Discovery of benzothiazole amides as potent antimycobacterial agents
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Published in Bioorganic & medicinal chemistry letters (15.10.2018)
Published in Bioorganic & medicinal chemistry letters (15.10.2018)
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RET 키나제를 억제하는데 유용한 화합물
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Year of Publication 09.01.2023
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RET 키나제 억제제로서의 피라졸 유도체
ANDREWS STEVEN W, MCKENNEY MEGAN L, PINTO MARTA, CONDROSKI KEVIN R, MCFADDIN ELIZABETH A, KOLAKOWSKI GABRIELLE R. A, IRVIN THOMAS C, MCLEAN JOHNATHAN ALEXANDER, ANDERSON ERIN D, KUMAR MANOJ, PILKINGTON MIKSA MICHAEL ALEXANDER, BOLDRON CHRISTOPHER PIERRE ALBERT JEAN, MOURET TIPHAINE, MUNCHHOF MICHAEL J, PANCALDI THOMAS PIERRE DINO
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Year of Publication 07.07.2023
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결정질 형태
JIANG YUTONG, KOLAKOWSKI GABRIELLE R, FRY DAVID, MCFADDIN ELIZABETH A, HAAS JULIA, METCALF ANDREW T, TANG TONY P
Year of Publication 13.05.2020
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Year of Publication 13.05.2020
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RET 키나제 억제제로서의 치환된 피라졸로[1,5-A]피리딘 화합물
JIANG YUTONG, ANDREWS STEVEN W, MCKENNEY MEGAN L, MORENO DAVID A, MCNULTY OREN T, BRANDHUBER BARBARA J, KOLAKOWSKI GABRIELLE R, COLLIER JAMES, MCFADDIN ELIZABETH A, RAMANN GINELLE A, HAAS JULIA, TANG TONY P, BLAKE JAMES F, REN LI, ARONOW SEAN, WALLS SHANE M, METCALF ANDREW T, COOK ADAM
Year of Publication 03.07.2019
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Year of Publication 03.07.2019
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RET 키나제 억제제로서의 치환된 피라졸로[1,5-A]피리딘 화합물
JIANG YUTONG, ANDREWS STEVEN W, MCKENNEY MEGAN L, MORENO DAVID A, MCNULTY OREN T, BRANDHUBER BARBARA J, KOLAKOWSKI GABRIELLE R, MCFADDIN ELIZABETH A, HAAS JULIA, TANG TONY P, BLAKE JAMES F, REN LI, ARONOW SEAN, METCALF ANDREW T, COOK ADAM
Year of Publication 02.07.2019
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Year of Publication 02.07.2019
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NOVEL ANTIMYCOBACTERIAL HETEROCYCLIC AMIDES
JARVIS, Thale, WONG, Christina, GRAHAM, James, MCFADDIN, Elizabeth, SUN, Xicheng, OCHSNER, Urs, DAY, Joshua
Year of Publication 16.10.2024
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Year of Publication 16.10.2024
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Antimycobacterial heterocyclic amides
Jarvis, Thale, Mcfaddin, Elizabeth, Day, Joshua, Sun, Xicheng, Wong, Christina, Ochsner, Urs, Graham, James
Year of Publication 23.05.2023
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Year of Publication 23.05.2023
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Processes and intermediates for the preparation of (s)-5-amino-3-(4-((5-fluoro-2-methoxybenzamido)methyl)phenyl)-1-(1,1,1-trifluoropropane-2-yl)-1H-pyrazole-4-carboxamide
ROTHHAAR, Roger Ryan, ARGUELLES DELGADO, Alonso Jose, FRANK, Scott Alan, MCFADDIN, Elizabeth Ann, EARY, Charles Todd, SPENCER, Stacey Renee, FENNELL, Jared Wade, MAGNUS, Nicholas Andrew, VAID, Radhe Krishan
Year of Publication 23.05.2024
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Year of Publication 23.05.2024
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PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF (S)-5-AMINO-3-(4-((5-FLUORO-2-METHOXYBENZAMIDO)METHYL)PHENYL)-1-(1,1,1-TRIFLUOROPROPANE-2-YL)-1H-PYRAZOLE-4-CARBOXAMIDE
ROTHHAAR, Roger Ryan, ARGUELLES DELGADO, Alonso Jose, FRANK, Scott Alan, MCFADDIN, Elizabeth Ann, EARY, Charles Todd, SPENCER, Stacey Renee, FENNELL, Jared Wade, MAGNUS, Nicholas Andrew, VAID, Radhe Krishan
Year of Publication 09.05.2024
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Year of Publication 09.05.2024
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Compounds useful for inhibiting RET kinase
Anderson, Erin D, Munchhof, Michael J, Welch, Michael B, Andrews, Steven W, McKenney, Megan, Irvin, Thomas C, Kumar, Manoj, McFaddin, Elizabeth A, Condroski, Kevin R, Kolakowski, Gabrielle R
Year of Publication 23.04.2024
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Year of Publication 23.04.2024
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CRYSTALLINE FORMS
FRY, DAVID, TANG, TONY P, JIANG, YUTONG, METCALF, ANDREW T, KOLAKOWSKI, GABRIELLE R, HAAS, JULIA, MCFADDIN, ELIZABETH A
Year of Publication 24.01.2023
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Year of Publication 24.01.2023
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NOVEL ANTIMYCOBACTERIAL HETEROCYCLIC AMIDES
JARVIS, Thale, WONG, Christina, GRAHAM, James, MCFADDIN, Elizabeth, SUN, Xicheng, OCHSNER, Urs, DAY, Joshua
Year of Publication 23.02.2022
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Year of Publication 23.02.2022
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PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF (S)-5-AMINO-3-(4-((5-FLUORO-2-METHOXYBENZAMIDO)METHYL)PHENYL)-1-(1,1,1-TRIFLUOROPROPANE-2-YL)-1H-PYRAZOLE-4-CARBOXAMIDE
ROTHHAAR, Roger Ryan, ARGUELLES DELGADO, Alonso Jose, FRANK, Scott Alan, MCFADDIN, Elizabeth Ann, EARY, Charles Todd, SPENCER, Stacey Renee, FENNELL, Jared Wade, MAGNUS, Nicholas Andrew, VAID, Radhe Krishan
Year of Publication 12.10.2023
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Year of Publication 12.10.2023
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COMPOUNDS USEFUL FOR INHIBITING RET KINASE
ANDERSON, Erin D, ANDREWS, Steven W, MCKENNEY, Megan, IRVIN, Thomas C, KUMAR, Manoj, WELCH, Michael B, KOLAKOWSKI, Gabrielle R, CONDROSKI, Kevin R, MUNCHHOF, Michael J, MCFADDIN, Elizabeth A
Year of Publication 05.10.2023
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Year of Publication 05.10.2023
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PYRAZOLE DERIVATIVES ASR ET KINASE INHIBITORS
PANCALDI, Thomas, KOLAKOWSKI, Gabrielle, BOLDRON, Christopher, MCKENNEY, Megan, CONDROSKI, Kevin, MUNCHHOF, Michael, ANDERSON, Erin, ANDREWS, Steven, IRVIN, Thomas, KUMAR, Manoj, MCFADDIN, Elizabeth, MCLEAN, Johnathan, PILKINGTON-MIKSA, Michael Alexander, PINTO, Marta, MOURET, Tiphaine
Year of Publication 01.08.2024
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Year of Publication 01.08.2024
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PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF (S)-5-AMINO-3-(4-((5-FLUORO-2-METHOXYBENZAMIDO)METHYL)PHENYL)-1-(1,1,1-TRIFLUOROPROPANE-2-YL)-1H-PYRAZOLE-4-CARBOXAMIDE
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Year of Publication 19.07.2023
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Year of Publication 19.07.2023
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Substituted pyrazolo[1,5-a]pyridine compounds as RET kinase inhibitors
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Year of Publication 04.06.2024
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Year of Publication 04.06.2024
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Fused heterocyclic compounds as RET kinase inhibitors
Ramann, Ginelle A, Prigaro, Brett, Zhang, Hailong, Blake, James F, McKenney, Megan L, McFaddin, Elizabeth A, Haas, Julia, Kolakowski, Gabrielle R, Kahn, Dean, Dai, Donghua, Metcalf, Andrew T, Ren, Li, Jiang, Yutong, Moreno, David A, Walls, Shane M
Year of Publication 23.04.2024
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Year of Publication 23.04.2024
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