer, Jeff, Dairaghi, Dan, Lawrence, Chris, Sullivan, Tim, Tonn, George, Schall, Thomas, Collins, Tassie, Medina, Julio
Published in Bioorganic & medicinal chemistry letters (15.06.2007)
Published in Bioorganic & medicinal chemistry letters (15.06.2007)
Get full text
Journal Article
Discovery of potent and specific CXCR3 antagonists
Chen, Xiaoqi, Mihalic, Jeff, Deignan, Jeff, Gustin, Darin J., Duquette, Jason, Du, Xiaohui, Chan, Johann, Fu, Zice, Johnson, Michael, Li, An-Rong, Henne, Kirk, Sullivan, Tim, Lemon, Bryan, Ma, Ji, Miao, Shichang, Tonn, George, Collins, Tassie, Medina, Julio C.
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
Get full text
Journal Article
Imidazo-pyrazine derivatives as potent CXCR3 antagonists
Du, Xiaohui, Gustin, Darin J., Chen, Xiaoqi, Duquette, Jason, McGee, Lawrence R., Wang, Zhulun, Ebsworth, Karen, Henne, Kirk, Lemon, Bryan, Ma, Ji, Miao, Shichang, Sabalan, Emmanuel, Sullivan, Timothy J., Tonn, George, Collins, Tassie L., Medina, Julio C.
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
Get full text
Journal Article
Discovery and Initial SAR of Arylsulfonylpiperazine Inhibitors of 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD1)
Sun, Daqing, Wang, Zhulun, Di, Yongmei, Jaen, Juan C., Labelle, Marc, Ma, Ji, Miao, Shichang, Sudom, Athena, Tang, Liang, Tomooka, Craig S., Tu, Hua, Ursu, Stefania, Walker, Nigel, Yan, Xuelei, Ye, Qiuping, Powers, Jay P.
Published in Bioorganic & medicinal chemistry (15.06.2008)
Published in Bioorganic & medicinal chemistry (15.06.2008)
Get full text
Journal Article
The synthesis and SAR of novel diarylsulfone 11β-HSD1 inhibitors
Yan, Xuelei, Wang, Zhulun, Sudom, Athena, Cardozo, Mario, DeGraffenreid, Michael, Di, Yongmei, Fan, Pingchen, He, Xiao, Jaen, Juan C., Labelle, Marc, Liu, Jinsong, Ma, Ji, McMinn, Dustin, Miao, Shichang, Sun, Daqing, Tang, Liang, Tu, Hua, Ursu, Stefania, Walker, Nigel, Ye, Qiuping, Powers, Jay P.
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
Get full text
Journal Article
Design and optimization of imidazole derivatives as potent CXCR3 antagonists
Du, Xiaohui, Chen, Xiaoqi, Mihalic, Jeffrey T., Deignan, Jeffrey, Duquette, Jason, Li, An-Rong, Lemon, Bryan, Ma, Ji, Miao, Shichang, Ebsworth, Karen, Sullivan, Timothy J., Tonn, George, Collins, Tassie L., Medina, Julio C.
Published in Bioorganic & medicinal chemistry (15.01.2008)
Published in Bioorganic & medicinal chemistry (15.01.2008)
Get full text
Journal Article
A novel series of IKKβ inhibitors part I: Initial SAR studies of a HTS hit
Cushing, Timothy D., Baichwal, Vijay, Berry, Karen, Billedeau, Roland, Bordunov, Viola, Broka, Chris, Cardozo, Mario, Cheng, Peng, Clark, David, Dalrymple, Stacie, DeGraffenreid, Michael, Gill, Adrian, Hao, Xiaolin, Hawley, Ronald C., He, Xiao, Jaen, Juan C., Labadie, Sharada S., Labelle, Marc, Lehel, Csaba, Lu, Pu-Ping, McIntosh, Joel, Miao, Shichang, Parast, Camran, Shin, Youngsook, Sjogren, Eric B., Smith, Marie-Louise, Talamas, Francisco X., Tonn, George, Walker, Keith M., Walker, Nigel P.C., Wesche, Holger, Whitehead, Chris, Wright, Matt, Browner, Michelle F.
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Get full text
Journal Article
A novel series of IKKβ inhibitors part II: Description of a potent and pharmacologically active series of analogs
Cushing, Timothy D., Baichwal, Vijay, Berry, Karen, Billedeau, Roland, Bordunov, Viola, Broka, Chris, Browner, Michelle F., Cardozo, Mario, Cheng, Peng, Clark, David, Dalrymple, Stacie, DeGraffenreid, Michael, Gill, Adrian, Hao, Xiaolin, Hawley, Ronald C., He, Xiao, Labadie, Sharada S., Labelle, Marc, Lehel, Csaba, Lu, Pu-Ping, McIntosh, Joel, Miao, Shichang, Parast, Camran, Shin, Youngsook, Sjogren, Eric B., Smith, Marie-Louise, Talamas, Francisco X., Tonn, George, Walker, Keith M., Walker, Nigel P.C., Wesche, Holger, Whitehead, Chris, Wright, Matt, Jaen, Juan C.
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Get full text
Journal Article
Circular RNA circ_0000020 promotes osteogenic differentiation to reduce osteoporosis via sponging microRNA miR-142-5p to up-regulate Bone Morphogenetic Protein BMP2
Zhou, Rongkui, Miao, Shichang, Xu, Jun, Sun, Liping, Chen, Yaofei
Published in Bioengineered (01.01.2021)
Published in Bioengineered (01.01.2021)
Get full text
Journal Article