The expanding role of prodrugs in contemporary drug design and development
Rautio, Jarkko, Meanwell, Nicholas A, Di, Li, Hageman, Michael J
Published in Nature reviews. Drug discovery (01.08.2018)
Published in Nature reviews. Drug discovery (01.08.2018)
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Metabolic and Pharmaceutical Aspects of Fluorinated Compounds
Johnson, Benjamin M, Shu, Yue-Zhong, Zhuo, Xiaoliang, Meanwell, Nicholas A
Published in Journal of medicinal chemistry (25.06.2020)
Published in Journal of medicinal chemistry (25.06.2020)
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Journal Article
Applications of Fluorine in Medicinal Chemistry
Gillis, Eric P, Eastman, Kyle J, Hill, Matthew D, Donnelly, David J, Meanwell, Nicholas A
Published in Journal of medicinal chemistry (12.11.2015)
Published in Journal of medicinal chemistry (12.11.2015)
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Journal Article
A Survey of the Role of Noncovalent Sulfur Interactions in Drug Design
Beno, Brett R, Yeung, Kap-Sun, Bartberger, Michael D, Pennington, Lewis D, Meanwell, Nicholas A
Published in Journal of medicinal chemistry (11.06.2015)
Published in Journal of medicinal chemistry (11.06.2015)
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Applications of fluorine-containing amino acids for drug design
Mei, Haibo, Han, Jianlin, Klika, Karel D., Izawa, Kunisuke, Sato, Tatsunori, Meanwell, Nicholas A., Soloshonok, Vadim A.
Published in European journal of medicinal chemistry (15.01.2020)
Published in European journal of medicinal chemistry (15.01.2020)
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Journal Article
Tailor‐Made Amino Acids and Fluorinated Motifs as Prominent Traits in Modern Pharmaceuticals
Mei, Haibo, Han, Jianlin, White, Sarah, Graham, Daniel J., Izawa, Kunisuke, Sato, Tatsunori, Fustero, Santos, Meanwell, Nicholas A., Soloshonok, Vadim A.
Published in Chemistry : a European journal (04.09.2020)
Published in Chemistry : a European journal (04.09.2020)
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Journal Article
Synthesis of Cyclobutane-Fused Tetracyclic Scaffolds via Visible-Light Photocatalysis for Building Molecular Complexity
Oderinde, Martins S, Mao, Edna, Ramirez, Antonio, Pawluczyk, Joseph, Jorge, Christine, Cornelius, Lyndon A. M, Kempson, James, Vetrichelvan, Muthalagu, Pitchai, Manivel, Gupta, Anuradha, Gupta, Arun Kumar, Meanwell, Nicholas A, Mathur, Arvind, Dhar, T. G. Murali
Published in Journal of the American Chemical Society (12.02.2020)
Published in Journal of the American Chemical Society (12.02.2020)
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Journal Article
Photocatalytic Dearomative Intermolecular [2+2] Cycloaddition of Heterocycles for Building Molecular Complexity
Oderinde, Martins S., Ramirez, Antonio, Dhar, T. G. Murali, Cornelius, Lyndon A. M., Jorge, Christine, Aulakh, Darpandeep, Sandhu, Bhupinder, Pawluczyk, Joseph, Sarjeant, Amy A., Meanwell, Nicholas A., Mathur, Arvind, Kempson, James
Published in Journal of organic chemistry (15.01.2021)
Published in Journal of organic chemistry (15.01.2021)
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Journal Article
The crystal structure of NS5A domain 1 from genotype 1a reveals new clues to the mechanism of action for dimeric HCV inhibitors
Lambert, Sebastian M., Langley, David R., Garnett, James A., Angell, Richard, Hedgethorne, Katy, Meanwell, Nicholas A., Matthews, Steve J.
Published in Protein science (01.06.2014)
Published in Protein science (01.06.2014)
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Journal Article
Preclinical Profile and Characterization of the Hepatitis C Virus NS3 Protease Inhibitor Asunaprevir (BMS-650032)
MCPHEE, Fiona, SHEAFFER, Amy K, CHAOQUN CHEN, LEE, Min S, MOSURE, Kathy, SUN, Li-Qiang, SINZ, Michael, MEANWELL, Nicholas A, COLONNO, Richard J, KNIPE, Jay, SCOLA, Paul, FRIBORG, Jacques, HERNANDEZ, Dennis, FALK, Paul, GUANGZHI ZHAI, LEVINE, Steven, CHANIEWSKI, Susan, FEI YU, BARRY, Diana
Published in Antimicrobial Agents and Chemotherapy (01.10.2012)
Published in Antimicrobial Agents and Chemotherapy (01.10.2012)
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Homology models of the HIV-1 attachment inhibitor BMS-626529 bound to gp120 suggest a unique mechanism of action
Langley, David R., Roy Kimura, S., Sivaprakasam, Prasanna, Zhou, Nannan, Dicker, Ira, McAuliffe, Brian, Wang, Tao, Kadow, John F., Meanwell, Nicholas A., Krystal, Mark
Published in Proteins, structure, function, and bioinformatics (01.02.2015)
Published in Proteins, structure, function, and bioinformatics (01.02.2015)
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Journal Article
In Vitro Antiviral Characteristics of HIV-1 Attachment Inhibitor BMS-626529, the Active Component of the Prodrug BMS-663068
NOWICKA-SANS, Beata, GONG, Yi-Fei, LI ZHU, MAJUMDAR, Antara, STOCK, David, LATAILLADE, Max, HANNA, George J, MATISKELLA, John D, UEDA, Yasutsugu, TAO WANG, KADOW, John F, MEANWELL, Nicholas A, MCAULIFFE, Brian, KRYSTAL, Mark, DICKER, Ira, HO, Hsu-Tso, NANNAN ZHOU, EGGERS, Betsy, LIN, Pin-Fang, RAY, Neelanjana, WIND-ROTOLO, Megan
Published in Antimicrobial Agents and Chemotherapy (01.07.2012)
Published in Antimicrobial Agents and Chemotherapy (01.07.2012)
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Journal Article
Discovery of BMS-986144, a Third-Generation, Pan-Genotype NS3/4A Protease Inhibitor for the Treatment of Hepatitis C Virus Infection
Sun, Li-Qiang, Mull, Eric, D’Andrea, Stanley, Zheng, Barbara, Hiebert, Sheldon, Gillis, Eric, Bowsher, Michael, Kandhasamy, Sarkunam, Baratam, Venkata Rao, Puttaswamy, Sunitha, Pulicharla, Nagalakshmi, Vishwakrishnan, Sureshbabu, Reddy, Subba, Trivedi, Ravi, Sinha, Sarmistha, Sivaprasad, Sankar, Rao, Abhijith, Desai, Salil, Ghosh, Kaushik, Anumula, Rushith, Kumar, Amit, Rajamani, Ramkumar, Wang, Ying-Kai, Fang, Hua, Mathur, Arvind, Rampulla, Richard, Zvyaga, Tatyana A, Mosure, Kathy, Jenkins, Susan, Falk, Paul, Tagore, Debarati M, Chen, Chaoqun, Rendunchintala, Kishore, Loy, James, Meanwell, Nicholas A, McPhee, Fiona, Scola, Paul M
Published in Journal of medicinal chemistry (10.12.2020)
Published in Journal of medicinal chemistry (10.12.2020)
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Journal Article
Identification of Hepatitis C Virus NS5A Inhibitors
LEMM, Julie A, O'BOYLE, Donald, ROMINE, Jeffrey L, MEANWELL, Nicholas A, MIN GAO, MENGPING LIU, NOWER, Peter T, COLONNO, Richard, DESHPANDE, Milind S, SNYDER, Lawrence B, MARTIN, Scott W, LAURENT, Denis R. St, SERRANO-WU, Michael H
Published in Journal of Virology (01.01.2010)
Published in Journal of Virology (01.01.2010)
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