Structural insights into biased G protein-coupled receptor signaling revealed by fluorescence spectroscopy
Rahmeh, Rita, Damian, Marjorie, Cottet, Martin, Orcel, Hélène, Mendre, Christiane, Durroux, Thierry, Sharma, K. Shivaji, Durand, Grégory, Pucci, Bernard, Trinquet, Eric, Zwier, Jurriaan M, Deupi, Xavier, Bron, Patrick, Banères, Jean-Louis, Mouillac, Bernard, Granier, Sébastien
Published in Proceedings of the National Academy of Sciences - PNAS (24.04.2012)
Published in Proceedings of the National Academy of Sciences - PNAS (24.04.2012)
Get full text
Journal Article
V1b vasopressin receptor trafficking and signaling: Role of arrestins, G proteins and Src kinase
Perkovska, Sanja, Méjean, Catherine, Ayoub, Mohammed Akli, Li, Juan, Hemery, Floriane, Corbani, Maithé, Laguette, Nadine, Ventura, Maria‐Angeles, Orcel, Hélène, Durroux, Thierry, Mouillac, Bernard, Mendre, Christiane
Published in Traffic (Copenhagen, Denmark) (01.01.2018)
Published in Traffic (Copenhagen, Denmark) (01.01.2018)
Get full text
Journal Article
Red Fluorescent Turn-On Ligands for Imaging and Quantifying G Protein-Coupled Receptors in Living Cells
Karpenko, Iuliia A., Kreder, Rémy, Valencia, Christel, Villa, Pascal, Mendre, Christiane, Mouillac, Bernard, Mély, Yves, Hibert, Marcel, Bonnet, Dominique, Klymchenko, Andrey S.
Published in Chembiochem : a European journal of chemical biology (10.02.2014)
Published in Chembiochem : a European journal of chemical biology (10.02.2014)
Get full text
Journal Article
Biased Agonist Pharmacochaperones of the AVP V2 Receptor May Treat Congenital Nephrogenic Diabetes Insipidus
JEAN-ALPHONSE, Frédéric, PERKOVSKA, Sanja, MENDRE, Christiane, FRANTZ, Marie-Céline, DURROUX, Thierry, MEJEAN, Catherine, MORIN, Denis, LOISON, Stéphanie, BONNET, Dominique, HIBERT, Marcel, MOUILLAC, Bernard
Published in Journal of the American Society of Nephrology (01.10.2009)
Published in Journal of the American Society of Nephrology (01.10.2009)
Get full text
Journal Article
Leukotriene BLT2 Receptor Monomers Activate the Gi2 GTP-binding Protein More Efficiently than Dimers
Arcemisbéhère, Laure, Sen, Tuhinadri, Boudier, Laure, Balestre, Marie-Noëlle, Gaibelet, Gérald, Detouillon, Emilie, Orcel, Hélène, Mendre, Christiane, Rahmeh, Rita, Granier, Sébastien, Vivès, Corinne, Fieschi, Franck, Damian, Marjorie, Durroux, Thierry, Banères, Jean-Louis, Mouillac, Bernard
Published in The Journal of biological chemistry (26.02.2010)
Published in The Journal of biological chemistry (26.02.2010)
Get full text
Journal Article
The constitutively active V2 receptor mutants conferring NSIAD are weakly sensitive to agonist and antagonist regulation
Tenenbaum, Julie, Ayoub, Mohammed A, Perkovska, Sanja, Adra-Delenne, Anne-Laure, Mendre, Christiane, Ranchin, Bruno, Bricca, Giamperro, Geelen, Ghislaine, Mouillac, Bernard, Durroux, Thierry, Morin, Denis
Published in PloS one (21.12.2009)
Published in PloS one (21.12.2009)
Get full text
Journal Article
Differential Coupling of the Vasopressin V1b Receptor through Compartmentalization within the Plasma Membrane
Orcel, Hélène, Albizu, Laura, Perkovska, Sanja, Durroux, Thierry, Mendre, Christiane, Ansanay, Hervé, Mouillac, Bernard, Rabié, Alain
Published in Molecular pharmacology (01.03.2009)
Published in Molecular pharmacology (01.03.2009)
Get full text
Journal Article
Characterization of a G Protein-activated Phosphoinositide 3-Kinase in Vascular Smooth Muscle Cell Nuclei
Bacqueville, Daniel, Déléris, Paul, Mendre, Christiane, Pieraggi, Marie-Thérèse, Chap, Hugues, Guillon, Gilles, Perret, Bertrand, Breton-Douillon, Monique
Published in The Journal of biological chemistry (22.06.2001)
Published in The Journal of biological chemistry (22.06.2001)
Get full text
Journal Article
A Cyclic Peptide Mimicking the Third Intracellular Loop of the V2 Vasopressin Receptor Inhibits Signaling through Its Interaction with Receptor Dimer and G Protein
Granier, Sébastien, Terrillon, Sonia, Pascal, Robert, Déméné, Hélène, Bouvier, Michel, Guillon, Gilles, Mendre, Christiane
Published in The Journal of biological chemistry (03.12.2004)
Published in The Journal of biological chemistry (03.12.2004)
Get full text
Journal Article
Characterization of a functional V1B vasopressin receptor in the male rat kidney: evidence for cross talk between V1B and V2 receptor signaling pathways
Hus-Citharel, Annette, Bouby, Nadine, Corbani, Maithé, Mion, Julie, Mendre, Christiane, Darusi, Judit, Tomboly, Csaba, Trueba, Miguel, Serradeil-Le Gal, Claudine, Llorens-Cortes, Catherine, Guillon, Gilles
Published in American journal of physiology. Renal physiology (01.09.2021)
Published in American journal of physiology. Renal physiology (01.09.2021)
Get full text
Journal Article
Characterization of a functional V 1B vasopressin receptor in the male rat kidney: evidence for cross talk between V 1B and V 2 receptor signaling pathways
Hus-Citharel, Annette, Bouby, Nadine, Corbani, Maithé, Mion, Julie, Mendre, Christiane, Darusi, Judit, Tomboly, Csaba, Trueba, Miguel, Serradeil-Le Gal, Claudine, Llorens-Cortes, Catherine, Guillon, Gilles
Published in American journal of physiology. Renal physiology (01.09.2021)
Published in American journal of physiology. Renal physiology (01.09.2021)
Get full text
Journal Article
Characterization of a functional V 1B vasopressin receptor in the male rat kidney, evidence for crosstalk between V 1B and V 2 receptor signaling pathways
Hus-Citharel, Annette, Bouby, Nadine, Corbani, Maithé, Mion, Julie, Mendre, Christiane, Darusi, Judit, Tomboly, Csaba, Trueba, Miguel, Serradeil-Le Gal, Claudine, Llorens-Cortes, Catherine, Guillon, Gilles
Published in American journal of physiology. Renal physiology (2021)
Published in American journal of physiology. Renal physiology (2021)
Get full text
Journal Article
Green mamba peptide targets type-2 vasopressin receptor against polycystic kidney disease
Ciolek, Justyna, Reinfrank, Helen, Quinton, Loïc, Viengchareun, Say, Stura, Enrico A., Vera, Laura, Sigismeau, Sabrina, Mouillac, Bernard, Orcel, Hélène, Peigneur, Steve, Tytgat, Jan, Droctové, Laura, Beau, Fabrice, Nevoux, Jerome, Lombès, Marc, Mourier, Gilles, De Pauw, Edwin, Servent, Denis, Mendre, Christiane, Witzgall, Ralph, Gilles, Nicolas
Published in Proceedings of the National Academy of Sciences - PNAS (03.07.2017)
Published in Proceedings of the National Academy of Sciences - PNAS (03.07.2017)
Get full text
Journal Article
Web Resource
A new Kunitz‐type snake toxin family associated with an original mode of interaction with the vasopressin 2 receptor
Droctové, Laura, Ciolek, Justyna, Mendre, Christiane, Chorfa, Amélia, Huerta, Paola, Carvalho, Chrystelle, Gouin, Charlotte, Lancien, Manon, Stanajic‐Petrovic, Goran, Braco, Lorine, Blanchet, Guillaume, Upert, Gregory, De Pauw, Gregory, Barbe, Peggy, Keck, Mathilde, Mourier, Gilles, Mouillac, Bernard, Denis, Servent, Rodríguez de la Vega, Ricardo C., Quinton, Loïc, Gilles, Nicolas
Published in British journal of pharmacology (01.07.2022)
Published in British journal of pharmacology (01.07.2022)
Get full text
Journal Article
Web Resource
V 1b vasopressin receptor trafficking and signaling: Role of arrestins, G proteins and Src kinase
Perkovska, Sanja, Méjean, Catherine, Ayoub, Mohammed Akli, Li, Juan, Hemery, Floriane, Corbani, Maithé, Laguette, Nadine, Ventura, Maria-Angeles, Orcel, Hélène, Durroux, Thierry, Mouillac, Bernard, Mendre, Christiane
Published in Traffic (Copenhagen, Denmark) (01.01.2018)
Published in Traffic (Copenhagen, Denmark) (01.01.2018)
Get full text
Journal Article
Crystal structure and functional domains of the Mambaquaretin-1, a vasopressin type 2 receptor peptide inhibitor for kidney cysts treatment
Droctové, Laura, Ciolek, Justyna, Lancien, Manon, Stura, Enrico A., Vera, Laura, Floquet, Nicolas, Witzgall, Ralph, Mouillac, Bernard, Mendre, Christiane, Mourier, Gilles, Servent, Denis, Gilles, Nicolas
Published in Toxicon (Oxford) (01.07.2018)
Published in Toxicon (Oxford) (01.07.2018)
Get full text
Journal Article