Effects of channel modulators on cloned large-conductance calcium-activated potassium channels
V K Gribkoff, J T Lum-Ragan, C G Boissard, D J Post-Munson, N A Meanwell, J E Starrett, Jr, E S Kozlowski, J L Romine, J T Trojnacki, M C Mckay, J Zhong, S I Dworetzky
Published in Molecular pharmacology (01.07.1996)
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Published in Molecular pharmacology (01.07.1996)
Journal Article
The substituted benzimidazolone NS004 is an opener of the cystic fibrosis chloride channel
GRIBKOFF, V. K, CHAMPIGNY, G, BARBRY, P, DWORETZKY, S. I, MEANWELL, N. A, LAZDUNSKI, M
Published in The Journal of biological chemistry (15.04.1994)
Published in The Journal of biological chemistry (15.04.1994)
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Journal Article
Opening of large-conductance calcium-activated potassium channels by the substituted benzimidazolone NS004
McKay, M C, Dworetzky, S I, Meanwell, N A, Olesen, S P, Reinhart, P H, Levitan, I B, Adelman, J P, Gribkoff, V K
Published in Journal of neurophysiology (01.05.1994)
Published in Journal of neurophysiology (01.05.1994)
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Journal Article
1,2-Benzisothiazol-3-one 1,1-Dioxide Inhibitors of Human Mast Cell Tryptase
Combrink, Keith D, Gülgeze, H. Belgin, Meanwell, Nicholas A, Pearce, Bradley C, Zulan, Pi, Bisacchi, Gregory S, Roberts, Daniel G. M, Stanley, Paul, Seiler, Steven M
Published in Journal of medicinal chemistry (19.11.1998)
Published in Journal of medicinal chemistry (19.11.1998)
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Journal Article
Salicylamide inhibitors of influenza virus fusion
Combrink, Keith D., Gulgeze, H.Belgin, Yu, Kuo-Long, Pearce, Bradley C., Trehan, Ashok K., Wei, Jianmei, Deshpande, Milind, Krystal, Mark, Torri, Albert, Luo, Guangxiang, Cianci, Christopher, Danetz, Stephanie, Tiley, Laurence, Meanwell, Nicholas A.
Published in Bioorganic & medicinal chemistry letters (07.08.2000)
Published in Bioorganic & medicinal chemistry letters (07.08.2000)
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Journal Article
Active site-directed synthetic thrombin inhibitors: synthesis, in vitro and in vivo activity profile of BMY 44621 and analogs. An examination of the role of the amino group in the D-Phe-Pro-Arg-H series
Balasubramanian, N, St. Laurent, D. R, Federici, M. E, Meanwell, N. A, Wright, J. J, Schumacher, W. A, Seiler, S. M
Published in Journal of medicinal chemistry (1993)
Published in Journal of medicinal chemistry (1993)
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Journal Article
Novel quinolizidine salicylamide influenza fusion inhibitors
Yu, Kuo-Long, Ruediger, Edward, Luo, Guangxiang, Cianci, Christopher, Danetz, Stephanie, Tiley, Laurence, Trehan, Ashok K., Monkovic, Ivo, Pearce, Bradley, Martel, Alain, Krystal, Mark, Meanwell, Nicholas A.
Published in Bioorganic & medicinal chemistry letters (02.08.1999)
Published in Bioorganic & medicinal chemistry letters (02.08.1999)
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Journal Article
Octimibate inhibition of platelet aggregation: stimulation of adenylate cyclase through prostacyclin receptor activation
S Seiler, C L Brassard, A J Arnold, N A Meanwell, J S Fleming, S L Keely, Jr
Published in The Journal of pharmacology and experimental therapeutics (01.12.1990)
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Published in The Journal of pharmacology and experimental therapeutics (01.12.1990)
Journal Article
Imidazoquinoline derivatives: Potent inhibitors of platelet cAMP phosphodiesterase which elevate cAMP levels and activate protein kinase in platelets
Seiler, S., Gillespie, E., Arnold, A.J., Brassard, C.L., Meanwell, N.A., Fleming, J.S.
Published in Thrombosis research (01.04.1991)
Published in Thrombosis research (01.04.1991)
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Journal Article
Azetidin-2-one derivatives as inhibitors of thrombin
Han, William T., Trehan, Ashok K., Kim Wright, J.J., Federici, Marianne E., Seiler, Steven M., Meanwell, Nicholas A.
Published in Bioorganic & medicinal chemistry (01.08.1995)
Published in Bioorganic & medicinal chemistry (01.08.1995)
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Journal Article
HIV-1 entry – an expanding portal for drug discovery
Blair, Wade S, Lin, Pin-Fang, Meanwell, Nicholas A, Wallace, Owen B
Published in Drug Discovery Today (01.05.2000)
Published in Drug Discovery Today (01.05.2000)
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Book Review
Journal Article
Nonprostanoid prostacyclin mimetics. 5. Structure-activity relationships associated with [3-[4-(4,5-diphenyl-2-oxazolyl)-5-oxazolyl]phenoxy]acetic acid
Meanwell, Nicholas A, Romine, Jeffrey L, Rosenfeld, Michael J, Martin, Scott W, Trehan, Ashok K, Wright, J. J. Kim, Malley, Mary F, Gougoutas, Jack Z, Brassard, Catherine L
Published in Journal of medicinal chemistry (26.11.1993)
Published in Journal of medicinal chemistry (26.11.1993)
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Journal Article
1,3-Dihydro-2H-imidazo[4,5-b]quinolin-2-ones - inhibitors of blood platelet cAMP phosphodiesterase and induced aggregation
Meanwell, Nicholas A, Roth, Herbert R, Smith, Edward C. R, Wedding, Donald L, Wright, J. J. Kim, Fleming, J. Stuart, Gillespie, Elizabeth
Published in Journal of medicinal chemistry (01.09.1991)
Published in Journal of medicinal chemistry (01.09.1991)
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Journal Article
Antithrombotic activity of BMY-43351, a new imidazoquinoline with enhanced aqueous solubility
Fleming, J.S., Buchanan, J.O., Seiler, S.M., Meanwell, N.A.
Published in Thrombosis research (01.07.1991)
Published in Thrombosis research (01.07.1991)
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Journal Article
Structure-activity relationships associated with 3,4,5-triphenyl-1H-pyrazole-1-nonanoic acid, a nonprostanoid prostacyclin mimetic
Meanwell, Nicholas A, Rosenfeld, Michael J, Wright, J. J. Kim, Brassard, Catherine L, Buchanan, John O, Federici, Marianne E, Fleming, J. Stuart, Seiler, Steven M
Published in Journal of medicinal chemistry (01.01.1992)
Published in Journal of medicinal chemistry (01.01.1992)
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Journal Article
Discovery of a novel class of BK channel openers : Enantiospecific synthesis and BK channel opening activity of 3-(5-chloro-2-hydroxyphenyl)-1,3-dihydro-3-hydroxy-6-(trifluoromethyl)-2H-indol-2-one
HEWAWASAM, P, MEANWELL, N. A, GRIBKOFF, V. K, DWORETZKY, S. I, BOISSARD, C. G
Published in Bioorganic & medicinal chemistry letters (20.05.1997)
Published in Bioorganic & medicinal chemistry letters (20.05.1997)
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Journal Article