Structure-Based Design and Synthesis of Potent Cyclic Peptides Inhibiting the YAP–TEAD Protein–Protein Interaction
Zhang, Zhisen, Lin, Zhaohu, Zhou, Zheng, Shen, Hong C, Yan, S. Frank, Mayweg, Alexander V, Xu, Zhiheng, Qin, Ning, Wong, Jason C, Zhang, Zhenshan, Rong, Yiping, Fry, David C, Hu, Taishan
Published in ACS medicinal chemistry letters (11.09.2014)
Published in ACS medicinal chemistry letters (11.09.2014)
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Design and Synthesis of Orally Bioavailable 4‑Methyl Heteroaryldihydropyrimidine Based Hepatitis B Virus (HBV) Capsid Inhibitors
Qiu, Zongxing, Lin, Xianfeng, Zhou, Mingwei, Liu, Yongfu, Zhu, Wei, Chen, Wenming, Zhang, Weixing, Guo, Lei, Liu, Haixia, Wu, Guolong, Huang, Mengwei, Jiang, Min, Xu, Zhiheng, Zhou, Zheng, Qin, Ning, Ren, Shuang, Qiu, Hongxia, Zhong, Sheng, Zhang, Yuxia, Zhang, Yi, Wu, Xiaoyue, Shi, Liping, Shen, Fang, Mao, Yi, Zhou, Xue, Yang, Wengang, Wu, Jim Z, Yang, Guang, Mayweg, Alexander V, Shen, Hong C, Tang, Guozhi
Published in Journal of medicinal chemistry (25.08.2016)
Published in Journal of medicinal chemistry (25.08.2016)
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Discovery of 3‑Pyridyl Isoindolin-1-one Derivatives as Potent, Selective, and Orally Active Aldosterone Synthase (CYP11B2) Inhibitors
Liu, Yongfu, Wu, Jun, Zhou, Mingwei, Chen, Wenming, Li, Dongbo, Wang, Zhanguo, Hornsperger, Benoit, Aebi, Johannes D, Märki, Hans-Peter, Kuhn, Bernd, Wang, Lisha, Kuglstatter, Andreas, Benz, Jörg, Müller, Stephan, Hochstrasser, Remo, Ottaviani, Giorgio, Xin, Jian, Kirchner, Stephan, Mohr, Susanne, Verry, Philippe, Riboulet, William, Shen, Hong C, Mayweg, Alexander V, Amrein, Kurt, Tan, Xuefei
Published in Journal of medicinal chemistry (09.07.2020)
Published in Journal of medicinal chemistry (09.07.2020)
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Journal Article
Discovery of 4‑Aryl-5,6,7,8-tetrahydroisoquinolines as Potent, Selective, and Orally Active Aldosterone Synthase (CYP11B2) Inhibitors: In Vivo Evaluation in Rodents and Cynomolgus Monkeys
Martin, Rainer E, Aebi, Johannes D, Hornsperger, Benoit, Krebs, Hans-Jakob, Kuhn, Bernd, Kuglstatter, Andreas, Alker, André M, Märki, Hans Peter, Müller, Stephan, Burger, Dominique, Ottaviani, Giorgio, Riboulet, William, Verry, Philippe, Tan, Xuefei, Amrein, Kurt, Mayweg, Alexander V
Published in Journal of medicinal chemistry (22.10.2015)
Published in Journal of medicinal chemistry (22.10.2015)
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Synthesis of annulated pyridines as inhibitors of aldosterone synthase (CYP11B2)
Martin, Rainer E., Lehmann, Johannes, Alzieu, Thibaut, Lenz, Mario, Corrales, Marjorie A. Carnero, Aebi, Johannes D., Marki, Hans Peter, Kuhn, Bernd, Amrein, Kurt, Mayweg, Alexander V., Britton, Robert
Published in Organic & biomolecular chemistry (01.01.2016)
Published in Organic & biomolecular chemistry (01.01.2016)
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Journal Article
Challenges and Rewards in Medicinal Chemistry Targeting Cardiovascular and Metabolic Diseases
Neidhart, Werner, Ackermann, Jean, Amrein, Kurt, Conte, Aurelia, Hunziker, Daniel, Kuhn, Bernd, Märki, Hans Peter, Nettekoven, Matthias, Ruf, Armin, Schulz-Gasch, Tanja, Mayweg, Alexander V
Published in Chimia (01.01.2015)
Published in Chimia (01.01.2015)
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Journal Article
Discovery of RG7834: The First-in-Class Selective and Orally Available Small Molecule Hepatitis B Virus Expression Inhibitor with Novel Mechanism of Action
Han, Xingchun, Zhou, Chengang, Jiang, Min, Wang, Yongguang, Wang, Jianhua, Cheng, Zhanling, Wang, Min, Liu, Yongqiang, Liang, Chungen, Wang, Jianping, Wang, Zhanguo, Weikert, Robert, Lv, Wenzhe, Xie, Jianxun, Yu, Xin, Zhou, Xue, Luangsay, Souphalone, Shen, Hong C, Mayweg, Alexander V, Javanbakht, Hassan, Yang, Song
Published in Journal of medicinal chemistry (13.12.2018)
Published in Journal of medicinal chemistry (13.12.2018)
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Journal Article
Discovery of Linvencorvir (RG7907), a Hepatitis B Virus Core Protein Allosteric Modulator, for the Treatment of Chronic HBV Infection
Zhang, Weixing, Guo, Lei, Liu, Haixia, Wu, Guolong, Shi, Houguang, Zhou, Mingwei, Zhang, Zhisen, Kou, Buyu, Hu, Taishan, Zhou, Zheng, Xu, Zhiheng, Zhou, Xue, Zhou, Yuan, Tian, Xiaojun, Yang, Guang, Young, John A. T., Qiu, Hongxia, Ottaviani, Giorgio, Xie, Jianxun, Mayweg, Alexander V., Shen, Hong C., Zhu, Wei
Published in Journal of medicinal chemistry (23.03.2023)
Published in Journal of medicinal chemistry (23.03.2023)
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Journal Article
β‑Secretase (BACE1) Inhibitors with High in Vivo Efficacy Suitable for Clinical Evaluation in Alzheimer’s Disease
Hilpert, Hans, Guba, Wolfgang, Woltering, Thomas J, Wostl, Wolfgang, Pinard, Emmanuel, Mauser, Harald, Mayweg, Alexander V, Rogers-Evans, Mark, Humm, Roland, Krummenacher, Daniela, Muser, Thorsten, Schnider, Christian, Jacobsen, Helmut, Ozmen, Laurence, Bergadano, Alessandra, Banner, David W, Hochstrasser, Remo, Kuglstatter, Andreas, David-Pierson, Pascale, Fischer, Holger, Polara, Alessandra, Narquizian, Robert
Published in Journal of medicinal chemistry (23.05.2013)
Published in Journal of medicinal chemistry (23.05.2013)
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Journal Article
Discovery of potent and selective CDK8 inhibitors through FBDD approach
Han, Xingchun, Jiang, Min, Zhou, Chengang, Zhou, Zheng, Xu, Zhiheng, Wang, Lisha, Mayweg, Alexander V., Niu, Rui, Jin, Tai-Guang, Yang, Song
Published in Bioorganic & medicinal chemistry letters (15.09.2017)
Published in Bioorganic & medicinal chemistry letters (15.09.2017)
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Journal Article
Discovery and Pre-Clinical Characterization of Third-Generation 4‑H Heteroaryldihydropyrimidine (HAP) Analogues as Hepatitis B Virus (HBV) Capsid Inhibitors
Qiu, Zongxing, Lin, Xianfeng, Zhang, Weixing, Zhou, Mingwei, Guo, Lei, Kocer, Buelent, Wu, Guolong, Zhang, Zhisen, Liu, Haixia, Shi, Houguang, Kou, Buyu, Hu, Taishan, Hu, Yimin, Huang, Mengwei, Yan, S. Frank, Xu, Zhiheng, Zhou, Zheng, Qin, Ning, Wang, Yue Fen, Ren, Shuang, Qiu, Hongxia, Zhang, Yuxia, Zhang, Yi, Wu, Xiaoyue, Sun, Kai, Zhong, Sheng, Xie, Jianxun, Ottaviani, Giorgio, Zhou, Yuan, Zhu, Lina, Tian, Xiaojun, Shi, Liping, Shen, Fang, Mao, Yi, Zhou, Xue, Gao, Lu, Young, John A. T, Wu, Jim Zhen, Yang, Guang, Mayweg, Alexander V, Shen, Hong C, Tang, Guozhi, Zhu, Wei
Published in Journal of medicinal chemistry (27.04.2017)
Published in Journal of medicinal chemistry (27.04.2017)
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Journal Article
A Concise, Selective Synthesis of the Polyketide Spacer Domain of a Potent Bryostatin Analogue
Wender, Paul A, Mayweg, Alexander V. W, VanDeusen, Christopher L
Published in Organic letters (06.02.2003)
Published in Organic letters (06.02.2003)
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Journal Article
Studies towards the synthesis of lindenene: Unexpected stereochemical outcome of an intramolecular cyclopropanation reaction and synthesis of (+/-)-epi-Lindenene and (+/-)-iso-Lindenene
Fenlon, Thomas W., Schwaebisch, Dirk, Mayweg, Alexander V. W., Lee, Victor, Adlington, Robert M., Baldwin, Jack E.
Published in Synlett (16.10.2007)
Published in Synlett (16.10.2007)
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Journal Article
Benzodioxoles: Novel Cannabinoid-1 Receptor Inverse Agonists for the Treatment of Obesity
Alig, Leo, Alsenz, Jochem, Andjelkovic, Mirjana, Bendels, Stefanie, Bénardeau, Agnès, Bleicher, Konrad, Bourson, Anne, David-Pierson, Pascale, Guba, Wolfgang, Hildbrand, Stefan, Kube, Dagmar, Lübbers, Thomas, Mayweg, Alexander V, Narquizian, Robert, Neidhart, Werner, Nettekoven, Matthias, Plancher, Jean-Marc, Rocha, Cynthia, Rogers-Evans, Mark, Röver, Stephan, Schneider, Gisbert, Taylor, Sven, Waldmeier, Pius
Published in Journal of medicinal chemistry (10.04.2008)
Published in Journal of medicinal chemistry (10.04.2008)
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Journal Article
Transannular, decarboxylative Claisen rearrangement reactions for the synthesis of sulfur-substituted vinylcyclopropanes
Craig, Donald, Gore, Sophie J., Lansdell, Mark I., Lewis, Simon E., Mayweg, Alexander V. W., White, Andrew J. P.
Published in Chemical communications (Cambridge, England) (01.01.2010)
Published in Chemical communications (Cambridge, England) (01.01.2010)
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Journal Article
NEW DIHYDROQUINOLINE-2-ONE DERIVATIVES AS ALDOSTERONE SYNTHASE(CYP1 1 B2 OR CYP1 1 B1) INHIBITORS
AMREIN KURT, MAYWEG ALEXANDER V, KUHN BERND, TAN XUEFEI, AEBI JOHANNES, MAERKI HANS P, HORNSPERGER BENOIT
Year of Publication 11.11.2015
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Year of Publication 11.11.2015
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