Synthesis and in vitro evaluation of novel highly potent coumarin inhibitors of gyrase B
Laurin, Patrick, Ferroud, Didier, Klich, Michel, Dupuis-Hamelin, Claudine, Mauvais, Pascale, Lassaigne, Patrice, Bonnefoy, Alain, Musicki, Branislav
Published in Bioorganic & medicinal chemistry letters (19.07.1999)
Published in Bioorganic & medicinal chemistry letters (19.07.1999)
Get full text
Journal Article
Activation of α- and β-estrogen receptors by persistent pesticides in reporter cell lines
Lemaire, Géraldine, Mnif, Wissem, Mauvais, Pascale, Balaguer, Patrick, Rahmani, Roger
Published in Life sciences (1973) (15.08.2006)
Published in Life sciences (1973) (15.08.2006)
Get full text
Journal Article
Pyrazine Arotinoids with Inverse Agonist Activities on the Retinoid and Rexinoid Receptors
García, José, Khanwalkar, Harshal, Pereira, Raquel, Erb, Cathie, Voegel, Johannes J, Collette, Pascal, Mauvais, Pascale, Bourguet, William, Gronemeyer, Hinrich, de Lera, Ángel R
Published in Chembiochem : a European journal of chemical biology (04.05.2009)
Published in Chembiochem : a European journal of chemical biology (04.05.2009)
Get full text
Journal Article
Highly Potent Naphthofuran‐Based Retinoic Acid Receptor Agonists
Santín, Efrén Pérez, Khanwalkar, Harshal, Voegel, Johannes, Collette, Pascal, Mauvais, Pascale, Gronemeyer, Hinrich, de Lera, Ángel R.
Published in ChemMedChem (01.05.2009)
Published in ChemMedChem (01.05.2009)
Get full text
Journal Article
PHENOL DERIVATIVES AND PHARMACEUTICAL OR COSMETIC USE THEREOF
RETHORE SANDRINE, COLLETTE PASCAL, MAUVAIS PASCALE, POINSARD CEDRIC, LINGET JEAN MICHEL
Year of Publication 07.09.2012
Get full text
Year of Publication 07.09.2012
Patent
PHENOL DERIVATIVES AND THE PHARMACEUTICAL OR COSMETIC USE THEREOF
RETHORE SANDRINE, COLLETTE PASCAL, MAUVAIS PASCALE, POINSARD CEDRIC, LINGET JEAN MICHEL
Year of Publication 29.08.2012
Get full text
Year of Publication 29.08.2012
Patent
PHENOL DERIVATIVES AND PHARMACEUTICAL OR COSMETIC USE THEREOF
RETHORE SANDRINE, COLLETTE PASCAL, MAUVAIS PASCALE, POINSARD CEDRIC, LINGET JEAN MICHEL
Year of Publication 29.08.2012
Get full text
Year of Publication 29.08.2012
Patent
Structure-activity relationship in two series of aminoalkyl substituted coumarin inhibitors of gyrase B
Laurin, Patrick, Ferroud, Didier, Schio, Laurent, Klich, Michael, Dupuis-Hamelin, Claudine, Mauvais, Pascale, Lassaigne, Patrice, Bonnefoy, Alain, Musicki, Branislav
Published in Bioorganic & medicinal chemistry letters (04.10.1999)
Published in Bioorganic & medicinal chemistry letters (04.10.1999)
Get full text
Journal Article
Synthesis and biological evaluation of coumarincarboxylic acids as inhibitors of gyrase B. L-rhamnose as an effective substitute for L-noviose
Ferroud, Didier, Collard, Jeannine, Klich, Michel, Dupuis-Hamelin, Claudine, Mauvais, Pascale, Lassaigne, Patrice, Bonnefoy, Alain, Musicki, Branislav
Published in Bioorganic & medicinal chemistry letters (04.10.1999)
Published in Bioorganic & medicinal chemistry letters (04.10.1999)
Get full text
Journal Article
Antibiotic Resistance Peptides: Interaction of Peptides Conferring Macrolide and Ketolide Resistance with Staphylococcus aureus Ribosomes. Conformation of Bound Peptides As Determined by Transferred NOE Experiments
Verdier, Laurent, Gharbi-Benarous, Josyane, Bertho, Gildas, Mauvais, Pascale, Girault, Jean-Pierre
Published in Biochemistry (Easton) (02.04.2002)
Published in Biochemistry (Easton) (02.04.2002)
Get full text
Journal Article
Fine Tuning of physico-chemical parameters to optimise a new series of novobiocin analogues
Schio, Laurent, Chatreaux, Fabienne, Loyau, Véronique, Murer, Michel, Ferreira, Anne, Mauvais, Pascale, Bonnefoy, Alain, Klich, Michel
Published in Bioorganic & medicinal chemistry letters (04.06.2001)
Published in Bioorganic & medicinal chemistry letters (04.06.2001)
Get full text
Journal Article
Synthesis of isothiochroman 2,2-dioxide and 1,2-benzooxathiin 2,2-dioxide gyrase B inhibitors
Peixoto, Christophe, Laurin, Patrick, Klich, Michel, Dupuis-Hamelin, Claudine, Mauvais, Pascale, Lassaigne, Patrice, Bonnefoy, Alain, Musicki, Branislav
Published in Tetrahedron letters (11.03.2000)
Published in Tetrahedron letters (11.03.2000)
Get full text
Journal Article
Coumarin inhibitors of gyrase B with N-propargyloxy-carbamate as an effective pyrrole bioisostere
PERIERS, A.-M, LAURIN, P, FERROUD, D, HAESSLEIN, J.-L, KLICH, M, DUPUIS-HAMELIN, C, MAUVAIS, P, LASSAIGNE, P, BONNEFOY, A, MUSICKI, B
Published in Bioorganic & medicinal chemistry letters (17.01.2000)
Published in Bioorganic & medicinal chemistry letters (17.01.2000)
Get full text
Journal Article
Phenol derivatives and the pharmaceutical or cosmetic use thereof
Linget, Jean-Michel, Collette, Pascal, Poinsard, Cedric, Rethore, Sandrine, Mauvais, Pascale
Year of Publication 12.02.2019
Get full text
Year of Publication 12.02.2019
Patent