Design, Synthesis, and Pharmacological Evaluation of Benzimidazolo-thiazoles as Potent CXCR3 Antagonists with Therapeutic Potential in Autoimmune Diseases: Discovery of ACT-672125
Caroff, Eva, Meyer, Emmanuel A., Äänismaa, Päivi, Froidevaux, Sylvie, Keller, Marcel, Piali, Luca
Published in Journal of medicinal chemistry (08.09.2022)
Published in Journal of medicinal chemistry (08.09.2022)
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Journal Article
Discovery and In Vivo Evaluation of ACT-660602: A Potent and Selective Antagonist of the Chemokine Receptor CXCR3 for Autoimmune Diseases
Meyer, Emmanuel A., Äänismaa, Päivi, Froidevaux, Sylvie, Keller, Marcel, Piali, Luca, Caroff, Eva
Published in Journal of medicinal chemistry (08.09.2022)
Published in Journal of medicinal chemistry (08.09.2022)
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Journal Article
Interactions with Aromatic Rings in Chemical and Biological Recognition
Meyer, Emmanuel A., Castellano, Ronald K., Diederich, François
Published in Angewandte Chemie (International ed.) (17.03.2003)
Published in Angewandte Chemie (International ed.) (17.03.2003)
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Journal Article
Discovery of the Clinical Candidate IDOR-1117-2520: A Potent and Selective Antagonist of CCR6 for Autoimmune Diseases
Meyer, Emmanuel A., Croxford, Andrew L., Gnerre, Carmela, Kulig, Paulina, Murphy, Mark J., Jacob, Elise M., Schäfer, Gabriel, Richard-Bildstein, Sylvia, Aissaoui, Hamed, Bouis, Patrick, Ertel, Eric A., de Kanter, Ruben, Keller, Marcel P., Lüthi, Urs, Caroff, Eva
Published in Journal of medicinal chemistry (23.05.2024)
Published in Journal of medicinal chemistry (23.05.2024)
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Journal Article
Discovery of Clinical Candidate ACT-777991, a Potent CXCR3 Antagonist for Antigen-Driven and Inflammatory Pathologies
Meyer, Emmanuel A., Äänismaa, Päivi, Ertel, Eric A., Hühn, Eva, Strasser, Daniel S., Rey, Markus, Murphy, Mark J., Martinic, Marianne M., Pouzol, Laetitia, Froidevaux, Sylvie, Keller, Marcel P., Caroff, Eva
Published in Journal of medicinal chemistry (23.03.2023)
Published in Journal of medicinal chemistry (23.03.2023)
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Journal Article
Real-Life Study of the Benefit of Concomitant Radiotherapy with Cemiplimab in Advanced Cutaneous Squamous Cell Carcinoma (cSCC): A Retrospective Cohort Study
Bailly-Caillé, Barbara, Kottler, Diane, Morello, Rémy, Lecornu, Marie, Kao, William, Meyer, Emmanuel, Dompmartin, Anne, L'Orphelin, Jean-Matthieu
Published in Cancers (13.01.2023)
Published in Cancers (13.01.2023)
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Journal Article
Simultaneous integrated boost on pathologic lymph nodes safely improves clinical outcomes compared to sequential boost in locally advanced cervical cancer: a multicenter retrospective study
Guigo, Marin, Dauda, Mohammed Sali, Lequesne, Justine, Blache, Alice, Pereira, Renata, Le Gall, Ioana, Pernin, Victor Emmanuel, Gaichies, Léopold, Clarisse, Bénédicte, Grellard, Jean-Michel, Joly, Florence, Meyer, Emmanuel, Balosso, Jacques
Published in Frontiers in oncology (03.06.2024)
Published in Frontiers in oncology (03.06.2024)
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Journal Article
Stereotactic body radiotherapy as a viable treatment on extracranial oligometastases in melanoma patients: a retrospective multicentric study
Trentesaux, Victorine, Maiezza, Sophie, Bogart, Emilie, Le Deley, Marie-Cécile, Meyer, Emmanuel, Vanquin, Ludovic, Pasquier, David, Mortier, Laurent, Mirabel, Xavier
Published in Frontiers in oncology (05.03.2024)
Published in Frontiers in oncology (05.03.2024)
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Journal Article
Randomized phase II trial in prostate cancer with hormone-sensitive OligometaSTatic relapse: Combining stereotactic ablative radiotherapy and durvalumab (POSTCARD GETUG P13): Study protocol
Rogé, Maximilien, Pointreau, Yoann, Sargos, Paul, Meyer, Emmanuel, Schick, Ulrike, Hasbini, Ali, Rio, Emmanuel, Bera, Guillaume, Ruffier, Amandine, Quivrin, Magali, Chasseray, Mathieu, Latorzeff, Igor, Martin, Etienne, Guimas, Valentine, Pommier, Pascal, Leroy, Thomas, Ronchin, Philippe, Lepinoy, Alexis, Grand, Audrey, Cartier, Lysian, Didas, Ossama, Denis, Fabrice, Libois, Vincent, Blanc-Lapierre, Audrey, Supiot, Stéphane
Published in Clinical and translational radiation oncology (01.05.2023)
Published in Clinical and translational radiation oncology (01.05.2023)
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Journal Article
Information-Theoretic Feature Selection in Microarray Data Using Variable Complementarity
Meyer, P.E., Schretter, C., Bontempi, G.
Published in IEEE journal of selected topics in signal processing (01.06.2008)
Published in IEEE journal of selected topics in signal processing (01.06.2008)
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Journal Article
Web Resource
Crystal Structures of tRNA-guanine Transglycosylase (TGT) in Complex with Novel and Potent Inhibitors Unravel Pronounced Induced-fit Adaptations and Suggest Dimer Formation Upon Substrate Binding
Stengl, Bernhard, Meyer, Emmanuel A., Heine, Andreas, Brenk, Ruth, Diederich, François, Klebe, Gerhard
Published in Journal of molecular biology (13.07.2007)
Published in Journal of molecular biology (13.07.2007)
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Journal Article
Synthesis, Biological Evaluation, and Crystallographic Studies of Extended Guanine-Based (lin-Benzoguanine) Inhibitors for tRNA-Guanine Transglycosylase (TGT)
Meyer, Emmanuel A., Donati, Nicola, Guillot, Marine, Schweizer, W. Bernd, Diederich, François, Stengl, Bernhard, Brenk, Ruth, Reuter, Klaus, Klebe, Gerhard
Published in Helvetica chimica acta (01.04.2006)
Published in Helvetica chimica acta (01.04.2006)
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Journal Article
Crystallographic Study of Inhibitors of tRNA-guanine Transglycosylase Suggests a New Structure-based Pharmacophore for Virtual Screening
Brenk, Ruth, Meyer, EmmanuelA, Reuter, Klaus, Stubbs, Milton T., Garcia, George A., Diederich, François, Klebe, Gerhard
Published in Journal of molecular biology (16.04.2004)
Published in Journal of molecular biology (16.04.2004)
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Journal Article
De Novo Design, Synthesis, and In Vitro Evaluation of Inhibitors for Prokaryotic tRNA-Guanine Transglycosylase: A Dramatic Sulfur Effect on Binding Affinity
Meyer, Emmanuel A., Brenk, Ruth, Castellano, Ronald K., Furler, Maya, Klebe, Gerhard, Diederich, François
Published in Chembiochem : a European journal of chemical biology (01.03.2002)
Published in Chembiochem : a European journal of chemical biology (01.03.2002)
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Journal Article
Enzymatic reactions in liposomes using the detergent-induced liposome loading method
Oberholzer, Thomas, Meyer, Emmanuel, Amato, Irene, Lustig, Ariel, Monnard, Pierre-Alain
Published in Biochimica et biophysica acta (12.01.1999)
Published in Biochimica et biophysica acta (12.01.1999)
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Journal Article
Salvage Stereotactic Body Radiation Therapy for Local Prostate Cancer Recurrence After Radiation Therapy: A Retrospective Multicenter Study of the GETUG
Pasquier, David, Martinage, Geoffrey, Janoray, Guillaume, Rojas, Damaris Patricia, Zerini, Dario, Goupy, Flora, De Crevoisier, Renaud, Bogart, Emilie, Calais, Gilles, Toledano, Alain, Chauveinc, Laurent, Scher, Nathaniel, Bondiau, Pierre Yves, Hannoun-Levi, Jean Michel, Silva, Marlon, Meyer, Emmanuel, Nickers, Philippe, Lacornerie, Thomas, Jereczek-Fossa, Barbara Alicja, Lartigau, Eric
Published in International journal of radiation oncology, biology, physics (15.11.2019)
Published in International journal of radiation oncology, biology, physics (15.11.2019)
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Journal Article