A high-throughput phenotypic screen identifies clofazimine as a potential treatment for cryptosporidiosis
Love, Melissa S, Beasley, Federico C, Jumani, Rajiv S, Wright, Timothy M, Chatterjee, Arnab K, Huston, Christopher D, Schultz, Peter G, McNamara, Case W
Published in PLoS neglected tropical diseases (03.02.2017)
Published in PLoS neglected tropical diseases (03.02.2017)
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Antimalarial Peptide and Polyketide Natural Products from the Fijian Marine Cyanobacterium Moorea producens
Sweeney-Jones, Anne Marie, Gagaring, Kerstin, Antonova-Koch, Jenya, Zhou, Hongyi, Mojib, Nazia, Soapi, Katy, Skolnick, Jeffrey, McNamara, Case W, Kubanek, Julia
Published in Marine drugs (18.03.2020)
Published in Marine drugs (18.03.2020)
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Mitotic evolution of Plasmodium falciparum shows a stable core genome but recombination in antigen families
Bopp, Selina E R, Manary, Micah J, Bright, A Taylor, Johnston, Geoffrey L, Dharia, Neekesh V, Luna, Fabio L, McCormack, Susan, Plouffe, David, McNamara, Case W, Walker, John R, Fidock, David A, Denchi, Eros Lazzerini, Winzeler, Elizabeth A
Published in PLoS genetics (01.02.2013)
Published in PLoS genetics (01.02.2013)
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The ReFRAME library as a comprehensive drug repurposing library and its application to the treatment of cryptosporidiosis
Janes, Jeff, Young, Megan E., Chen, Emily, Rogers, Nicole H., Burgstaller-Muehlbacher, Sebastian, Hughes, Laura D., Love, Melissa S., Hull, Mitchell V., Kuhen, Kelli L., Woods, Ashley K., Joseph, Sean B., Petrassi, H. Michael, McNamara, Case W., Tremblay, Matthew S., Su, Andrew I., Schultz, Peter G., Chatterjee, Arnab K.
Published in Proceedings of the National Academy of Sciences - PNAS (16.10.2018)
Published in Proceedings of the National Academy of Sciences - PNAS (16.10.2018)
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Na+ Regulation in the Malaria Parasite Plasmodium falciparum Involves the Cation ATPase PfATP4 and Is a Target of the Spiroindolone Antimalarials
Spillman, Natalie J., Allen, Richard J.W., McNamara, Case W., Yeung, Bryan K.S., Winzeler, Elizabeth A., Diagana, Thierry T., Kirk, Kiaran
Published in Cell host & microbe (13.02.2013)
Published in Cell host & microbe (13.02.2013)
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Pharmacological and genetic activation of cAMP synthesis disrupts cholesterol utilization in Mycobacterium tuberculosis
Wilburn, Kaley M, Montague, Christine R, Qin, Bo, Woods, Ashley K, Love, Melissa S, McNamara, Case W, Schultz, Peter G, Southard, Teresa L, Huang, Lu, Petrassi, H Michael, VanderVen, Brian C
Published in PLoS pathogens (01.02.2022)
Published in PLoS pathogens (01.02.2022)
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Cell-based screen for discovering lipopolysaccharide biogenesis inhibitors
Zhang, Ge, Baidin, Vadim, Pahil, Karanbir S., Moison, Eileen, Tomasek, David, Ramadoss, Nitya S., Chatterjee, Arnab K., McNamara, Case W., Young, Travis S., Schultz, Peter G., Meredith, Timothy C., Kahne, Daniel
Published in Proceedings of the National Academy of Sciences - PNAS (26.06.2018)
Published in Proceedings of the National Academy of Sciences - PNAS (26.06.2018)
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Antibacterial Oligomeric Polyphenols from the Green Alga Cladophora socialis
Lavoie, Serge, Sweeney-Jones, Anne Marie, Mojib, Nazia, Dale, Brandon, Gagaring, Kerstin, McNamara, Case W, Quave, Cassandra L, Soapi, Katy, Kubanek, Julia
Published in Journal of organic chemistry (03.05.2019)
Published in Journal of organic chemistry (03.05.2019)
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MalDA, Accelerating Malaria Drug Discovery
Yang, Tuo, Ottilie, Sabine, Istvan, Eva S., Godinez-Macias, Karla P., Lukens, Amanda K., Baragaña, Beatriz, Campo, Brice, Walpole, Chris, Niles, Jacquin C., Chibale, Kelly, Dechering, Koen J., Llinás, Manuel, Lee, Marcus C.S., Kato, Nobutaka, Wyllie, Susan, McNamara, Case W., Gamo, Francisco Javier, Burrows, Jeremy, Fidock, David A., Goldberg, Daniel E., Gilbert, Ian H., Wirth, Dyann F., Winzeler, Elizabeth A.
Published in Trends in parasitology (01.06.2021)
Published in Trends in parasitology (01.06.2021)
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High-Content Screening for Cryptosporidium Drug Discovery
Love, Melissa S, McNamara, Case W
Published in Methods in molecular biology (Clifton, N.J.) (01.01.2020)
Published in Methods in molecular biology (Clifton, N.J.) (01.01.2020)
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A suite of phenotypic assays to ensure pipeline diversity when prioritizing drug-like Cryptosporidium growth inhibitors
Jumani, Rajiv S, Hasan, Muhammad M, Stebbins, Erin E, Donnelly, Liam, Miller, Peter, Klopfer, Connor, Bessoff, Kovi, Teixeira, Jose E, Love, Melissa S, McNamara, Case W, Huston, Christopher D
Published in Nature communications (23.04.2019)
Published in Nature communications (23.04.2019)
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Identification of a potent benzoxaborole drug candidate for treating cryptosporidiosis
Lunde, Christopher S, Stebbins, Erin E, Jumani, Rajiv S, Hasan, Md Mahmudul, Miller, Peter, Barlow, John, Freund, Yvonne R, Berry, Pamela, Stefanakis, Rianna, Gut, Jiri, Rosenthal, Philip J, Love, Melissa S, McNamara, Case W, Easom, Eric, Plattner, Jacob J, Jacobs, Robert T, Huston, Christopher D
Published in Nature communications (27.06.2019)
Published in Nature communications (27.06.2019)
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Selective and Specific Inhibition of the Plasmodium falciparum Lysyl-tRNA Synthetase by the Fungal Secondary Metabolite Cladosporin
Hoepfner, Dominic, McNamara, Case W., Lim, Chek Shik, Studer, Christian, Riedl, Ralph, Aust, Thomas, McCormack, Susan L., Plouffe, David M., Meister, Stephan, Schuierer, Sven, Plikat, Uwe, Hartmann, Nicole, Staedtler, Frank, Cotesta, Simona, Schmitt, Esther K., Petersen, Frank, Supek, Frantisek, Glynne, Richard J., Tallarico, John A., Porter, Jeffrey A., Fishman, Mark C., Bodenreider, Christophe, Diagana, Thierry T., Movva, N. Rao, Winzeler, Elizabeth A.
Published in Cell host & microbe (14.06.2012)
Published in Cell host & microbe (14.06.2012)
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Utilizing Chemical Genomics to Identify Cytochrome b as a Novel Drug Target for Chagas Disease
Khare, Shilpi, Roach, Steven L, Barnes, S Whitney, Hoepfner, Dominic, Walker, John R, Chatterjee, Arnab K, Neitz, R Jeffrey, Arkin, Michelle R, McNamara, Case W, Ballard, Jaime, Lai, Yin, Fu, Yue, Molteni, Valentina, Yeh, Vince, McKerrow, James H, Glynne, Richard J, Supek, Frantisek
Published in PLoS pathogens (01.07.2015)
Published in PLoS pathogens (01.07.2015)
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Cryptosporidium life cycle small molecule probing implicates translational repression and an Apetala 2 transcription factor in macrogamont differentiation
Hasan, Muhammad M, Mattice, Ethan B, Teixeira, José E, Jumani, Rajiv S, Stebbins, Erin E, Klopfer, Connor E, Franco, Sebastian E, Love, Melissa S, McNamara, Case W, Huston, Christopher D
Published in PLoS pathogens (26.04.2024)
Published in PLoS pathogens (26.04.2024)
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Spiroindolones, a Potent Compound Class for the Treatment of Malaria
Rottmann, Matthias, McNamara, Case, Yeung, Bryan K.S, Lee, Marcus C.S, Zou, Bin, Russell, Bruce, Seitz, Patrick, Plouffe, David M, Dharia, Neekesh V, Tan, Jocelyn, Cohen, Steven B, Spencer, Kathryn R, González-Páez, Gonzalo E, Lakshminarayana, Suresh B, Goh, Anne, Suwanarusk, Rossarin, Jegla, Timothy, Schmitt, Esther K, Beck, Hans-Peter, Brun, Reto, Nosten, Francois, Renia, Laurent, Dartois, Veronique, Keller, Thomas H, Fidock, David A, Winzeler, Elizabeth A, Diagana, Thierry T
Published in Science (American Association for the Advancement of Science) (03.09.2010)
Published in Science (American Association for the Advancement of Science) (03.09.2010)
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Bicyclic azetidines kill the diarrheal pathogen Cryptosporidium in mice by inhibiting parasite phenylalanyl-tRNA synthetase
Vinayak, Sumiti, Jumani, Rajiv S, Miller, Peter, Hasan, Muhammad M, McLeod, Briana I, Tandel, Jayesh, Stebbins, Erin E, Teixeira, Jose E, Borrel, Julien, Gonse, Arthur, Zhang, Mingliang, Yu, Xianshui, Wernimont, Amy, Walpole, Chris, Eckley, Sean, Love, Melissa S, McNamara, Case W, Sharma, Manmohan, Sharma, Amit, Scherer, Christina A, Kato, Nobutaka, Schreiber, Stuart L, Melillo, Bruno, Striepen, Boris, Huston, Christopher D, Comer, Eamon
Published in Science translational medicine (30.09.2020)
Published in Science translational medicine (30.09.2020)
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Safe drugs with high potential to block malaria transmission revealed by a spleen-mimetic screening
Carucci, Mario, Duez, Julien, Tarning, Joel, García-Barbazán, Irene, Fricot-Monsinjon, Aurélie, Sissoko, Abdoulaye, Dumas, Lucie, Gamallo, Pablo, Beher, Babette, Amireault, Pascal, Dussiot, Michael, Dao, Ming, Hull, Mitchell V, McNamara, Case W, Roussel, Camille, Ndour, Papa Alioune, Sanz, Laura Maria, Gamo, Francisco Javier, Buffet, Pierre
Published in Nature communications (07.04.2023)
Published in Nature communications (07.04.2023)
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Peyssonnosides A–B, Unusual Diterpene Glycosides with a Sterically Encumbered Cyclopropane Motif: Structure Elucidation Using an Integrated Spectroscopic and Computational Workflow
Khatri Chhetri, Bhuwan, Lavoie, Serge, Sweeney-Jones, Anne Marie, Mojib, Nazia, Raghavan, Vijay, Gagaring, Kerstin, Dale, Brandon, McNamara, Case W, Soapi, Katy, Quave, Cassandra L, Polavarapu, Prasad L, Kubanek, Julia
Published in Journal of organic chemistry (05.07.2019)
Published in Journal of organic chemistry (05.07.2019)
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