Solution Conformations Shed Light on PROTAC Cell Permeability
Atilaw, Yoseph, Poongavanam, Vasanthanathan, Nilsson, Caroline Svensson, Duy Nguyen, Giese, Anja, Meibom, Daniel, Erdelyi, Mate, Kihlberg, Jan
Published in ACS medicinal chemistry letters (14.01.2021)
Published in ACS medicinal chemistry letters (14.01.2021)
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Potent and Selective Human Prostaglandin F (FP) Receptor Antagonist (BAY-6672) for the Treatment of Idiopathic Pulmonary Fibrosis (IPF)
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Published in Journal of medicinal chemistry (22.10.2020)
Published in Journal of medicinal chemistry (22.10.2020)
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Linker-Dependent Folding Rationalizes PROTAC Cell Permeability
Poongavanam, Vasanthanathan, Atilaw, Yoseph, Siegel, Stephan, Giese, Anja, Lehmann, Lutz, Meibom, Daniel, Erdelyi, Mate, Kihlberg, Jan
Published in Journal of medicinal chemistry (13.10.2022)
Published in Journal of medicinal chemistry (13.10.2022)
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Linker-Dependent Folding Rationalizes PROTAC Cell Permeability br
Poongavanam, Vasanthanathan, Atilaw, Yoseph, Siegel, Stephan, Giese, Anja, Lehmann, Lutz, Meibom, Daniel, Erdélyi, Máté, Kihlberg, Jan
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Published in Journal of medicinal chemistry (28.09.2022)
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High pressure chiral recognition experiments – a route to homochiral 4-fluorocyclohexenones
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BAY-6096: A Potent, Selective, and Highly Water-Soluble Adrenergic ?(2B) Antagonist
Meibom, Daniel, Meyer, Jutta, von Buehler, Clemens-Jeremias, Collins, Karl D., Maassen, Stefanie, Gericke, Kersten Matthias, Hueser, Joerg, Mittendorf, Joachim, Hernandez, Nuria Ortega, Schamberger, Jens, Stampfuss, Jan, Straub, Alexander, Torge, Afra, Witowski, Norbert, Wunder, Frank
Published in Journal of medicinal chemistry (13.04.2023)
Published in Journal of medicinal chemistry (13.04.2023)
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Roehrig, Susanne, Ackerstaff, Jens, Jiménez Núñez, Eloísa, Teller, Henrik, Ellerbrock, Pascal, Meier, Katharina, Heitmeier, Stefan, Tersteegen, Adrian, Stampfuss, Jan, Lang, Dieter, Schlemmer, Karl-Heinz, Schaefer, Martina, Gericke, Kersten M., Kinzel, Tom, Meibom, Daniel, Schmidt, Martina, Gerdes, Christoph, Follmann, Markus, Hillisch, Alexander
Published in Journal of medicinal chemistry (14.09.2023)
Published in Journal of medicinal chemistry (14.09.2023)
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BAY-6096: A Potent, Selective, and Highly Water-Soluble Adrenergic α 2B Antagonist
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Published in Journal of medicinal chemistry (13.04.2023)
Published in Journal of medicinal chemistry (13.04.2023)
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Novel non-xanthine antagonist of the A(2B) adenosine receptor: From HTS hit to lead structure
Haerter, Michael, Kalthof, Bernd, Delbeck, Martina, Lustig, Klemens, Gerisch, Michael, Schulz, Simone, Kast, Raimund, Meibom, Daniel, Lindner, Niels
Published in European journal of medicinal chemistry (01.02.2019)
Published in European journal of medicinal chemistry (01.02.2019)
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BAY-9835: Discovery of the First Orally Bioavailable ADAMTS7 Inhibitor
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Published in Journal of medicinal chemistry (22.12.2022)
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BAY-6096: A Potent, Selective, and Highly Water-Soluble Adrenergic α2B Antagonist
Meibom, Daniel, Meyer, Jutta, von Buehler, Clemens-Jeremias, Collins, Karl D., Maassen, Stefanie, Gericke, Kersten Matthias, Hüser, Jörg, Mittendorf, Joachim, Ortega Hernandez, Nuria, Schamberger, Jens, Stampfuss, Jan, Straub, Alexander, Torge, Afra, Witowski, Norbert, Wunder, Frank
Published in Journal of medicinal chemistry (13.04.2023)
Published in Journal of medicinal chemistry (13.04.2023)
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Novel non-xanthine antagonist of the A2B adenosine receptor: From HTS hit to lead structure
Härter, Michael, Kalthof, Bernd, Delbeck, Martina, Lustig, Klemens, Gerisch, Michael, Schulz, Simone, Kast, Raimund, Meibom, Daniel, Lindner, Niels
Published in European journal of medicinal chemistry (01.02.2019)
Published in European journal of medicinal chemistry (01.02.2019)
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Neladenoson Bialanate Hydrochloride: A Prodrug of a Partial Adenosine A1 Receptor Agonist for the Chronic Treatment of Heart Diseases
Meibom, Daniel, Albrecht‐Küpper, Barbara, Diedrichs, Nicole, Hübsch, Walter, Kast, Raimund, Krämer, Thomas, Krenz, Ursula, Lerchen, Hans‐Georg, Mittendorf, Joachim, Nell, Peter G., Süssmeier, Frank, Vakalopoulos, Alexandros, Zimmermann, Katja
Published in ChemMedChem (22.05.2017)
Published in ChemMedChem (22.05.2017)
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Published in ChemMedChem (22.05.2017)
Published in ChemMedChem (22.05.2017)
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Published in ACS omega (14.02.2023)
Published in ACS omega (14.02.2023)
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Published in ChemMedChem (01.07.2015)
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Published in ChemMedChem (19.01.2016)
Published in ChemMedChem (19.01.2016)
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DELBECK MARTINA, DIETZ LISA, BUCHGRABER PHILIPP, MEIBOM DANIEL, PLATZK MAGDALENA, BECKER PELSTER EVA MARIA, HAHN MICHAEL, MUELLER THOMAS, SCHMECK CARSTEN, LINDNER NIELS
Year of Publication 11.07.2022
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Year of Publication 11.07.2022
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Novel non-xanthine antagonist of the A 2B adenosine receptor: From HTS hit to lead structure
Härter, Michael, Kalthof, Bernd, Delbeck, Martina, Lustig, Klemens, Gerisch, Michael, Schulz, Simone, Kast, Raimund, Meibom, Daniel, Lindner, Niels
Published in European journal of medicinal chemistry (01.02.2019)
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Published in European journal of medicinal chemistry (01.02.2019)
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