Fadraciclib (CYC065), a novel CDK inhibitor, targets key pro-survival and oncogenic pathways in cancer
Frame, Sheelagh, Saladino, Chiara, MacKay, Craig, Atrash, Butrus, Sheldrake, Peter, McDonald, Edward, Clarke, Paul A, Workman, Paul, Blake, David, Zheleva, Daniella
Published in PloS one (09.07.2020)
Published in PloS one (09.07.2020)
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Novel Clinical and Pathologic Findings in a Heartland Virus—Associated Death
Fill, Mary—Margaret A., Compton, Margaret L., McDonald, Edward C., Moncayo, Abelardo C., Schaffner, John R. Dunn William, Bhatnagar, Julu, Zaki, Sherif R., Jones, Timothy F., Shieh, Wun—Ju
Published in Clinical infectious diseases (15.02.2017)
Published in Clinical infectious diseases (15.02.2017)
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NVP-AUY922: a novel heat shock protein 90 inhibitor active against xenograft tumor growth, angiogenesis, and metastasis
Eccles, Suzanne A, Massey, Andy, Raynaud, Florence I, Sharp, Swee Y, Box, Gary, Valenti, Melanie, Patterson, Lisa, de Haven Brandon, Alexis, Gowan, Sharon, Boxall, Frances, Aherne, Wynne, Rowlands, Martin, Hayes, Angela, Martins, Vanessa, Urban, Frederique, Boxall, Kathy, Prodromou, Chrisostomos, Pearl, Laurence, James, Karen, Matthews, Thomas P, Cheung, Kwai-Ming, Kalusa, Andrew, Jones, Keith, McDonald, Edward, Barril, Xavier, Brough, Paul A, Cansfield, Julie E, Dymock, Brian, Drysdale, Martin J, Finch, Harry, Howes, Rob, Hubbard, Roderick E, Surgenor, Alan, Webb, Paul, Wood, Mike, Wright, Lisa, Workman, Paul
Published in Cancer research (Chicago, Ill.) (15.04.2008)
Published in Cancer research (Chicago, Ill.) (15.04.2008)
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Biological properties of potent inhibitors of class I phosphatidylinositide 3-kinases: from PI-103 through PI-540, PI-620 to the oral agent GDC-0941
Raynaud, Florence I, Eccles, Suzanne A, Patel, Sonal, Alix, Sonia, Box, Gary, Chuckowree, Irina, Folkes, Adrian, Gowan, Sharon, De Haven Brandon, Alexis, Di Stefano, Francesca, Hayes, Angela, Henley, Alan T, Lensun, Letitia, Pergl-Wilson, Giles, Robson, Anthony, Saghir, Nahid, Zhyvoloup, Alexander, McDonald, Edward, Sheldrake, Peter, Shuttleworth, Stephen, Valenti, Melanie, Wan, Nan Chi, Clarke, Paul A, Workman, Paul
Published in Molecular cancer therapeutics (01.07.2009)
Published in Molecular cancer therapeutics (01.07.2009)
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MAGNETIC RESONANCE IMAGING OF LATERAL MENISCAL POSTERIOR ROOT TEARS IN THE ADOLESCENT KNEE: IS THE DIAGNOSIS MISSED, MENTIONED, OR MADE?
Schlechter, John A., Gornick, Bryn, McDonald, Edward J., Pak, Theresa
Published in Orthopaedic journal of sports medicine (01.07.2021)
Published in Orthopaedic journal of sports medicine (01.07.2021)
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Mechanism-based screen for G1/S checkpoint activators identifies a selective activator of EIF2AK3/PERK signalling
Stockwell, Simon R, Platt, Georgina, Barrie, S Elaine, Zoumpoulidou, Georgia, Te Poele, Robert H, Aherne, G Wynne, Wilson, Stuart C, Sheldrake, Peter, McDonald, Edward, Venet, Mathilde, Soudy, Christelle, Elustondo, Frédéric, Rigoreau, Laurent, Blagg, Julian, Workman, Paul, Garrett, Michelle D, Mittnacht, Sibylle
Published in PloS one (12.01.2012)
Published in PloS one (12.01.2012)
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Molecular profiling and combinatorial activity of CCT068127: a potent CDK2 and CDK9 inhibitor
Whittaker, Steven R., Barlow, Clare, Martin, Mathew P., Mancusi, Caterina, Wagner, Steve, Self, Annette, Barrie, Elaine, Te Poele, Robert, Sharp, Swee, Brown, Nathan, Wilson, Stuart, Jackson, Wayne, Fischer, Peter M., Clarke, Paul A., Walton, Michael I., McDonald, Edward, Blagg, Julian, Noble, Martin, Garrett, Michelle D., Workman, Paul
Published in Molecular oncology (01.03.2018)
Published in Molecular oncology (01.03.2018)
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A Useful Approach to Identify Novel Small-Molecule Inhibitors of Wnt-Dependent Transcription
EWAN, Kenneth, PAJAK, Bożena, BATTERSBY, Alysia, RAYNAUD, Florence, ALLEN, Nicholas, WILSON, Stephen, LATINKIC, Branko, WORKMAN, Paul, MCDONALD, Edward, BLAGG, Julian, AHERNE, Wynne, DALE, Trevor, STUBBS, Mark, TODD, Helen, BARBEAU, Olivier, QUEVEDO, Camilo, BOTFIELD, Hannah, YOUNG, Rodrigo, RUDDLE, Ruth, SAMUEL, Lee
Published in Cancer research (Chicago, Ill.) (15.07.2010)
Published in Cancer research (Chicago, Ill.) (15.07.2010)
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Discovery and development of pyrazole-scaffold Hsp90 inhibitors
McDonald, Edward, Jones, Keith, Brough, Paul A, Drysdale, Martin J, Workman, Paul
Published in Current topics in medicinal chemistry (01.06.2006)
Published in Current topics in medicinal chemistry (01.06.2006)
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Inhibitors of the HSP90 molecular chaperone: attacking the master regulator in cancer
McDonald, Edward, Workman, Paul, Jones, Keith
Published in Current topics in medicinal chemistry (01.06.2006)
Published in Current topics in medicinal chemistry (01.06.2006)
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Journal Article
Novel, Potent Small-Molecule Inhibitors of the Molecular Chaperone Hsp90 Discovered through Structure-Based Design
Dymock, Brian W, Barril, Xavier, Brough, Paul A, Cansfield, Julie E, Massey, Andrew, McDonald, Edward, Hubbard, Roderick E, Surgenor, Allan, Roughley, Stephen D, Webb, Paul, Workman, Paul, Wright, Lisa, Drysdale, Martin J
Published in Journal of medicinal chemistry (30.06.2005)
Published in Journal of medicinal chemistry (30.06.2005)
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Isothiazolones as inhibitors of PCAF and p300 histone acetyltransferase activity
Stimson, Lindsay, Rowlands, Martin G, Newbatt, Yvette M, Smith, Nicola F, Raynaud, Florence I, Rogers, Paul, Bavetsias, Vassilios, Gorsuch, Stephen, Jarman, Michael, Bannister, Andrew, Kouzarides, Tony, McDonald, Edward, Workman, Paul, Aherne, G Wynne
Published in Molecular cancer therapeutics (01.10.2005)
Published in Molecular cancer therapeutics (01.10.2005)
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Inhibition of the heat shock protein 90 molecular chaperone in vitro and in vivo by novel, synthetic, potent resorcinylic pyrazole/isoxazole amide analogues
Sharp, Swee Y, Prodromou, Chrisostomos, Boxall, Kathy, Powers, Marissa V, Holmes, Joanna L, Box, Gary, Matthews, Thomas P, Cheung, Kwai-Ming J, Kalusa, Andrew, James, Karen, Hayes, Angela, Hardcastle, Anthea, Dymock, Brian, Brough, Paul A, Barril, Xavier, Cansfield, Julie E, Wright, Lisa, Surgenor, Allan, Foloppe, Nicolas, Hubbard, Roderick E, Aherne, Wynne, Pearl, Laurence, Jones, Keith, McDonald, Edward, Raynaud, Florence, Eccles, Sue, Drysdale, Martin, Workman, Paul
Published in Molecular cancer therapeutics (01.04.2007)
Published in Molecular cancer therapeutics (01.04.2007)
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Nonlinear progressive wave equation for stratified atmospheres
Edward McDonald, B, Piacsek, Andrew A
Published in The Journal of the Acoustical Society of America (01.11.2011)
Published in The Journal of the Acoustical Society of America (01.11.2011)
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Enhanced sound transmission from water to air at low frequencies
McDonald, B Edward, Calvo, David C
Published in The Journal of the Acoustical Society of America (01.12.2007)
Published in The Journal of the Acoustical Society of America (01.12.2007)
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In vitro biological characterization of a novel, synthetic diaryl pyrazole resorcinol class of heat shock protein 90 inhibitors
SHARP, Swee Y, BOXALL, Kathy, PATTERSON, Lisa, MATTHEWS, Thomas P, CHEUNG, Kwai-Ming J, BALL, Karen, HAYES, Angela, RAYNAUD, Florence, MARAIS, Richard, PEARL, Laurence, ECCLES, Sue, AHERNE, Wynne, ROWLANDS, Martin, MCDONALD, Edward, WORKMAN, Paul, PRODROMOU, Chrisostomos, ROE, S. Mark, MALONEY, Alison, POWERS, Marissa, CLARKE, Paul A, BOX, Gary, SANDERSON, Sharon
Published in Cancer research (Chicago, Ill.) (01.03.2007)
Published in Cancer research (Chicago, Ill.) (01.03.2007)
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Mechanism of action of the Aurora kinase inhibitor CCT129202 and in vivo quantification of biological activity
Chan, Florence, Sun, Chongbo, Perumal, Meg, Nguyen, Quang-De, Bavetsias, Vassilios, McDonald, Edward, Martins, Vanessa, Wilsher, Nicola E, Raynaud, Florence I, Valenti, Melanie, Eccles, Sue, Te Poele, Robert, Workman, Paul, Aboagye, Eric O, Linardopoulos, Spiros
Published in Molecular cancer therapeutics (01.12.2007)
Published in Molecular cancer therapeutics (01.12.2007)
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