Nucleo-cytoplasmic transport as a therapeutic target of cancer
Gravina, Giovanni Luca, Senapedis, William, McCauley, Dilara, Baloglu, Erkan, Shacham, Sharon, Festuccia, Claudio
Published in Journal of hematology and oncology (05.12.2014)
Published in Journal of hematology and oncology (05.12.2014)
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Inhibition of the Nuclear Export Receptor XPO1 as a Therapeutic Target for Platinum-Resistant Ovarian Cancer
Chen, Ying, Camacho, Sandra Catalina, Silvers, Thomas R, Razak, Albiruni R A, Gabrail, Nashat Y, Gerecitano, John F, Kalir, Eva, Pereira, Elena, Evans, Brad R, Ramus, Susan J, Huang, Fei, Priedigkeit, Nolan, Rodriguez, Estefania, Donovan, Michael, Khan, Faisal, Kalir, Tamara, Sebra, Robert, Uzilov, Andrew, Chen, Rong, Sinha, Rileen, Halpert, Richard, Billaud, Jean-Noel, Shacham, Sharon, McCauley, Dilara, Landesman, Yosef, Rashal, Tami, Kauffman, Michael, Mirza, Mansoor R, Mau-Sørensen, Morten, Dottino, Peter, Martignetti, John A
Published in Clinical cancer research (15.03.2017)
Published in Clinical cancer research (15.03.2017)
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XPO1 (CRM1) inhibition represses STAT3 activation to drive a survivin-dependent oncogenic switch in triple-negative breast cancer
Cheng, Yan, Holloway, Michael P, Nguyen, Kevin, McCauley, Dilara, Landesman, Yosef, Kauffman, Michael G, Shacham, Sharon, Altura, Rachel A
Published in Molecular cancer therapeutics (01.03.2014)
Published in Molecular cancer therapeutics (01.03.2014)
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Nuclear export inhibitors avert progression in preclinical models of inflammatory demyelination
Haines, Jeffery D, Herbin, Olivier, de la Hera, Belén, Vidaurre, Oscar G, Moy, Gregory A, Sun, Qingxiang, Fung, Ho Yee Joyce, Albrecht, Stefanie, Alexandropoulos, Konstantina, McCauley, Dilara, Chook, Yuh Min, Kuhlmann, Tanja, Kidd, Grahame J, Shacham, Sharon, Casaccia, Patrizia
Published in Nature neuroscience (01.04.2015)
Published in Nature neuroscience (01.04.2015)
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Journal Article
XPO1/CRM1-selective inhibitors of nuclear export (SINE) reduce tumor spreading and improve overall survival in preclinical models of prostate cancer (PCa)
Gravina, Giovanni Luca, Tortoreto, Monica, Mancini, Andrea, Addis, Alessandro, Di Cesare, Ernesto, Lenzi, Andrea, Landesman, Yosef, McCauley, Dilara, Kauffman, Michael, Shacham, Sharon, Zaffaroni, Nadia, Festuccia, Claudio
Published in Journal of hematology and oncology (05.10.2014)
Published in Journal of hematology and oncology (05.10.2014)
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Journal Article
Preclinical evaluation of the novel, orally bioavailable Selective Inhibitor of Nuclear Export (SINE) KPT-335 in spontaneous canine cancer: results of a phase I study
London, Cheryl A, Bernabe, Luis Feo, Barnard, Sandra, Kisseberth, William C, Borgatti, Antonella, Henson, Mike, Wilson, Heather, Jensen, Kiersten, Ito, Daisuke, Modiano, Jaime F, Bear, Misty D, Pennell, Michael L, Saint-Martin, Jean-Richard, McCauley, Dilara, Kauffman, Michael, Shacham, Sharon
Published in PloS one (04.02.2014)
Published in PloS one (04.02.2014)
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Sequential loss of tumor vessel pericytes and endothelial cells after inhibition of platelet-derived growth factor B by selective aptamer AX102
SENNINO, Barbara, FALCON, Beverly L, MCCAULEY, Dilara, LE, Tom, MCCAULEY, Thomas, KURZ, Jeffrey C, HASKELL, Amy, EPSTEIN, David M, MCDONALD, Donald M
Published in Cancer research (Chicago, Ill.) (01.08.2007)
Published in Cancer research (Chicago, Ill.) (01.08.2007)
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Selective inhibitors of nuclear export for the treatment of non-Hodgkin’s lymphomas
Azmi, A. S., Al-Katib, A., Aboukameel, A., McCauley, D., Kauffman, M., Shacham, S., Mohammad, R. M.
Published in Haematologica (Roma) (01.07.2013)
Published in Haematologica (Roma) (01.07.2013)
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Benzofuran Derivatives as Potent, Orally Active S1P1 Receptor Agonists: A Preclinical Lead Molecule for MS
Saha, Ashis K, Yu, Xiang, Lin, Jian, Lobera, Mercedes, Sharadendu, Anurag, Chereku, Srinivas, Schutz, Nili, Segal, Dalia, Marantz, Yael, McCauley, Dilara, Middleton, Scot, Siu, Jerry, Bürli, Roland W, Buys, Janet, Horner, Michelle, Salyers, Kevin, Schrag, Michael, Vargas, Hugo M, Xu, Yang, McElvain, Michele, Xu, Han
Published in ACS medicinal chemistry letters (10.02.2011)
Published in ACS medicinal chemistry letters (10.02.2011)
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Journal Article
First-in-Class, First-in-Human Phase I Study of Selinexor, a Selective Inhibitor of Nuclear Export, in Patients With Advanced Solid Tumors
Abdul Razak, Albiruni R, Mau-Soerensen, Morten, Gabrail, Nashat Y, Gerecitano, John F, Shields, Anthony F, Unger, Thaddeus J, Saint-Martin, Jean R, Carlson, Robert, Landesman, Yosef, McCauley, Dilara, Rashal, Tami, Lassen, Ulrik, Kim, Richard, Stayner, Lee-Anne, Mirza, Mansoor R, Kauffman, Michael, Shacham, Sharon, Mahipal, Amit
Published in Journal of clinical oncology (01.12.2016)
Published in Journal of clinical oncology (01.12.2016)
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Journal Article
Selective inhibitors of nuclear export show that CRM1/XPO1 is a target in chronic lymphocytic leukemia
Lapalombella, Rosa, Sun, Qingxiang, Williams, Katie, Tangeman, Larissa, Jha, Shruti, Zhong, Yiming, Goettl, Virginia, Mahoney, Emilia, Berglund, Caroline, Gupta, Sneha, Farmer, Alicia, Mani, Rajeswaran, Johnson, Amy J., Lucas, David, Mo, Xiaokui, Daelemans, Dirk, Sandanayaka, Vincent, Shechter, Sharon, McCauley, Dilara, Shacham, Sharon, Kauffman, Michael, Chook, Yuh Min, Byrd, John C.
Published in Blood (29.11.2012)
Published in Blood (29.11.2012)
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HYDRAZIDE CONTAINING NUCLEAR TRANSPORT MODULATORS AND USES THEREOF
SHACHAM SHARON, MCCAULEY DILARA, SHECHTER SHARON, SANDANAYAKA VINCENT P
Year of Publication 08.05.2024
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Year of Publication 08.05.2024
Patent
Verdinexor, a novel selective inhibitor of nuclear export, reduces influenza a virus replication in vitro and in vivo
Perwitasari, Olivia, Johnson, Scott, Yan, Xiuzhen, Howerth, Elizabeth, Shacham, Sharon, Landesman, Yosef, Baloglu, Erkan, McCauley, Dilara, Tamir, Sharon, Tompkins, S Mark, Tripp, Ralph A
Published in Journal of virology (01.09.2014)
Published in Journal of virology (01.09.2014)
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Journal Article
KPT‐330 inhibitor of CRM1 (XPO1)‐mediated nuclear export has selective anti‐leukaemic activity in preclinical models of T‐cell acute lymphoblastic leukaemia and acute myeloid leukaemia
Etchin, Julia, Sanda, Takaomi, Mansour, Marc R., Kentsis, Alex, Montero, Joan, Le, Bonnie T., Christie, Amanda L., McCauley, Dilara, Rodig, Scott J., Kauffman, Michael, Shacham, Sharon, Stone, Richard, Letai, Anthony, Kung, Andrew L., Thomas Look, A.
Published in British journal of haematology (01.04.2013)
Published in British journal of haematology (01.04.2013)
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Journal Article
HYDRAZIDE CONTAINING NUCLEAR TRANSPORT MODULATORS AND USES THEREOF
SHACHAM SHARON, MCCAULEY DILARA, SHECHTER SHARON, SANDANAYAKA VINCENT P
Year of Publication 27.03.2023
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Year of Publication 27.03.2023
Patent
Synergistic Myeloma Cell Death via Novel Intracellular Activation of Caspase-10-Dependent Apoptosis by Carfilzomib and Selinexor
Rosebeck, Shaun, Alonge, Mattina M, Kandarpa, Malathi, Mayampurath, Anoop, Volchenboum, Samuel L, Jasielec, Jagoda, Dytfeld, Dominik, Maxwell, Sean P, Kraftson, Stephanie J, McCauley, Dilara, Shacham, Sharon, Kauffman, Michael, Jakubowiak, Andrzej J
Published in Molecular cancer therapeutics (01.01.2016)
Published in Molecular cancer therapeutics (01.01.2016)
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Journal Article
HYDRAZIDE CONTAINING NUCLEAR TRANSPORT MODULATORS AND USES THEREOF
SHACHAM SHARON, MCCAULEY DILARA, SHECHTER SHARON, SANDANAYAKA VINCENT P
Year of Publication 06.07.2021
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Year of Publication 06.07.2021
Patent
Preclinical antitumor efficacy of selective exportin 1 inhibitors in glioblastoma
Green, Adam L, Ramkissoon, Shakti H, McCauley, Dilara, Jones, Kristen, Perry, Jennifer A, Hsu, Jessie Hao-Ru, Ramkissoon, Lori A, Maire, Cecile L, Hubbell-Engler, Benjamin, Knoff, David S, Shacham, Sharon, Ligon, Keith L, Kung, Andrew L
Published in Neuro-oncology (Charlottesville, Va.) (01.05.2015)
Published in Neuro-oncology (Charlottesville, Va.) (01.05.2015)
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Journal Article
HYDRAZIDE CONTAINING NUCLEAR TRANSPORT MODULATORS AND USES THEREOF
SHACHAM SHARON, MCCAULEY DILARA, SHECHTER SHARON, SANDANAYAKA VINCENT P
Year of Publication 22.07.2020
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Year of Publication 22.07.2020
Patent
Anti-Myeloma Activity of Combined Inhibition of the Proteasome with Carfilzomib (CFZ) and XPO1/CRM1-Dependent Nuclear Export By Selinexor (KPT-330) Via a Novel Mechanism of Intracellular Activation of Caspase 10-Dependent Apoptosis
Rosebeck, Shaun, Alonge, Mattina, Jasielec, Jagoda, McCauley, Dilara, Shacham, Sharon, Kauffman, Michael, Jakubowiak, Andrzej
Published in Blood (06.12.2014)
Published in Blood (06.12.2014)
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