Search Results - "MENGE WIRO M.P.B" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Synthesis and use of FSCPX, an irreversible adenosine A1 antagonist, as a 'Receptor knock-down' tool

Synthesis and use of FSCPX, an irreversible adenosine A1 antagonist, as a 'Receptor knock-down' tool

by VAN MUIJLWIJK-KOEZEN, Jacqueline E, TIMMERMAN, Henk, VAN DER SLUIS, Richard P, VAN DE STOLPE, Andrea C, MENGE, Wiro M. P. B, BEUKERS, Margot W, VAN DER GRAAF, Piet H, DE GROOTE, Miriam, IJZERMAN, Adriaan P
Published in Bioorganic & medicinal chemistry letters (26.03.2001)

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New synthetic flavonoids as potent protectors against doxorubicin-induced cardiotoxicity

New synthetic flavonoids as potent protectors against doxorubicin-induced cardiotoxicity

by van Acker, Frédérique A.A, Hulshof, Janneke W, Haenen, Guido R.M.M, Menge, Wiro M.P.B, van der Vijgh, Wim J.F, Bast, Aalt
Published in Free radical biology & medicine (01.07.2001)

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New high affinity H3 receptor agonists without a basic side chain

New high affinity H3 receptor agonists without a basic side chain

by KITBUNNADAJ, Ruengwit, HOFFMANN, Marcel, LEURS, Rob, FRATANTONI, Silvina A, BONGERS, Gerold, BAKKER, Remko A, WIELAND, Kerstin, EL JILALI, Ahmed, DE ESCH, Iwan J. P, MENGE, Wiro M. P. B, TIMMERMAN, Henk
Published in Bioorganic & medicinal chemistry (01.12.2005)

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A role for spinal, but not supraspinal, α2 adrenergic receptors in the actions of improgan, a powerful, non-opioid analgesic

A role for spinal, but not supraspinal, α2 adrenergic receptors in the actions of improgan, a powerful, non-opioid analgesic

by SVOKOS, Konstantina, NALWALK, Julia W, LEURS, Rob, MENGE, Wiro M. P. B, TIMMERMAN, Henk, HOUGH, Lindsay B
Published in Brain research (27.12.2001)

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Synthesis and histamine H3 receptor activity of 4-(n-alkyl)-1H-imidazoles and 4-(ω-phenylalkyl)-1H-imidazoles

Synthesis and histamine H3 receptor activity of 4-(n-alkyl)-1H-imidazoles and 4-(ω-phenylalkyl)-1H-imidazoles

by DE ESCH, I. J. P, GAFFAR, A, MENGE, W. M. P. B, TIMMERMAN, H
Published in Bioorganic & medicinal chemistry (01.12.1999)

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Cytotoxicity of a series of mono- and di-substituted thiourea in freshly isolated rat hepatocytes: a preliminary structure-toxicity relationship study

Cytotoxicity of a series of mono- and di-substituted thiourea in freshly isolated rat hepatocytes: a preliminary structure-toxicity relationship study

by Onderwater, Rob C.A, Commandeur, Jan N.M, Groot, Ed J, Sitters, Astrid, Menge, Wiro M.P.B, Vermeulen, Nico P.E
Published in Toxicology (Amsterdam) (06.02.1998)

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Absence of antinociceptive tolerance to improgan, a cimetidine analog, in rats

Absence of antinociceptive tolerance to improgan, a cimetidine analog, in rats

by Bannoura, Michelle D, Nalwalk, Julia W, Tang, Yuming, Carlile, MaryEllen, Leurs, Rob, Menge, Wiro M.P.B, Timmerman, Henk, Hough, Lindsay B
Published in Brain research (14.12.1998)

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Identification of 4-(1H-Imidazol-4(5)-ylmethyl)pyridine (Immethridine) as a Novel, Potent, and Highly Selective Histamine H3 Receptor Agonist

Identification of 4-(1H-Imidazol-4(5)-ylmethyl)pyridine (Immethridine) as a Novel, Potent, and Highly Selective Histamine H3 Receptor Agonist

by Kitbunnadaj, Ruengwit, Zuiderveld, Obbe P, Christophe, Bernard, Hulscher, Saskia, Menge, Wiro M. P. B, Gelens, Edith, Snip, Erwin, Bakker, Remko A, Celanire, Sylvain, Gillard, Michel, Talaga, Patrice, Timmerman, Henk, Leurs, Rob
Published in Journal of medicinal chemistry (06.05.2004)

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Isoquinoline and Quinazoline Urea Analogues as Antagonists for the Human Adenosine A3 Receptor

Isoquinoline and Quinazoline Urea Analogues as Antagonists for the Human Adenosine A3 Receptor

by van Muijlwijk-Koezen, Jacqueline E, Timmerman, Henk, van der Goot, Henk, Menge, Wiro M. P. B, Frijtag von Drabbe Künzel, Jacobien, de Groote, Miriam, IJzerman, Adriaan P
Published in Journal of medicinal chemistry (01.06.2000)

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N-Substituted Piperidinyl Alkyl Imidazoles: Discovery of Methimepip as a Potent and Selective Histamine H3 Receptor Agonist

N-Substituted Piperidinyl Alkyl Imidazoles: Discovery of Methimepip as a Potent and Selective Histamine H3 Receptor Agonist

by Kitbunnadaj, Ruengwit, Hashimoto, Takeshi, Poli, Enzo, Zuiderveld, Obbe P, Menozzi, Alessandro, Hidaka, Ryoko, de Esch, Iwan J. P, Bakker, Remko A, Menge, Wiro M. P. B, Yamatodani, Atsushi, Coruzzi, Gabriella, Timmerman, Henk, Leurs, Rob
Published in Journal of medicinal chemistry (24.03.2005)

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Synthesis and Structure−Activity Relationships of Conformationally Constrained Histamine H3 Receptor Agonists

Synthesis and Structure−Activity Relationships of Conformationally Constrained Histamine H3 Receptor Agonists

by Kitbunnadaj, Ruengwit, Zuiderveld, Obbe P, De Esch, Iwan J. P, Vollinga, Roeland C, Bakker, Remko, Lutz, Martin, Spek, Anthony L, Cavoy, Emile, Deltent, Marie-France, Menge, Wiro M. P. B, Timmerman, Henk, Leurs, Rob
Published in Journal of medicinal chemistry (04.12.2003)

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Synthesis and Structure−Activity Relationship of the First Nonpeptidergic Inverse Agonists for the Human Cytomegalovirus Encoded Chemokine Receptor US28

Synthesis and Structure−Activity Relationship of the First Nonpeptidergic Inverse Agonists for the Human Cytomegalovirus Encoded Chemokine Receptor US28

by Hulshof, Janneke W, Casarosa, Paola, Menge, Wiro M. P. B, Kuusisto, Leena M. S, van der Goot, Henk, Smit, Martine J, de Esch, Iwan J. P, Leurs, Rob
Published in Journal of medicinal chemistry (06.10.2005)

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A Chemical Switch for the Modulation of the Functional Activity of Higher Homologues of Histamine on the Human Histamine H3 Receptor: Effect of Various Substitutions at the Primary Amino Function

A Chemical Switch for the Modulation of the Functional Activity of Higher Homologues of Histamine on the Human Histamine H3 Receptor: Effect of Various Substitutions at the Primary Amino Function

by Govoni, Marinella, Lim, Herman D., El-Atmioui, Dris, Menge, Wiro M. P. B., Timmerman, Henk, Bakker, Remko A., Leurs, Rob, De Esch, Iwan J. P.
Published in Journal of medicinal chemistry (20.04.2006)

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New high affinity H 3 receptor agonists without a basic side chain

New high affinity H 3 receptor agonists without a basic side chain

by Kitbunnadaj, Ruengwit, Hoffmann, Marcel, Fratantoni, Silvina A., Bongers, Gerold, Bakker, Remko A., Wieland, Kerstin, Jilali, Ahmed el, De Esch, Iwan J.P., Menge, Wiro M.P.B., Timmerman, Henk, Leurs, Rob
Published in Bioorganic & medicinal chemistry (01.12.2005)

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Synthesis of Novel Se-Substituted Selenocysteine Derivatives as Potential Kidney Selective Prodrugs of Biologically Active Selenol Compounds: Evaluation of Kinetics of β-Elimination Reactions in Rat Renal Cytosol

Synthesis of Novel Se-Substituted Selenocysteine Derivatives as Potential Kidney Selective Prodrugs of Biologically Active Selenol Compounds: Evaluation of Kinetics of β-Elimination Reactions in Rat Renal Cytosol

by Andreadou, Ioanna, Menge, Wiro M. P. B, Commandeur, Jan N. M, Worthington, Eduard A, Vermeulen, Nico P. E
Published in Journal of medicinal chemistry (10.05.1996)

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Evaluation of [ 18 F]VUF 5000 as a potential PET ligand for brain imaging of the histamine H 3 receptor

Evaluation of [ 18 F]VUF 5000 as a potential PET ligand for brain imaging of the histamine H 3 receptor

by Windhorst, Albert D., Timmerman, Henk, Klok, Rob P., Menge, Wiro M.P.B., Leurs, Rob, Herscheid, Jacobus D.M.
Published in Bioorganic & medicinal chemistry (01.09.1999)

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A role for spinal, but not supraspinal, α 2 adrenergic receptors in the actions of improgan, a powerful, non-opioid analgesic

A role for spinal, but not supraspinal, α 2 adrenergic receptors in the actions of improgan, a powerful, non-opioid analgesic

by Svokos, Konstantina, Nalwalk, Julia W, Leurs, Rob, Menge, Wiro M.P.B, Timmerman, Henk, Hough, Lindsay B
Published in Brain research (2001)

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Journal Article

A New Potent and Selective Histamine H3 Receptor Agonist, 4-(1H-imidazol-4-ylmethyl)piperidine

A New Potent and Selective Histamine H3 Receptor Agonist, 4-(1H-imidazol-4-ylmethyl)piperidine

by Vollinga, Roeland C, de Koning, Johannes P, Jansen, Frank P, Leurs, Rob, Menge, Wiro M. P. B, Timmerman, Hendrik
Published in Journal of medicinal chemistry (01.02.1994)

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A Third Life for Burimamide: Discovery and Characterization of a Novel Class of Non-Opioid Analgesics Derived from Histamine Antagonists

A Third Life for Burimamide: Discovery and Characterization of a Novel Class of Non-Opioid Analgesics Derived from Histamine Antagonists

by HOUGH, LINDSAY B., NALWALK, JULIA W., BARNES, WILLIAM G., LEURS, ROB, MENGE, WIRO M. P. B., TIMMERMAN, HENK, WENTLAND, MARK
Published in Annals of the New York Academy of Sciences (01.01.2000)

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Evaluation of [18F]VUF 5000 as a potential PET ligand for brain imaging of the histamine H3 receptor

Evaluation of [18F]VUF 5000 as a potential PET ligand for brain imaging of the histamine H3 receptor

by WINDHORST, A. D, TIMMERMAN, H, KLOK, R. P, MENGE, W. M. P. B, LEURS, R, HERSCHEID, J. D. M
Published in Bioorganic & medicinal chemistry (01.09.1999)

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