Adsorbent Screening for Metal Impurity Removal in Pharmaceutical Process Research
Welch, Christopher J, Albaneze-Walker, Jennifer, Leonard, William R, Biba, Mirlinda, DaSilva, Jimmy, Henderson, Derek, Laing, Brian, Mathre, David J, Spencer, Sandra, Bu, Xiaodong, Wang, Tiebang
Published in Organic process research & development (01.03.2005)
Published in Organic process research & development (01.03.2005)
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Development of a pharmaceutical cocrystal of a monophosphate salt with phosphoric acid
Chen, Alex M, Ellison, Martha E, Peresypkin, Andrey, Wenslow, Robert M, Variankaval, Narayan, Savarin, Cecile G, Natishan, Theresa K, Mathre, David J, Dormer, Peter G, Euler, Danielle H, Ball, Richard G, Ye, Zhixiong, Wang, Yaling, Santos, Ivan
Published in Chemical communications (Cambridge, England) (01.01.2007)
Published in Chemical communications (Cambridge, England) (01.01.2007)
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Journal Article
Efficient Synthesis of NK1 Receptor Antagonist Aprepitant Using a Crystallization-Induced Diastereoselective Transformation
Brands, Karel M. J, Payack, Joseph F, Rosen, Jonathan D, Nelson, Todd D, Candelario, Alexander, Huffman, Mark A, Zhao, Matthew M, Li, Jing, Craig, Bridgette, Song, Zhiguo J, Tschaen, David M, Hansen, Karl, Devine, Paul N, Pye, Philip J, Rossen, Kai, Dormer, Peter G, Reamer, Robert A, Welch, Christopher J, Mathre, David J, Tsou, Nancy N, McNamara, James M, Reider, Paul J
Published in Journal of the American Chemical Society (26.02.2003)
Published in Journal of the American Chemical Society (26.02.2003)
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Lipid nanoparticle purification by Spin Centrifugation–Dialysis (SCD): A facile and high-throughput approach for small scale preparation of siRNA–lipid complexes
Mihaila, Radu, Chang, Silvia, Wei, Alan T., Hu, Zhi Y., Ruhela, Dipali, Shadel, Timothy R., Duenwald, Sven, Payson, Elmer, Cunningham, James J., Kuklin, Nelly, Mathre, David J.
Published in International journal of pharmaceutics (25.11.2011)
Published in International journal of pharmaceutics (25.11.2011)
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Journal Article
Nucleophilic Displacement at Benzhydryl Centers: Asymmetric Synthesis of 1,1-Diarylalkyl Derivatives
Bolshan, Yuri, Chen, Cheng-yi, Chilenski, Jennifer R, Gosselin, Francis, Mathre, David J, O'Shea, Paul D, Roy, Amélie, Tillyer, Richard D
Published in Organic letters (08.01.2004)
Published in Organic letters (08.01.2004)
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Highly Diastereoselective Heterogeneously Catalyzed Hydrogenation of Enamines for the Synthesis of Chiral β-Amino Acid Derivatives
Ikemoto, Norihiro, Tellers, David M, Dreher, Spencer D, Liu, Jinchu, Huang, Angie, Rivera, Nelo R, Njolito, Eugenia, Hsiao, Yi, McWilliams, J. Christopher, Williams, J. Michael, Armstrong, Joseph D, Sun, Yongkui, Mathre, David J, Grabowski, Edward J. J, Tillyer, Richard D
Published in Journal of the American Chemical Society (17.03.2004)
Published in Journal of the American Chemical Society (17.03.2004)
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Mechanistic Studies of the Molybdenum-Catalyzed Asymmetric Alkylation Reaction
Hughes, David L., Lloyd-Jones, Guy C., Krska, Shane W., Gouriou, Laure, Bonnet, Veronique D., Jack, Kevin, Sun, Yongkui, Mathre, David J., Reamer, Robert A., Trost, Barry M.
Published in Proceedings of the National Academy of Sciences - PNAS (13.04.2004)
Published in Proceedings of the National Academy of Sciences - PNAS (13.04.2004)
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Direct conversion of activated alcohols to azides using diphenyl phosphorazidate. A practical alternative to Mitsunobu conditions
Thompson, Andrew S, Humphrey, Guy R, DeMarco, Anthony M, Mathre, David J, Grabowski, Edward J. J
Published in Journal of organic chemistry (01.10.1993)
Published in Journal of organic chemistry (01.10.1993)
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Journal Article
An Efficient Asymmetric Synthesis of an Estrogen Receptor Modulator by Sulfoxide-Directed Borane Reduction
Song, Zhiguo J., King, Anthony O., Waters, Marjorie S., Lang, Fengrui, Zewge, Daniel, Bio, Matthew, Leazer, Johnnie L., Javadi, Gary, Kassim, Amude, Tschaen, David M., Reamer, Robert A., Rosner, Thorsten, Chilenski, Jennifer R., Mathre, David J., Volante, R. P., Tillyer, Richard, Trost, Barry M.
Published in Proceedings of the National Academy of Sciences - PNAS (20.04.2004)
Published in Proceedings of the National Academy of Sciences - PNAS (20.04.2004)
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Chromatography as an Enabling Technology in Pharmaceutical Process Development: Expedited Multikilogram Preparation of a Candidate HIV Protease Inhibitor
Welch, Christopher J, Fleitz, Fred, Antia, Firoz, Yehl, Pete, Waters, Robert, Ikemoto, Norihiro, Armstrong, Joseph D, Mathre, David J
Published in Organic process research & development (01.03.2004)
Published in Organic process research & development (01.03.2004)
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A practical process for the preparation of tetrahydro-1-methyl-3,3-diphenyl-1H,3H-pyrrolo[1,2-c][1,3,2]oxazaborole-borane. A highly enantioselective stoichiometric and catalytic reducing agent
Mathre, David J, Thompson, Andrew S, Douglas, Alan W, Hoogsteen, Karst, Carroll, James D, Corley, Edward G, Grabowski, Edward J. J
Published in Journal of organic chemistry (01.05.1993)
Published in Journal of organic chemistry (01.05.1993)
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Journal Article
Crystal structure and surface properties of an investigational drug—A case study
Kiang, Y.-H., Shi, H.Galen, Mathre, David J., Xu, Wei, Zhang, Dina, Panmai, Santipharp
Published in International journal of pharmaceutics (06.08.2004)
Published in International journal of pharmaceutics (06.08.2004)
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Journal Article
Studies on the racemization of a stereolabile 5-aryl-thiazolidinedione
Welch, Christopher J., Kress, Michael H., Beconi, Maria, Mathre, David J.
Published in Chirality (New York, N.Y.) (2003)
Published in Chirality (New York, N.Y.) (2003)
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Journal Article
Scalable, efficient process for the synthesis of ( R)-3,5-bistrifluoromethylphenyl ethanol via catalytic asymmetric transfer hydrogenation and isolation as a DABCO inclusion complex
Hansen, Karl B., Chilenski, Jennifer R., Desmond, Richard, Devine, Paul N., Grabowski, Edward J.J., Heid, Richard, Kubryk, Michele, Mathre, David J., Varsolona, Richard
Published in Tetrahedron: asymmetry (14.11.2003)
Published in Tetrahedron: asymmetry (14.11.2003)
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Journal Article
Microplate evaluation of process adsorbents
Welch, Christopher J., Shaimi, Mohamed, Biba, Mirlinda, Chilenski, Jennifer R., Szumigala Jr, Ronald H., Dolling, Ulf, Mathre, David J., Reider, Paul J.
Published in Journal of separation science (01.09.2002)
Published in Journal of separation science (01.09.2002)
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Journal Article
A practical enantioselective synthesis of .alpha.,.alpha.-diaryl-2-pyrrolidinemethanol. Preparation and chemistry of the corresponding oxazaborolidines
Mathre, David J, Jones, Todd K, Xavier, Lyndon C, Blacklock, Thomas J, Reamer, Robert A, Mohan, Julie J, Jones, E. Tracy Turner, Hoogsteen, Karst, Baum, Mary W, Grabowski, E. J. J
Published in Journal of organic chemistry (01.01.1991)
Published in Journal of organic chemistry (01.01.1991)
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Synthesis of 3-Aminopyrazinone Mediated by 2-Pyridylthioimidate−ZnCl2 Complexes. Development of an Efficient Route to a Thrombin Inhibitor
Chung, John Y. L, Cvetovich, Raymond J, Tsay, Fuh-Rong, Dormer, Peter G, DiMichele, Lisa, Mathre, David J, Chilenski, Jennifer R, Mao, Bing, Wenslow, Robert
Published in Journal of organic chemistry (14.11.2003)
Published in Journal of organic chemistry (14.11.2003)
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