Design, Synthesis, and SAR of New Pyrrole-Oxindole Progesterone Receptor Modulators Leading to 5-(7-Fluoro-3,3-dimethyl-2-oxo-2,3-dihydro-1H-indol-5-yl)-1-methyl-1H-pyrrole-2-carbonitrile (WAY-255348)
Fensome, Andrew, Adams, William R, Adams, Andrea L, Berrodin, Tom J, Cohen, Jeff, Huselton, Christine, Illenberger, Arthur, Kern, Jeffrey C, Hudak, Valerie A, Marella, Michael A, Melenski, Edward G, McComas, Casey C, Mugford, Cheryl A, Slayden, Ov D, Yudt, Matthew, Zhang, Zhiming, Zhang, Puwen, Zhu, Yuan, Winneker, Richard C, Wrobel, Jay E
Published in Journal of medicinal chemistry (27.03.2008)
Published in Journal of medicinal chemistry (27.03.2008)
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A new generation of progesterone receptor modulators
Winneker, Richard C., Fensome, Andrew, Zhang, Puwen, Yudt, Matthew R., McComas, Casey C., Unwalla, Rayomond J.
Published in Steroids (01.08.2008)
Published in Steroids (01.08.2008)
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Development of a New Structural Class of Broadly Acting HCV Non‐Nucleoside Inhibitors Leading to the Discovery of MK‐8876
McComas, Casey C., Palani, Anandan, Chang, Wei, Holloway, M. Katharine, Lesburg, Charles A., Li, Peng, Liverton, Nigel, Meinke, Peter T., Olsen, David B., Peng, Xuanjia, Soll, Richard M., Ummat, Ajay, Wu, Jie, Wu, Jin, Zorn, Nicolas, Ludmerer, Steven W.
Published in ChemMedChem (07.09.2017)
Published in ChemMedChem (07.09.2017)
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A general approach to access 5,6-dihydroindolo-naphthyridine ring system
He, Shuwen, Li, Peng, Dai, Xing, Liu, Hong, Lai, Zhong, Xiao, Dong, McComas, Casey C., Du, Chunyan, Liu, Yuehui, Yin, Jingjun, Dang, Qun, Zorn, Nicolas, Peng, Xuanjia, Nargund, Ravi P., Palani, Anandan
Published in Tetrahedron letters (05.04.2017)
Published in Tetrahedron letters (05.04.2017)
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Front Cover: Development of a New Structural Class of Broadly Acting HCV Non‐Nucleoside Inhibitors Leading to the Discovery of MK‐8876 (ChemMedChem 17/2017)
McComas, Casey C., Palani, Anandan, Chang, Wei, Holloway, M. Katharine, Lesburg, Charles A., Li, Peng, Liverton, Nigel, Meinke, Peter T., Olsen, David B., Peng, Xuanjia, Soll, Richard M., Ummat, Ajay, Wu, Jie, Wu, Jin, Zorn, Nicolas, Ludmerer, Steven W.
Published in ChemMedChem (07.09.2017)
Published in ChemMedChem (07.09.2017)
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Facile functionalization at the C2 position of a highly substituted benzofuran
He, Shuwen, Li, Peng, Dai, Xing, McComas, Casey C., Du, Chunyan, Wang, Ping, Lai, Zhong, Liu, Hong, Yin, Jingjun, Bulger, Paul G., Dang, Qun, Xiao, Dong, Zorn, Nicolas, Peng, Xuanjia, Nargund, Ravi P., Palani, Anandan
Published in Tetrahedron letters (02.04.2014)
Published in Tetrahedron letters (02.04.2014)
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Journal Article
Total Synthesis of the Ristocetin Aglycon
Crowley, Brendan M, Mori, Yoshiki, McComas, Casey C, Tang, Datong, Boger, Dale L
Published in Journal of the American Chemical Society (07.04.2004)
Published in Journal of the American Chemical Society (07.04.2004)
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Discovery of Novel Selective Norepinephrine Reuptake Inhibitors: 4-[3-Aryl-2,2-dioxido-2,1,3-benzothiadiazol-1(3H)-yl]-1-(methylamino)butan-2-ols (WYE-103231)
O’Neill, David J, Adedoyin, Adedayo, Alfinito, Peter D, Bray, Jenifer A, Cosmi, Scott, Deecher, Darlene C, Fensome, Andrew, Harrison, Jim, Leventhal, Liza, Mann, Charles, McComas, Casey C, Sullivan, Nicole R, Spangler, Taylor B, Uveges, Albert J, Trybulski, Eugene J, Whiteside, Garth T, Zhang, Puwen
Published in Journal of medicinal chemistry (10.06.2010)
Published in Journal of medicinal chemistry (10.06.2010)
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Structure–activity relationships of norepinephrine reuptake inhibitors with benzothiadiazine dioxide or dihydrosulfostyril cores
Fensome, Andrew, Goldberg, Joel, McComas, Casey C., Trybulski, Eugene J., Woodworth, Richard P., Deecher, Darlene C., Whiteside, Garth T., Zhang, Puwen
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
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Synthesis and activity of novel 1-or 3-(3-amino-1-phenyl propyl)-1,3-dihydro-2H-benzimidazol-2-ones as selective norepinephrine reuptake inhibitors
PUWEN ZHANG, TEREFENKO, Eugene A, MCCOMAS, Casey C, MAHANEY, Paige E, AN VU, TRYBULSKI, Eugene, KOURY, Elizabeth, JOHNSTON, Grace, BRAY, Jenifer, DEECHER, Darlene
Published in Bioorganic & medicinal chemistry (01.12.2008)
Published in Bioorganic & medicinal chemistry (01.12.2008)
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Synthesis and activity of a new class of dual acting norepinephrine and serotonin reuptake inhibitors: 3-(1 H-indol-1-yl)-3-arylpropan-1-amines
Mahaney, Paige E., Vu, An T., McComas, Casey C., Zhang, Puwen, Nogle, Lisa M., Watts, William L., Sarkahian, Ani, Leventhal, Liza, Sullivan, Nicole R., Uveges, Albert J., Trybulski, Eugene J.
Published in Bioorganic & medicinal chemistry (15.12.2006)
Published in Bioorganic & medicinal chemistry (15.12.2006)
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Large-Scale Synthesis of a Selective Inhibitor of the Norepinephrine Transporter: Mechanistic Aspects of Conversion of Indolinone Diol to Indolinone Aminoalcohol and Process Implications
Alimardanov, Asaf, Gontcharov, Alexander, Nikitenko, Antonia, Chan, Anita W, Ding, Zhixian, Ghosh, Mousumi, Levent, Mahmut, Raveendranath, Panolil, Ren, Jianxin, Zhou, Maotang, Mahaney, Paige E, McComas, Casey C, Ashcroft, Joseph, Potoski, John R
Published in Organic process research & development (18.09.2009)
Published in Organic process research & development (18.09.2009)
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1- or 3-(3-Amino-2-hydroxy-1-phenyl propyl)-1,3-dihydro-2H-benzimidazol-2-ones: Potent, Selective, and Orally Efficacious Norepinephrine Reuptake Inhibitors
Zhang, Puwen, Terefenko, Eugene A., Bray, Jenifer, Deecher, Darlene, Fensome, Andrew, Harrison, Jim, Kim, Callain, Koury, Elizabeth, Mark, Lilly, McComas, Casey C., Mugford, Cheryl A., Trybulski, Eugene J., Vu, An T., Whiteside, Garth T., Mahaney, Paige E.
Published in Journal of medicinal chemistry (24.09.2009)
Published in Journal of medicinal chemistry (24.09.2009)
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A new and improved method for deglycosidation of glycopeptide antibiotics exemplified with vancomycin, ristocetin, and ramoplanin
Wanner, Jutta, Tang, Datong, McComas, Casey C, Crowley, Brendan M, Jiang, Wanlong, Moss, Jason, Boger, Dale L
Published in Bioorganic & medicinal chemistry letters (24.03.2003)
Published in Bioorganic & medicinal chemistry letters (24.03.2003)
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Dianions and Tetraanions of Bowl-Shaped Fullerene Fragments Dibenzo[a,g]corannulene and Dibenzo[a,g]cyclopenta[kl]corannulene
Weitz, Amir, Shabtai, Elad, Rabinovitz, Mordecai, Bratcher, Matthew S., McComas, Casey C., Best, Michael D., Scott, Lawrence T.
Published in Chemistry : a European journal (10.02.1998)
Published in Chemistry : a European journal (10.02.1998)
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Stereochemistry of 3-Alkylindole Dimerization: Acyclic δ1,δ1‘-Tryptophan Dimers
McComas, Casey C, Gilbert, Eric J, Van Vranken, David L
Published in Journal of organic chemistry (28.11.1997)
Published in Journal of organic chemistry (28.11.1997)
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