A novel JAK inhibitor, peficitinib, demonstrates potent efficacy in a rat adjuvant-induced arthritis model
Ito, Misato, Yamazaki, Shunji, Yamagami, Kaoru, Kuno, Masako, Morita, Yoshiaki, Okuma, Kenji, Nakamura, Koji, Chida, Noboru, Inami, Masamichi, Inoue, Takayuki, Shirakami, Shohei, Higashi, Yasuyuki
Published in Journal of pharmacological sciences (01.01.2017)
Published in Journal of pharmacological sciences (01.01.2017)
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Regulation of Allergic Airway Inflammation through Toll-Like Receptor 4-Mediated Modification of Mast Cell Function
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Published in Proceedings of the National Academy of Sciences - PNAS (14.02.2006)
Published in Proceedings of the National Academy of Sciences - PNAS (14.02.2006)
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Identification of a Conserved GATA3 Response Element Upstream Proximal from the Interleukin-13 Gene Locus
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Published in The Journal of biological chemistry (01.11.2002)
Published in The Journal of biological chemistry (01.11.2002)
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src homology 2 domain-containing tyrosine phosphatase SHP-1 controls the development of allergic airway inflammation
Kamata, Tohru, Yamashita, Masakatsu, Kimura, Motoko, Murata, Kaoru, Inami, Masamichi, Shimizu, Chiori, Sugaya, Kaoru, Wang, Chrong-Reen, Taniguchi, Masaru, Nakayama, Toshinori
Published in The Journal of clinical investigation (01.01.2003)
Published in The Journal of clinical investigation (01.01.2003)
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src homology 2 domain–containing tyrosine phosphatase SHP-1 controls the development of allergic airway inflammation
Kamata, Tohru, Yamashita, Masakatsu, Kimura, Motoko, Murata, Kaoru, Inami, Masamichi, Shimizu, Chiori, Sugaya, Kaoru, Wang, Chrong-Reen, Taniguchi, Masaru, Nakayama, Toshinori
Published in The Journal of clinical investigation (01.01.2003)
Published in The Journal of clinical investigation (01.01.2003)
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CD28 Costimulation Controls Histone Hyperacetylation of the Interleukin 5 Gene Locus in Developing Th2 Cells
Inami, Masamichi, Yamashita, Masakatsu, Tenda, Yoshiyuki, Hasegawa, Akihiro, Kimura, Motoko, Hashimoto, Kahoko, Seki, Nobuo, Taniguchi, Masaru, Nakayama, Toshinori
Published in The Journal of biological chemistry (28.05.2004)
Published in The Journal of biological chemistry (28.05.2004)
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CD69‐null mice protected from arthritis induced with anti‐type II collagen antibodies
Murata, Kaoru, Inami, Masamichi, Hasegawa, Akihiro, Kubo, Shuichi, Kimura, Motoko, Yamashita, Masakatsu, Hosokawa, Hiroyuki, Nagao, Tomokazu, Suzuki, Kazuo, Hashimoto, Kahoko, Shinkai, Hiroshi, Koseki, Haruhiko, Taniguchi, Masaru, Ziegler, Steven F., Nakayama, Toshinori
Published in International immunology (01.08.2003)
Published in International immunology (01.08.2003)
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CS3B-2-2 ASP015K: A Novel Janus Kinase Inhibitor Demonstrated Potent Efficacy in Adjuvant-Induced Arthritis and Chronic Oxazolone-Induced Dermatitis Model in Rats
Masamichi Inami, Shunji Yamazaki, Misato Ito, Noboru Chida, Tomonori Nakanishi, Shinsuke Ooshima, Kaori Hanaoka, Keiko Ohkubo, Shohei Shirakami, Takayuki Inoue, Yasutomo Fujii, Yasuyuki Higashi
Published in Journal of Pharmacological Sciences (15.03.2013)
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Published in Journal of Pharmacological Sciences (15.03.2013)
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FR177391, a new anti-hyperlipidemic agent from Serratia. II. Pharmacological activity of FR177391
Inami, Masamichi, Kawamura, Ikuo, Tsujimoto, Susumu, Yasuno, Tohru, Lacey, Elizabeth, Hirosumi, Jiro, Takakura, Shoji, Nishigaki, Fusako, Naoe, Yoshinori, Manda, Toshitaka, Mutoh, Seitaro
Published in Journal of antibiotics (01.10.2005)
Published in Journal of antibiotics (01.10.2005)
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Prolonged skin allograft survival by IL-10 gene-introduced CD4 T cell administration
Miyamoto, Takeshi, Kaneko, Takaaki, Yamashita, Masakatsu, Tenda, Yoshiyuki, Inami, Masamichi, Suzuki, Akane, Ishii, Sohtaro, Kimura, Motoko, Hashimoto, Kahoko, Shimada, Hideaki, Yahata, Hiroshi, Ochiai, Takenori, Saito, Izumu, DeGregori, James, Nakayama, Toshinori
Published in International immunology (01.06.2005)
Published in International immunology (01.06.2005)
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FR177391, A New Anti-hyperlipidemic Agent from Serratia
Inami, Masamichi, Kawamura, Ikuo, Tsujimoto, Susumu, Yasuno, Tohru, Lacey, Elizabeth, Hirosumi, Jiro, Takakura, Shoji, Nishigaki, Fusako, Naoe, Yoshinori, Manda, Toshitaka, Mutoh, Seitaro
Published in Journal of antibiotics (01.10.2005)
Published in Journal of antibiotics (01.10.2005)
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AS2553627, a novel JAK inhibitor, prevents chronic rejection in rat cardiac allografts
Nakamura, Koji, Inami, Masamichi, Morio, Hiroki, Okuma, Kenji, Ito, Misato, Noto, Takahisa, Shirakami, Shohei, Hirose, Jun, Morokata, Tatsuaki
Published in European journal of pharmacology (05.02.2017)
Published in European journal of pharmacology (05.02.2017)
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Anti‐cachectic Effect of FK317, a Novel Anti‐cancer Agent, in Colon26 and LX‐1 Models in Mice
Naoe, Yoshinori, Kawamura, Ikuo, Inami, Masamichi, Matsumoto, Sanae, Nishigaki, Fusako, Tsujimoto, Susumu, Manda, Toshitaka, Shimomura, Kyoichi
Published in Cancer science (01.12.1998)
Published in Cancer science (01.12.1998)
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FK317, a Novel Substituted Dihydrobenzoxazine, Exhibits Potent Antitumor Activity against Human Tumor Xenografts in Nude Mice
Naoe, Yoshinori, Inami, Masamichi, Matsumoto, Sanae, Takagaki, Shoji, Fujiwara, Tomoichi, Yamazaki, Sachiko, Kawamura, Ikuo, Nishigaki, Fusako, Tsujimoto, Susumu, Manda, Toshitaka, Shimomura, Kyoichi
Published in Cancer science (01.12.1998)
Published in Cancer science (01.12.1998)
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Replacement of mycophenolate mofetil with a JAK inhibitor, AS2553627, in combination with low-dose tacrolimus, for renal allograft rejection in non-human primates
Nakamura, Koji, Oshima, Shinsuke, Maeda, Masashi, Morio, Hiroki, Fukahori, Hidehiko, Nakanishi, Tomonori, Tsujimoto, Susumu, Hirose, Jun, Noto, Takahisa, Hamakawa, Nozomu, Inami, Masamichi, Morokata, Tatsuaki
Published in International immunopharmacology (01.11.2018)
Published in International immunopharmacology (01.11.2018)
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Discovery of 3,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-2(1H)-one derivatives as novel JAK inhibitors
Yamagishi, Hiroaki, Shirakami, Shohei, Nakajima, Yutaka, Tanaka, Akira, Takahashi, Fumie, Hamaguchi, Hisao, Hatanaka, Keiko, Moritomo, Ayako, Inami, Masamichi, Higashi, Yasuyuki, Inoue, Takayuki
Published in Bioorganic & medicinal chemistry (01.08.2015)
Published in Bioorganic & medicinal chemistry (01.08.2015)
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Design, synthesis, and evaluation of 4,6-diaminonicotinamide derivatives as novel and potent immunomodulators targeting JAK3
Nakajima, Yutaka, Aoyama, Naohiro, Takahashi, Fumie, Sasaki, Hiroshi, Hatanaka, Keiko, Moritomo, Ayako, Inami, Masamichi, Ito, Misato, Nakamura, Koji, Nakamori, Fumihiro, Inoue, Takayuki, Shirakami, Shohei
Published in Bioorganic & medicinal chemistry (01.10.2016)
Published in Bioorganic & medicinal chemistry (01.10.2016)
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Effective suppression of donor specific antibody production by Cathepsin S inhibitors in a mouse transplantation model
Kubo, Kaori, Kawato, Yuka, Nakamura, Koji, Nakajima, Yutaka, Nakagawa, Terry Y., Hanaoka, Kaori, Oshima, Shinsuke, Fukahori, Hidehiko, Inami, Masamichi, Morokata, Tatsuaki, Higashi, Yasuyuki
Published in European journal of pharmacology (05.11.2018)
Published in European journal of pharmacology (05.11.2018)
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Synthesis and evaluation of novel 1H-pyrrolo[2,3-b]pyridine-5-carboxamide derivatives as potent and orally efficacious immunomodulators targeting JAK3
Nakajima, Yutaka, Inoue, Takayuki, Nakai, Kazuo, Mukoyoshi, Koichiro, Hamaguchi, Hisao, Hatanaka, Keiko, Sasaki, Hiroshi, Tanaka, Akira, Takahashi, Fumie, Kunikawa, Shigeki, Usuda, Hiroyuki, Moritomo, Ayako, Higashi, Yasuyuki, Inami, Masamichi, Shirakami, Shohei
Published in Bioorganic & medicinal chemistry (01.08.2015)
Published in Bioorganic & medicinal chemistry (01.08.2015)
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Different Effects of FK317 on Multidrug‐resistant Tumor in vivo and in vitro
Naoe, Yoshinori, Inami, Masamichi, Takagaki, Shoji, Matsumoto, Sanae, Kawamura, Ikuo, Nishigaki, Fusako, Tsujimoto, Susumu, Manda, Toshitaka, Shimomura, Kyoichi
Published in Cancer science (01.10.1998)
Published in Cancer science (01.10.1998)
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