The Crystal Structures of Eukaryotic Phosphofructokinases from Baker's Yeast and Rabbit Skeletal Muscle
Banaszak, Katarzyna, Mechin, Ingrid, Obmolova, Galina, Oldham, Michael, Chang, Simon H., Ruiz, Teresa, Radermacher, Michael, Kopperschläger, Gerhard, Rypniewski, Wojciech
Published in Journal of molecular biology (25.03.2011)
Published in Journal of molecular biology (25.03.2011)
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Prevention of Proteinuria by a Novel, Subnanomolar ApoL1 Inhibitor: FR-OR105
Antonio, Brett M., Zahler, Nathan, Mechin, Ingrid, Theile, Jonathan W., Dow, Robert L., Volkmann, Robert A., Zellmer, Shannon G., Chdid, Lhoucine, Nair, Anil, Krafte, Douglas
Published in Journal of the American Society of Nephrology (01.11.2023)
Published in Journal of the American Society of Nephrology (01.11.2023)
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Discovery of N-substituted 7-azaindoles as PIM1 kinase inhibitors – Part I
Barberis, Claude, Moorcroft, Neil, Arendt, Chris, Levit, Mikhail, Moreno-Mazza, Sandra, Batchelor, Joseph, Mechin, Ingrid, Majid, Tahir
Published in Bioorganic & medicinal chemistry letters (15.10.2017)
Published in Bioorganic & medicinal chemistry letters (15.10.2017)
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Molecular basis of action of a small molecule positive allosteric modulator (PAM)-agonist at the type 1 cholecystokinin holoreceptor
Desai, Aditya J, Mechin, Ingrid, Nagarajan, Karthigeyan, Valant, Celine, Wootten, Denise, Lam, Polo C H, Orry, Andrew, Abagyan, Ruben, Nair, Anil, Sexton, Patrick M, Christopoulos, Arthur, Miller, Laurence J
Published in Molecular pharmacology (01.03.2019)
Published in Molecular pharmacology (01.03.2019)
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KV7.2 억제제로서의 신규 헤테로아릴-우레아 화합물
GRAHAM CHRISTOPHER JOHN, NAIR ANIL, DAVIES NICHOLAS GARETH MORSE, SAFAROVA ALENA, MA NINA, LEBRETON SYLVAIN, MOWREY DAVID, REDONDO PENA ROGER LLUIS, GERLACH AARON, SMRCINA MARTIN, MECHIN INGRID, LI RONGHUA, DAVIDSON JAMES, CHAPMAN MARK, NORCROSS ROGER DAVID, NAGARAJAN KARTHIGEYAN
Year of Publication 11.07.2024
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Year of Publication 11.07.2024
Patent
Evaluation of Cancer Dependence and Druggability of PRP4 Kinase Using Cellular, Biochemical, and Structural Approaches
Gao, Qiang, Mechin, Ingrid, Kothari, Nayantara, Guo, Zhuyan, Deng, Gejing, Haas, Kimberly, McManus, Jessica, Hoffmann, Dietmar, Wang, Anlai, Wiederschain, Dmitri, Rocnik, Jennifer, Czechtizky, Werngard, Chen, Xin, McLean, Larry, Arlt, Heike, Harper, David, Liu, Feng, Majid, Tahir, Patel, Vinod, Lengauer, Christoph, Garcia-Echeverria, Carlos, Zhang, Bailin, Cheng, Hong, Dorsch, Marion, Huang, Shih-Min A.
Published in The Journal of biological chemistry (18.10.2013)
Published in The Journal of biological chemistry (18.10.2013)
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결핍된 CFTR 활성에 의해 매개된 병태를 치료하기 위한 5-원 헤테로아릴아미노설폰아미드
FREED BRIAN, BALTZER SYLVIE, GAO ZHONGLI, THURAIRATNAM SUKANTHINI, MA NINA, YEOMAN HELEN, MUNSON MARK, LEBRETON SYLVAIN, LIAO JUNKAI, VIVET BERTRAND, SMRCINA MARTIN, MECHIN INGRID, NESTLER HANS PETER, WIRE WILLIAM, HARTUNG RYAN, HURLBUT GREGORY
Year of Publication 18.08.2022
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Year of Publication 18.08.2022
Patent
Abstract 4376: Evaluation of PRP4 kinase as a potential drug target in cancer
Gao, Qiang, Mechin, Ingrid, Kothari, Nayantara, Guo, Zhuyan, Deng, Gejing, Wang, Anlai, Wiederschain, Dmitri, Rocnik, Jennifer, Czechtizky, Werngard, Liu, Feng, Majid, Tahir, Patel, Vinod, Lengauer, Christoph, Garcia-Echeverria, Carlos, Zhang, Bailin, Cheng, Hong, Dorsch, Marion, Huang, Shih-Min A.
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
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The 10.8-Å structure of Saccharomyces cerevisiae phosphofructokinase determined by cryoelectron microscopy: localization of the putative fructose 6-phosphate binding sites
Ruiz, Teresa, Mechin, Ingrid, Bär, Jörg, Rypniewski, Wojciech, Kopperschläger, Gerhard, Radermacher, Michael
Published in Journal of structural biology (01.08.2003)
Published in Journal of structural biology (01.08.2003)
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PYRIDINE COMPOUNDS AS KV7.2 ENHANCERS
DAVIES, Nicholas Gareth Morse, MOWREY, David, MECHIN, Ingrid, REDONDO PENA, Roger Lluis, NAGARAJAN, Karthigeyan, NAIR, Anil, NORCROSS, Roger David, CHAPMAN, Mark, SMRCINA, Martin, LEBRETON, Sylvain, SAFAROVA, Alena, GERLACH, Aaron
Year of Publication 25.09.2024
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Year of Publication 25.09.2024
Patent
NOVEL HETEROARYL-UREA COMPOUNDS AS KV7.2 INHIBITORS
MOWREY, David, REDONDO PENA, Roger Lluis, NAIR, Anil, NAGARAJAN, Karthigeyan, MA, Nina, LI, Ronghua, DAVIES, Nicholas, MECHIN, Ingrid, NORCROSS, Roger, CHAPMAN, Mark, GRAHAM, Christopher, DAVIDSON, James, SMRCINA, Martin, LEBRETON, Sylvain, SAFAROVA, Alena, GERLACH, Aaron
Year of Publication 30.05.2024
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Year of Publication 30.05.2024
Patent
NOVEL HETEROARYL-UREA COMPOUNDS AS KV7.2 INHIBITORS
MOWREY, David, REDONDO PENA, Roger Lluis, NAIR, Anil, NAGARAJAN, Karthigeyan, MA, Nina, LI, Ronghua, DAVIES, Nicholas, MECHIN, Ingrid, NORCROSS, Roger, CHAPMAN, Mark, GRAHAM, Christopher, DAVIDSON, James, SMRCINA, Martin, LEBRETON, Sylvain, SAFAROVA, Alena, GERLACH, Aaron
Year of Publication 23.05.2024
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Year of Publication 23.05.2024
Patent
PYRIDINE COMPOUNDS AS KV7.2 ENHANCERS
MOWREY, David, REDONDO, Roger, MECHIN, Ingrid, NORCROSS, Roger, NAIR, Anil, NAGARAJAN, Karthigeyan, CHAPMAN, Mark, SMRCINA, Martin, LEBRETON, Sylvain, SAFAROVA, Alena, GERLACH, Aaron, DAVIES, Nicholas Gareth
Year of Publication 25.05.2023
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Year of Publication 25.05.2023
Patent
ARYLAMIDES AND METHODS OF USE THEREOF
Gao, Zhongli, Hurlbut, Gregory, Mechin, Ingrid, Li, Ronghua, Smrcina, Martin, Kim, Joseph, Munson, Mark, Vivet, Bertrand, Hartung, Ryan, Nestler, Hans Peter, Ma, Nina, Bock, William, Liao, Junkai
Year of Publication 25.05.2023
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Year of Publication 25.05.2023
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ARYLAMIDES AND METHODS OF USE THEREOF
Gao, Zhongli, Smrcina, Martin, Scholte, Andrew, Munson, Mark, Vivet, Bertrand, Hurlbut, Gregory, Hartung, Ryan, Nestler, Hans Peter, Mechin, Ingrid, Li, Ronghua, Bock, William, Liao, Junkai
Year of Publication 11.05.2023
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Year of Publication 11.05.2023
Patent
5-MEMBERED HETEROARYLAMINOSULFONAMIDES FOR TREATING CONDITIONS MEDIATED BY DEFICIENT CFTR ACTIVITY
Gao, Zhongli, Freed, Brian, Lebreton, Sylvain, Hurlbut, Gregory, Mechin, Ingrid, Wire, William, Smrcina, Martin, Baltzer, Sylvie, Munson, Mark, Vivet, Bertrand, Hartung, Ryan, Nestler, Hans Peter, Ma, Nina, Yeoman, Helen, Liao, Junkai, Thurairatnam, Sukanthini
Year of Publication 04.01.2024
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Year of Publication 04.01.2024
Patent
NOVEL HETEROARYL-UREA COMPOUNDS AS KV7.2 INHIBITORS
MOWREY, David, REDONDO PENA, Roger Lluis, DAVIES, Nicholas, Gareth Morse, NAGARAJAN, Karthigeyan, NAIR, Anil, MA, Nina, LI, Ronghua, MECHIN, Ingrid, NORCROSS, Roger David, CHAPMAN, Mark, DAVIDSON, James, SMRCINA, Martin, GRAHAM, Christopher, John, LEBRETON, Sylvain, SAFAROVA, Alena, GERLACH, Aaron
Year of Publication 25.09.2024
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Year of Publication 25.09.2024
Patent
Novel heteroaryl-urea compounds as kv7.2 inhibitors
NORCROSS Roger David, LI Ronghua, REDONDO PENA Roger Lluis, DAVIDSON James, GERLACH Aaron, SMRCINA Martin, MA Nina, MECHIN Ingrid, GRAHAM Christopher John, DAVIES Nicholas Gareth Morse, CHAPMAN Mark, NAIR Anil, LEBRETON Sylvain, MOWREY David, NAGARAJAN Karthigeyan, SAFAROVA Alena
Year of Publication 01.07.2024
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Year of Publication 01.07.2024
Patent