Small-Molecule Covalent Modification of Conserved Cysteine Leads to Allosteric Inhibition of the TEAD⋅Yap Protein-Protein Interaction
Bum-Erdene, Khuchtumur, Zhou, Donghui, Gonzalez-Gutierrez, Giovanni, Ghozayel, Mona K, Si, Yubing, Xu, David, Shannon, Harlan E, Bailey, Barbara J, Corson, Timothy W, Pollok, Karen E, Wells, Clark D, Meroueh, Samy O
Published in Cell chemical biology (21.03.2019)
Published in Cell chemical biology (21.03.2019)
Get full text
Journal Article
Atractylenolide I enhances responsiveness to immune checkpoint blockade therapy by activating tumor antigen presentation
Xu, Hanchen, Van der Jeught, Kevin, Zhou, Zhuolong, Zhang, Lu, Yu, Tao, Sun, Yifan, Li, Yujing, Wan, Changlin, So, Ka Man, Liu, Degang, Frieden, Michael, Fang, Yuanzhang, Mosley, Amber L, He, Xiaoming, Zhang, Xinna, Sandusky, George E, Liu, Yunlong, Meroueh, Samy O, Zhang, Chi, Wijeratne, Aruna B, Huang, Cheng, Ji, Guang, Lu, Xiongbin
Published in The Journal of clinical investigation (15.05.2021)
Published in The Journal of clinical investigation (15.05.2021)
Get full text
Journal Article
Small-Molecule Cyanamide Pan-TEAD·YAP1 Covalent Antagonists
Bum-Erdene, Khuchtumur, Yeh, I-Ju, Gonzalez-Gutierrez, Giovanni, Ghozayel, Mona K., Pollok, Karen, Meroueh, Samy O.
Published in Journal of medicinal chemistry (12.01.2023)
Published in Journal of medicinal chemistry (12.01.2023)
Get full text
Journal Article
Small-molecule covalent bond formation at tyrosine creates a binding site and inhibits activation of Ral GTPases
Bum-Erdene, Khuchtumur, Liu, Degang, Gonzalez-Gutierrez, Giovanni, Ghozayel, Mona K., Xu, David, Meroueh, Samy O.
Published in Proceedings of the National Academy of Sciences - PNAS (31.03.2020)
Published in Proceedings of the National Academy of Sciences - PNAS (31.03.2020)
Get full text
Journal Article
Crystal Packing Reveals a Potential Autoinhibited KRAS Dimer Interface and a Strategy for Small-Molecule Inhibition of RAS Signaling
Brenner, Robert J, Landgraf, Alexander D, Bum-Erdene, Khuchtumur, Gonzalez-Gutierrez, Giovanni, Meroueh, Samy O
Published in Biochemistry (Easton) (21.11.2023)
Published in Biochemistry (Easton) (21.11.2023)
Get full text
Journal Article
Covalent Fragment Inhibits RhoA Activation by Guanine Exchange Factors
Hussain, Muhammad S., Liu, Degang, Alilain, Warren J., Meroueh, Samy O.
Published in ACS chemical neuroscience (19.07.2023)
Published in ACS chemical neuroscience (19.07.2023)
Get full text
Journal Article
Discovery and characterization of small molecules that target the GTPase Ral
Yan, Chao, Liu, Degang, Li, Liwei, Wempe, Michael F, Guin, Sunny, Khanna, May, Meier, Jeremy, Hoffman, Brenton, Owens, Charles, Wysoczynski, Christina L, Nitz, Matthew D, Knabe, William E, Ahmed, Mansoor, Brautigan, David L, Paschal, Bryce M, Schwartz, Martin A, Jones, David N M, Ross, David, Meroueh, Samy O, Theodorescu, Dan
Published in Nature (London) (20.11.2014)
Published in Nature (London) (20.11.2014)
Get full text
Journal Article
Mimicking Intermolecular Interactions of Tight Protein–Protein Complexes for Small‐Molecule Antagonists
Xu, David, Bum‐Erdene, Khuchtumur, Si, Yubing, Zhou, Donghui, Ghozayel, Mona K., Meroueh, Samy O.
Published in ChemMedChem (08.11.2017)
Published in ChemMedChem (08.11.2017)
Get full text
Journal Article
Three-Dimensional Structure of the Bacterial Cell Wall Peptidoglycan
Meroueh, Samy O., Bencze, Krisztina Z., Hesek, Dusan, Lee, Mijoon, Fisher, Jed F., Stemmler, Timothy L., Mobashery, Shahriar
Published in Proceedings of the National Academy of Sciences - PNAS (21.03.2006)
Published in Proceedings of the National Academy of Sciences - PNAS (21.03.2006)
Get full text
Journal Article
Chemical Proteomics Reveals Soluble Epoxide Hydrolase as a Therapeutic Target for Ocular Neovascularization
Sulaiman, Rania S, Park, Bomina, Sheik Pran Babu, Sardar Pasha, Si, Yubing, Kharwadkar, Rakshin, Mitter, Sayak K, Lee, Bit, Sun, Wei, Qi, Xiaoping, Boulton, Michael E, Meroueh, Samy O, Fei, Xiang, Seo, Seung-Yong, Corson, Timothy W
Published in ACS chemical biology (19.01.2018)
Published in ACS chemical biology (19.01.2018)
Get full text
Journal Article
Suppression of inflammatory and neuropathic pain by uncoupling CRMP-2 from the presynaptic Ca²⁺ channel complex
Brittain, Joel M, Duarte, Djane B, Wilson, Sarah M, Zhu, Weiguo, Ballard, Carrie, Johnson, Philip L, Liu, Naikui, Xiong, Wenhui, Ripsch, Matthew S, Wang, Yuying, Fehrenbacher, Jill C, Fitz, Stephanie D, Khanna, May, Park, Chul-Kyu, Schmutzler, Brian S, Cheon, Bo Myung, Due, Michael R, Brustovetsky, Tatiana, Ashpole, Nicole M, Hudmon, Andy, Meroueh, Samy O, Hingtgen, Cynthia M, Brustovetsky, Nickolay, Ji, Ru-Rong, Hurley, Joyce H, Jin, Xiaoming, Shekhar, Anantha, Xu, Xiao-Ming, Oxford, Gerry S, Vasko, Michael R, White, Fletcher A, Khanna, Rajesh
Published in Nature medicine (05.06.2011)
Published in Nature medicine (05.06.2011)
Get full text
Journal Article
A small molecule Inauhzin inhibits SIRT1 activity and suppresses tumour growth through activation of p53
Zhang, Qi, Zeng, Shelya X., Zhang, Yu, Zhang, Yiwei, Ding, Derong, Ye, Qizhuang, Meroueh, Samy O., Lu, Hua
Published in EMBO molecular medicine (01.04.2012)
Published in EMBO molecular medicine (01.04.2012)
Get full text
Journal Article