Pharmacokinetic Properties of Mirabegron, a β3 -Adrenoceptor Agonist: Results From Two Phase I, Randomized, Multiple-Dose Studies in Healthy Young and Elderly Men and Women
Krauwinkel, Walter, MSc, van Dijk, Jan, BSc, Schaddelee, Marloes, PhD, Eltink, Charlotte, MSc, Meijer, John, MSc, Strabach, Grégory, MD, van Marle, Sjoerd, MD, Kerbusch, Virginie, PhD, van Gelderen, Marcel, PhD
Published in Clinical therapeutics (01.10.2012)
Published in Clinical therapeutics (01.10.2012)
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An Exploratory Study in Healthy Male Subjects of the Mechanism of Mirabegron-Induced Cardiovascular Effects
van Gelderen, Marcel, Stölzel, Matthias, Meijer, John, Kerbusch, Virginie, Collins, Christiane, Korstanje, Cees
Published in Journal of clinical pharmacology (01.12.2017)
Published in Journal of clinical pharmacology (01.12.2017)
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Development of a high-speed synchronous micro motor and its application in intravascular imaging
Wang, Tianshi, Lancée, Charles, Beurskens, Robert, Meijer, John, Knapen, Bart, van der Steen, Antonius F.W., van Soest, Gijs
Published in Sensors and actuators. A. Physical. (01.10.2014)
Published in Sensors and actuators. A. Physical. (01.10.2014)
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Pilocarpine‐Induced Effects on Salivary Secretion as a Pharmacological Biomarker for Cholinergic Parasympathetic Activation
Treijtel, Nicoline, Groenendaal‐van de Meent, Dorien, Michon, Ingrid, Korstanje, Cees, Meijer, John, Francke, Klaus, Grossmann, Matthias, Vries, Michiel
Published in Clinical pharmacology in drug development (01.01.2022)
Published in Clinical pharmacology in drug development (01.01.2022)
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Pharmacokinetics of solifenacin in pediatric populations with overactive bladder or neurogenic detrusor overactivity
Tannenbaum, Stacey, den Adel, Martin, Krauwinkel, Walter, Meijer, John, Hollestein‐Havelaar, Adriana, Verheggen, Frank, Newgreen, Donald
Published in Pharmacology research & perspectives (01.12.2020)
Published in Pharmacology research & perspectives (01.12.2020)
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The effect of mirabegron, a potent and selective β3-adrenoceptor agonist, on the pharmacokinetics of CYP2D6 substrates desipramine and metoprolol
Krauwinkel, Walter, Dickinson, James, Schaddelee, Marloes, Meijer, John, Tretter, Reiner, van de Wetering, Jeroen, Strabach, Gregory, van Gelderen, Marcel
Published in European journal of drug metabolism and pharmacokinetics (01.03.2014)
Published in European journal of drug metabolism and pharmacokinetics (01.03.2014)
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Journal Article
Role of Cytochrome P450 Isoenzymes 3A and 2D6 in the In Vivo Metabolism of Mirabegron, a β3-Adrenoceptor Agonist
Lee, Jennifer, Moy, Selina, Meijer, John, Krauwinkel, Walter, Sawamoto, Taiji, Kerbusch, Virginie, Kowalski, Donna, Roy, Michael, Marion, Alan, Takusagawa, Shin, van Gelderen, Marcel, Keirns, James
Published in Clinical drug investigation (01.06.2013)
Published in Clinical drug investigation (01.06.2013)
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Journal Article
Evaluation of the Pharmacokinetic Interaction Between the β3 -Adrenoceptor Agonist Mirabegron and the Muscarinic Receptor Antagonist Solifenacin In Healthy Subjects
Krauwinkel, Walter J J, Kerbusch, Virginie M M, Meijer, John, Tretter, Reiner, Strabach, Gregory, Van Gelderen, E Marcel
Published in Clinical pharmacology in drug development (01.07.2013)
Published in Clinical pharmacology in drug development (01.07.2013)
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Validation of LC–MS/MS methods for the determination of mirabegron and eight metabolites in human plasma in a paediatric population
Meijer, John, van den Berg, Tom, Huls, Robert, Hofstede, Vincent, Niesing, Willem, van den Beld, Cas, Krauwinkel, Walter
Published in Journal of pharmaceutical and biomedical analysis (15.04.2019)
Published in Journal of pharmaceutical and biomedical analysis (15.04.2019)
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Investigation of Safety and Tolerability of ASP3652 Based on Clinical Studies of Cerebrospinal Fluid Transfer After Multiple Doses and Exposure After Single Doses at High Dose Levels
Takizawa, Masaomi, Cerneus, Dirk, Michon, Ingrid, Rijnders, Sanne, Meijer, John, Someya, Akiyoshi, Sato, Yuichiro
Published in Advances in therapy (01.09.2020)
Published in Advances in therapy (01.09.2020)
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Journal Article
The Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of ASP3652 in First-in-Human and Ascending Multiple Oral Dose Studies in Healthy Subjects
Takizawa, Masaomi, Cerneus, Dirk, Michon, Ingrid, Rijnders, Sanne, van der Heide, Desiree, Meijer, John, Stoelzel, Matthias, Sato, Yuichiro
Published in Advances in therapy (01.09.2020)
Published in Advances in therapy (01.09.2020)
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Journal Article
Absorption, Metabolism and Excretion of [ 14 C]Mirabegron (YM178), a Potent and Selective β 3 -Adrenoceptor Agonist, after Oral Administration to Healthy Male Volunteers
Takusagawa, Shin, van Lier, Jan Jaap, Suzuki, Katsuhiro, Nagata, Masanori, Meijer, John, Krauwinkel, Walter, Schaddelee, Marloes, Sekiguchi, Mitsuhiro, Miyashita, Aiji, Iwatsubo, Takafumi, van Gelderen, Marcel, Usui, Takashi
Published in Drug metabolism and disposition (01.04.2012)
Published in Drug metabolism and disposition (01.04.2012)
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Journal Article
Absorption, metabolism and excretion of [(14)C]mirabegron (YM178), a potent and selective β(3)-adrenoceptor agonist, after oral administration to healthy male volunteers
Takusagawa, Shin, van Lier, Jan Jaap, Suzuki, Katsuhiro, Nagata, Masanori, Meijer, John, Krauwinkel, Walter, Schaddelee, Marloes, Sekiguchi, Mitsuhiro, Miyashita, Aiji, Iwatsubo, Takafumi, van Gelderen, Marcel, Usui, Takashi
Published in Drug metabolism and disposition (01.04.2012)
Published in Drug metabolism and disposition (01.04.2012)
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Development and validation of LC–MS/MS methods for the determination of mirabegron and its metabolites in human plasma and their application to a clinical pharmacokinetic study
van Teijlingen, Raymond, Meijer, John, Takusagawa, Shin, van Gelderen, Marcel, van den Beld, Cas, Usui, Takashi
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.03.2012)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.03.2012)
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Journal Article
Pharmacokinetic Interactions Between Mirabegron and Metformin, Warfarin, Digoxin or Combined Oral Contraceptives
Groen-Wijnberg, Monique, van Dijk, Jan, Krauwinkel, Walter, Kerbusch, Virginie, Meijer, John, Tretter, Reiner, Zhang, Wenhui, van Gelderen, Marcel
Published in European journal of drug metabolism and pharmacokinetics (01.06.2017)
Published in European journal of drug metabolism and pharmacokinetics (01.06.2017)
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