Discovery of Potent and Selective SH2 Inhibitors of the Tyrosine Kinase ZAP-70
Vu, Chi B, Corpuz, Evelyn G, Merry, Taylor J, Pradeepan, Selvaluxmi G, Bartlett, Catherine, Bohacek, Regine S, Botfield, Martyn C, Eyermann, Charles J, Lynch, Berkley A, MacNeil, Ian A, Ram, Mary K, van Schravendijk, Marie Rose, Violette, Shelia, Sawyer, Tomi K
Published in Journal of medicinal chemistry (07.10.1999)
Published in Journal of medicinal chemistry (07.10.1999)
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Journal Article
Early Point-of-Care Testing at Triage Reduces Care Time in Stable Adult Emergency Department Patients
Singer, Adam J., Taylor, Merry, LeBlanc, Deborah, Meyers, Kristen, Perez, Karol, Thode, Henry C., Pines, Jesse M.
Published in The Journal of emergency medicine (01.08.2018)
Published in The Journal of emergency medicine (01.08.2018)
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Diagnostic Characteristics of a Clinical Screening Tool in Combination With Measuring Bedside Lactate Level in Emergency Department Patients With Suspected Sepsis
Singer, Adam J., Taylor, Merry, Domingo, Anna, Ghazipura, Saad, Khorasonchi, Adam, Thode, Henry C., Shapiro, Nathan I., Jang, Timothy
Published in Academic emergency medicine (01.08.2014)
Published in Academic emergency medicine (01.08.2014)
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Structure-Based Design of an Osteoclast-Selective, Nonpeptide Src Homology 2 Inhibitor with in vivo Antiresorptive Activity
Shakespeare, William, Yang, Michael, Bohacek, Regine, Cerasoli, Franklin, Stebbins, Karin, Sundaramoorthi, Raji, Azimioara, Mihai, Vu, Chi, Pradeepan, Selvi, Metcalf, Chester, Haraldson, Chad, Merry, Taylor, Dalgarno, David, Narula, Surinder, Hatada, Marcos, Lu, Xiaode, van Schravendijk, Marie Rose, Adams, Susan, Violette, Shelia, Smith, Jeremy, Guan, Wei, Bartlett, Catherine, Herson, Jay, Iuliucci, John, Weigele, Manfred, Sawyer, Tomi
Published in Proceedings of the National Academy of Sciences - PNAS (15.08.2000)
Published in Proceedings of the National Academy of Sciences - PNAS (15.08.2000)
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Journal Article
Bone-Targeted Src kinase inhibitors: novel pyrrolo- and pyrazolopyrimidine analogues
Sundaramoorthi, Raji, Shakespeare, William C., Keenan, Terence P., Metcalf, Chester A., Wang, Yihan, Mani, Ukti, Taylor, Merry, Liu, Shuangying, Bohacek, Regine S., Narula, Surinder S., Dalgarno, David C., Van Schravandijk, Marie Rose, Violette, Sheila M., Liou, Shuenn, Adams, Susan, Ram, Mary K., Keats, Jeffrey A., Weigele, Manfred, Sawyer, Tomi K.
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
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Journal Article
X-ray Structure of Citrate Bound to Src SH2 Leads to a High-Affinity, Bone-Targeted Src SH2 Inhibitor
Bohacek, Regine S, Dalgarno, David C, Hatada, Marcos, Jacobsen, Virginia A, Lynch, Berkley A, Macek, Karina J, Merry, Taylor, Metcalf, Chester A, Narula, Surinder S, Sawyer, Tomi K, Shakespeare, William C, Violette, Shelia M, Weigele, Manfred
Published in Journal of medicinal chemistry (01.03.2001)
Published in Journal of medicinal chemistry (01.03.2001)
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Journal Article
Bone-Targeted pyrido[2,3- d]pyrimidin-7-ones: potent inhibitors of Src tyrosine kinase as novel antiresorptive agents
Vu, Chi B., Luke, George P., Kawahata, Noriyuki, Shakespeare, William C., Wang, Yihan, Sundaramoorthi, Raji, Metcalf, Chester A., Keenan, Terence P., Pradeepan, Selvi, Corpuz, Evelyn, Merry, Taylor, Bohacek, Regine S., Dalgarno, David C., Narula, Surinder S., van Schravendijk, Marie Rose, Ram, Mary K., Adams, Susan, Liou, Shuenn, Keats, Jeffrey A., Violette, Shelia M., Guan, Wei, Weigele, Manfred, Sawyer, Tomi K.
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
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Journal Article
Structure-based design of novel nonpeptide inhibitors of the Src SH2 domain: Phosphotyrosine mimetics exploiting multifunctional group replacement chemistry
Sundaramoorthi, Raji, Kawahata, Noriyuki, Yang, Michael G., Shakespeare, William C., Metcalf III, Chester A., Wang, Yihan, Merry, Taylor, Eyermann, Charles J., Bohacek, Regine S., Narula, Surinder, Dalgarno, David C., Sawyer, Tomi K.
Published in Biopolymers (2003)
Published in Biopolymers (2003)
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Journal Article
Structure-activity relationships of a novel class of Src SH2 inhibitors
Buchanan, John L., Vu, Chi B., Merry, Taylor J., Corpuz, Evelyn G., Pradeepan, Selvaluxmi G., Mani, Ukti N., Yang, Michael, Plake, Hilary R., Varkhedkar, Vaibhav M., Lynch, Berkley A., MacNeil, Ian A., Loiacono, Kara A., Tiong, Choi Lai, Holt, Dennis A.
Published in Bioorganic & medicinal chemistry letters (16.08.1999)
Published in Bioorganic & medicinal chemistry letters (16.08.1999)
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Journal Article
A novel phosphotyrosine mimetic 4'-carboxymethyloxy-3'-phosphonophenylalanine (Cpp): exploitation in the design of nonpeptide inhibitors of pp60(Src) SH2 domain
Kawahata, N, Yang, M G, Luke, G P, Shakespeare, W C, Sundaramoorthi, R, Wang, Y, Johnson, D, Merry, T, Violette, S, Guan, W, Bartlett, C, Smith, J, Hatada, M, Lu, X, Dalgarno, D C, Eyermann, C J, Bohacek, R S, Sawyer, T K
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
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Journal Article
Corrigendum to “Bone-Targeted Src Kinase Inhibitors: Novel Pyrrolo- and Pyrazolopyrimidine Analogues”[Bioorg. Med. Chem. Lett. 13 (2003) 3063]
Sundaramoorthi, Raji, Shakespeare, William C, Keenan, Terence P, Metcalf, Chester A, Wang, Yihan, Mani, Ukti, Merry, Taylor, Liu, Shuangying, Bohacek, Regine S, Narula, Surinder S, Dalgarno, David C, Van Schravendijk, Marie Rose, Violette, Shelia M, Liou, Shuenn, Adams, Susan, Ram, Mary K, Keats, Jeffrey A, Weigle, Manfred, Sawyer, Tomi K
Published in Bioorganic & medicinal chemistry letters (01.12.2003)
Published in Bioorganic & medicinal chemistry letters (01.12.2003)
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Journal Article
Bone-targeted Src kinase inhibitors: Novel pyrrolo- and pyrazolopyrimidine analogues: Recent advances in the design of kinase inhibitors as novel therapeutic agents
SUNDARAMOORTHI, Raji, SHAKESPEARE, William C, DALGARNO, David C, VAN SCHRAVANDIJK, Marie Rose, VIOLETTE, Sheila M, LIOU, Shuenn, ADAMS, Susan, RAM, Mary K, KEATS, Jeffrey A, WEIGELE, Manfred, SAWYER, Tomi K, KEENAN, Terence P, METCALF, Chester A, YIHAN WANG, MANI, Ukti, TAYLOR, Merry, SHUANGYING LIU, BOHACEK, Regine S, NARULA, Surinder S
Published in Bioorganic & medicinal chemistry letters (2003)
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Published in Bioorganic & medicinal chemistry letters (2003)
Journal Article
A novel phosphotyrosine mimetic 4'-carboxymethyloxy-3'-phosphonophenylalanine (Cpp) : Exploitation in the design of nonpeptide inhibitors of pp60Src SH2 domain
KAWAHATA, Noriyuki, YANG, Michael G, BARTLETT, Catherine, SMITH, Jeremy, HATADA, Marcos, XIAODE LU, DALGARNO, David C, EYERMANN, Charles J, BOHACEK, Regine S, SAWYER, Tomi K, LUKE, George P, SHAKESPEARE, William C, SUNDARAMOORTHI, Raji, YIHAN WANG, JOHNSON, Daniel, MERRY, Taylor, VIOLETTE, Shelia, WEI GUAN
Published in Bioorganic & medicinal chemistry letters (01.09.2001)
Published in Bioorganic & medicinal chemistry letters (01.09.2001)
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Journal Article
A novel phosphotyrosine mimetic 4′-carboxymethyloxy-3′-phosphonophenylalanine (cpp): exploitation in the design of nonpeptide inhibitors of pp60 Src SH2 domain
Kawahata, Noriyuki, Yang, Michael G., Luke, George P., Shakespeare, William C., Sundaramoorthi, Raji, Wang, Yihan, Johnson, Daniel, Merry, Taylor, Violette, Shelia, Guan, Wei, Bartlett, Catherine, Smith, Jeremy, Hatada, Marcos, Lu, Xiaode, Dalgarno, David C., Eyermann, Charles J., Bohacek, Regine S., Sawyer, Tomi K.
Published in Bioorganic & medicinal chemistry letters (2001)
Published in Bioorganic & medicinal chemistry letters (2001)
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Journal Article
Novel phosphate ester-linked resins: The solid-phase generation of phenyl phosphate-containing compounds for SH2 inhibition
Metcalf, Chester A., Vu, Chi B., Sundaramoorthi, Raji, Jacobsen, Virginia A., Laborde, Edgardo A., Green, Jeremy, Green, Yinka, Macek, Karina J., Merry, Taylor J., Pradeepan, Selvi G., Uesugi, Mayumi, Varkhedkar, Vaibhav M., Holt, Dennis A.
Published in Tetrahedron letters (21.05.1998)
Published in Tetrahedron letters (21.05.1998)
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Journal Article
Bone-targeted pyrido[2,3-d]pyrimidin-7-ones: Potent inhibitors of Src tyrosine kinase as novel antiresorptive agents: Recent advances in the design of kinase inhibitors as novel therapeutic agents
VU, Chi B, LUKE, George P, MERRY, Taylor, BOHACEK, Regine S, DALGARNO, David C, NARULA, Surinder S, VAN SCHRAVENDIJK, Marie Rose, RAM, Mary K, ADAMS, Susan, LIOU, Shuenn, KEATS, Jeffrey A, VIOLETTE, Shelia M, KAWAHATA, Noriyuki, WEI GUAN, WEIGELE, Manfred, SAWYER, Tomi K, SHAKESPEARE, William C, YIHAN WANG, SUNDARAMOORTHI, Raji, METCALF, Chester A, KEENAN, Terence P, PRADEEPAN, Selvi, CORPUZ, Evelyn
Published in Bioorganic & medicinal chemistry letters (2003)
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Published in Bioorganic & medicinal chemistry letters (2003)
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