QUINOXALINES AND AZA-QUINOXALINES AS CRTH2 RECEPTOR MODULATORS
QIN JUN, MAZZOLA ROBERT D. JR, LEYHANE ANDREW J, XIAO DONG, BOYCE CHRISTOPHER W, WU JIE, SILIPHAIVANH PHIENG, YU YOUNONG, ZHANG HONGJUN, MCCORMICK KEVIN D, HUANG XIANHAI, BIJU PURAKKATTLE JOHNY, METHOT JOEY LEE, RAO ASHWIN UMESH, JIANG QIN, DEGRADO SYLVIA JOANNA, GAUUAN JOLICIA POLIVINA, KELLEY ELIZABETH HELEN, PALANI ANANDAN, DONG LI, ASLANIAN ROBERT GEORGE, BROWN WILLIAM COLBY, FEVRIER SALEM, VACCARO HENRY M, CHEN XIAO, DHONDI PAWAN K
Year of Publication 06.12.2013
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Year of Publication 06.12.2013
Patent
Discovery of novel hydroxamates as highly potent tumor necrosis factor-α converting enzyme inhibitors. Part II: Optimization of the S3′ pocket
Mazzola, Robert D., Zhu, Zhaoning, Sinning, Lisa, McKittrick, Brian, Lavey, Brian, Spitler, James, Kozlowski, Joseph, Neng-Yang, Shih, Zhou, Guowei, Guo, Zhuyan, Orth, Peter, Madison, Vincent, Sun, Jing, Lundell, Daniel, Niu, Xiaoda
Published in Bioorganic & medicinal chemistry (01.11.2008)
Published in Bioorganic & medicinal chemistry (01.11.2008)
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Journal Article
Discovery of novel hydroxamates as highly potent tumor necrosis factor-[alpha] converting enzyme inhibitors. Part II: Optimization of the S3′ pocket
Mazzola Jr., Robert D., Zhu, Zhaoning, Sinning, Lisa, McKittrick, Brian, Lavey, Brian, Spitler, James, Kozlowski, Joseph, Neng-Yang, Shih, Zhou, Guowei, Guo, Zhuyan, Orth, Peter, Madison, Vincent, Sun, Jing, Lundell, Daniel, Niu, Xiaoda
Published in Bioorganic & medicinal chemistry letters (01.10.2010)
Published in Bioorganic & medicinal chemistry letters (01.10.2010)
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Journal Article
Discovery of new SCH 39166 analogs as potent and selective dopamine D1 receptor antagonists
Qiang, Li, Sasikumar, T K, Burnett, Duane A, Su, Jing, Tang, Haiqun, Ye, Yuanzan, Mazzola, Jr, Robert D, Zhu, Zhaoning, McKittrick, Brian A, Greenlee, William J, Fawzi, Ahmad, Smith, Michelle, Zhang, Hongtao, Lachowicz, Jean E
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Journal Article
Stereoselective Nazarov Cyclizations of Bridged Bicyclic Dienones
Mazzola, Robert D, White, Timothy D, Vollmer-Snarr, Heidi R, West, F. G
Published in Organic letters (23.06.2005)
Published in Organic letters (23.06.2005)
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Journal Article
Azabicyclo[4.1.0]heptane allosteric modulators of the M4 muscarinic acetylcholine receptor
Clausen, Dane James, Liu, Ping, Fells, James I, Mazzola, Jr., Robert D, Kozlowski, Joseph A
Year of Publication 16.03.2021
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Year of Publication 16.03.2021
Patent
3-(1H-PYRAZOL-4-YL)PYRIDINE ALLOSTERIC MODULATORS OF THE M4 MUSCARINIC ACETYLCHOLINE RECEPTOR
TONG, Ling, MULHEARN, James, SELYUTIN, Oleg, B, RADA, Vanessa, L, ZHANG, Fengqi, ACTON, John, J., III, EGBERTSON, Melissa, SCHUBERT, Jeffrey, W, TELLERS, David, M, BAO, Jianming, LO, Michael Man-Chu, LI, Chunsing, HENDERSON, Timothy, J, HARRISON, Scott, T, GAO, Xiaolei, MAZZOLA, Robert, D., Jr, MENG, Zhaoyang
Year of Publication 28.08.2024
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Year of Publication 28.08.2024
Patent
3-(1H-pyrazol-4-yl)pyridine allosteric modulators of the M4 muscarinic acetylcholine receptor
Zhang, Fengqi, Gao, Xiaolei, Selyutin, Oleg B, Bao, Jianming, Schubert, Jeffrey W, Egbertson, Melissa, Henderson, Timothy J, Lo, Michael Man-Chu, Tellers, David M, Li, Chunsing, Acton, III, John J, Harrison, Scott T, Rada, Vanessa L, Mazzola, Jr., Robert D, Tong, Ling, Meng, Zhaoyang, Mulhearn, James
Year of Publication 30.04.2024
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Year of Publication 30.04.2024
Patent
3-(1H-PYRAZOL-4-YL)PYRIDINE ALLOSTERIC MODULATORS OF THE M4 MUSCARINIC ACETYLCHOLINE RECEPTOR
SUZUKI, Takao, HARRISON, Scott Timothy, SELYUTIN, Oleg, B, FERGUSON, Ronald, III, ZHANG, Fengqi, ACTON, John, J., III, EGBERTSON, Melissa, BAO, Jianming, LO, Michael Man-Chu, HENDERSON, Timothy, J, NA, Meng, KNOWLES, Sandra, L, GAO, Xiaolei, MAZZOLA, Robert, D., Jr, DENG, Qiaolin
Year of Publication 02.08.2023
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Year of Publication 02.08.2023
Patent
3-(1H-PYRAZOL-4-YL)PYRIDINE ALLOSTERIC MODULATORS OF THE M4 MUSCARINIC ACETYLCHOLINE RECEPTOR
TONG, Ling, HARRISON, Scott Timothy, MAZZOLA, Robert D., Jr, FERGUSON, Ronald, III, ZHANG, Fengqi, ACTON, John, J., III, EGBERTSON, Melissa, BAO, Jianming, LO, Michael Man-Chu, KNOWLES, Sandra L, LI, Chunsing, TELLERS, David M, RUDD, Michael T, NA, Meng, SELYUTIN, Oleg B, GAO, Xiaolei, DENG, Qiaolin, MENG, Zhaoyang
Year of Publication 29.03.2023
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Year of Publication 29.03.2023
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