Discovery of a functionally selective ghrelin receptor (GHSR 1a ) ligand for modulating brain dopamine
Gross, J D, Kim, D W, Zhou, Y, Jansen, D, Slosky, L M, Clark, N B, Ray, C R, Hu, X, Southall, N, Wang, A, Xu, X, Barnaeva, E, Wetsel, W C, Ferrer, M, Marugan, J J, Caron, M G, Barak, L S, Toth, K
Published in Proceedings of the National Academy of Sciences - PNAS (08.03.2022)
Published in Proceedings of the National Academy of Sciences - PNAS (08.03.2022)
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Efficacy and Mechanism of Action of Low Dose Emetine against Human Cytomegalovirus
Mukhopadhyay, Rupkatha, Roy, Sujayita, Venkatadri, Rajkumar, Su, Yu-Pin, Ye, Wenjuan, Barnaeva, Elena, Mathews Griner, Lesley, Southall, Noel, Hu, Xin, Wang, Amy Q, Xu, Xin, Dulcey, Andrés E, Marugan, Juan J, Ferrer, Marc, Arav-Boger, Ravit
Published in PLoS pathogens (01.06.2016)
Published in PLoS pathogens (01.06.2016)
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Repurposing of the antihistamine chlorcyclizine and related compounds for treatment of hepatitis C virus infection
He, Shanshan, Lin, Billy, Chu, Virginia, Hu, Zongyi, Hu, Xin, Xiao, Jingbo, Wang, Amy Q, Schweitzer, Cameron J, Li, Qisheng, Imamura, Michio, Hiraga, Nobuhiko, Southall, Noel, Ferrer, Marc, Zheng, Wei, Chayama, Kazuaki, Marugan, Juan J, Liang, T Jake
Published in Science translational medicine (08.04.2015)
Published in Science translational medicine (08.04.2015)
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Discovery, Structure–Activity Relationship, and Biological Evaluation of Noninhibitory Small Molecule Chaperones of Glucocerebrosidase
Patnaik, Samarjit, Zheng, Wei, Choi, Jae H, Motabar, Omid, Southall, Noel, Westbroek, Wendy, Lea, Wendy A, Velayati, Arash, Goldin, Ehud, Sidransky, Ellen, Leister, William, Marugan, Juan J
Published in Journal of medicinal chemistry (28.06.2012)
Published in Journal of medicinal chemistry (28.06.2012)
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A widely-applicable high-throughput cellular thermal shift assay (CETSA) using split Nano Luciferase
Martinez, Natalia J., Asawa, Rosita R., Cyr, Matthew G., Zakharov, Alexey, Urban, Daniel J., Roth, Jacob S., Wallgren, Eric, Klumpp-Thomas, Carleen, Coussens, Nathan P., Rai, Ganesha, Yang, Shyh-Ming, Hall, Matthew D., Marugan, Juan J., Simeonov, Anton, Henderson, Mark J.
Published in Scientific reports (21.06.2018)
Published in Scientific reports (21.06.2018)
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Disease models for the development of therapies for lysosomal storage diseases
Xu, Miao, Motabar, Omid, Ferrer, Marc, Marugan, Juan J., Zheng, Wei, Ottinger, Elizabeth A.
Published in Annals of the New York Academy of Sciences (01.05.2016)
Published in Annals of the New York Academy of Sciences (01.05.2016)
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Kinetic modelling of the first step of Mn2O3/MnO thermochemical cycle for solar hydrogen production
Botas, J.A., Marugán, J., Molina, R., Herradón, C.
Published in International journal of hydrogen energy (01.12.2012)
Published in International journal of hydrogen energy (01.12.2012)
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Targeting ATM ameliorates mutant Huntingtin toxicity in cell and animal models of Huntington's disease
Lu, Xiao-Hong, Mattis, Virginia B, Wang, Nan, Al-Ramahi, Ismael, van den Berg, Nick, Fratantoni, Silvina A, Waldvogel, Henry, Greiner, Erin, Osmand, Alex, Elzein, Karla, Xiao, Jingbo, Dijkstra, Sipke, de Pril, Remko, Vinters, Harry V, Faull, Richard, Signer, Ethan, Kwak, Seung, Marugan, Juan J, Botas, Juan, Fischer, David F, Svendsen, Clive N, Munoz-Sanjuan, Ignacio, Yang, X William
Published in Science translational medicine (24.12.2014)
Published in Science translational medicine (24.12.2014)
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ML290 is a biased allosteric agonist at the relaxin receptor RXFP1
Kocan, Martina, Sarwar, Mohsin, Ang, Sheng Y., Xiao, Jingbo, Marugan, Juan J., Hossain, Mohammed A., Wang, Chao, Hutchinson, Dana S., Samuel, Chrishan S., Agoulnik, Alexander I., Bathgate, Ross A. D., Summers, Roger J.
Published in Scientific reports (07.06.2017)
Published in Scientific reports (07.06.2017)
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Neural stem cells for disease modeling and evaluation of therapeutics for infantile (CLN1/PPT1) and late infantile (CLN2/TPP1) neuronal ceroid lipofuscinoses
Sima, Ni, Li, Rong, Huang, Wei, Xu, Miao, Beers, Jeanette, Zou, Jizhong, Titus, Steven, Ottinger, Elizabeth A, Marugan, Juan J, Xie, Xing, Zheng, Wei
Published in Orphanet journal of rare diseases (10.04.2018)
Published in Orphanet journal of rare diseases (10.04.2018)
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In Silico Screening of Inhibitors of the Venezuelan Equine Encephalitis Virus Nonstructural Protein 2 Cysteine Protease
Hu, Xin, Morazzani, Elaine, Compton, Jaimee R, Harmon, Moeshia, Soloveva, Veronica, Glass, Pamela J, Garcia, Andres Dulcey, Marugan, Juan J, Legler, Patricia M
Published in Viruses (01.07.2023)
Published in Viruses (01.07.2023)
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Identification of a G-Protein-Independent Activator of GIRK Channels
Zhao, Yulin, Ung, Peter Man-Un, Zahoránszky-Kőhalmi, Gergely, Zakharov, Alexey V., Martinez, Natalia J., Simeonov, Anton, Glaaser, Ian W., Rai, Ganesha, Schlessinger, Avner, Marugan, Juan J., Slesinger, Paul A.
Published in Cell reports (Cambridge) (16.06.2020)
Published in Cell reports (Cambridge) (16.06.2020)
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Induction and reversal of myotonic dystrophy type 1 pre-mRNA splicing defects by small molecules
Childs-Disney, Jessica L., Stepniak-Konieczna, Ewa, Tran, Tuan, Yildirim, Ilyas, Park, HaJeung, Chen, Catherine Z., Hoskins, Jason, Southall, Noel, Marugan, Juan J., Patnaik, Samarjit, Zheng, Wei, Austin, Chris P., Schatz, George C., Sobczak, Krzysztof, Thornton, Charles A., Disney, Matthew D.
Published in Nature communications (28.06.2013)
Published in Nature communications (28.06.2013)
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Prophylactic treatment with the c-Abl inhibitor, neurotinib, diminishes neuronal damage and the convulsive state in pilocarpine-induced mice
Chandía-Cristi, América, Gutiérrez, Daniela A., Dulcey, Andrés E., Lara, Marcelo, Vargas, Lina, Lin, Yi-Han, Jimenez-Muñoz, Pablo, Larenas, Gabriela, Xu, Xin, Wang, Amy, Owens, Ashley, Dextras, Christopher, Chen, YuChi, Pinto, Claudio, Marín, Tamara, Almarza-Salazar, Hugo, Acevedo, Keryma, Cancino, Gonzalo I., Hu, Xin, Rojas, Patricio, Ferrer, Marc, Southall, Noel, Henderson, Mark J., Zanlungo, Silvana, Marugan, Juan J., Álvarez R, Alejandra
Published in Cell reports (Cambridge) (28.05.2024)
Published in Cell reports (Cambridge) (28.05.2024)
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Niemann-Pick Disease Type C: Induced Pluripotent Stem Cell-Derived Neuronal Cells for Modeling Neural Disease and Evaluating Drug Efficacy
Yu, Daozhan, Swaroop, Manju, Wang, Mengqiao, Baxa, Ulrich, Yang, Rongze, Yan, Yiping, Coksaygan, Turhan, DeTolla, Louis, Marugan, Juan J, Austin, Christopher P, McKew, John C, Gong, Da-Wei, Zheng, Wei
Published in Journal of biomolecular screening (01.09.2014)
Published in Journal of biomolecular screening (01.09.2014)
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Identification and optimization of small-molecule agonists of the human relaxin hormone receptor RXFP1
Xiao, Jingbo, Huang, Zaohua, Chen, Catherine Z., Agoulnik, Irina U., Southall, Noel, Hu, Xin, Jones, Raisa E., Ferrer, Marc, Zheng, Wei, Agoulnik, Alexander I., Marugan, Juan J.
Published in Nature communications (2013)
Published in Nature communications (2013)
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Discovery, Optimization, and Characterization of Novel Chlorcyclizine Derivatives for the Treatment of Hepatitis C Virus Infection
He, Shanshan, Xiao, Jingbo, Dulcey, Andrés E, Lin, Billy, Rolt, Adam, Hu, Zongyi, Hu, Xin, Wang, Amy Q, Xu, Xin, Southall, Noel, Ferrer, Marc, Zheng, Wei, Liang, T. Jake, Marugan, Juan J
Published in Journal of medicinal chemistry (11.02.2016)
Published in Journal of medicinal chemistry (11.02.2016)
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c-Abl tyrosine kinase down-regulation as target for memory improvement in Alzheimer's disease
León, Rilda, Gutiérrez, Daniela A, Pinto, Claudio, Morales, Cristian, de la Fuente, Catalina, Riquelme, Cristóbal, Cortés, Bastián I, González-Martin, Adrián, Chamorro, David, Espinosa, Nelson, Fuentealba, Pablo, Cancino, Gonzalo I, Zanlungo, Silvana, Dulcey, Andrés E, Marugan, Juan J, Álvarez Rojas, Alejandra
Published in Frontiers in aging neuroscience (05.06.2023)
Published in Frontiers in aging neuroscience (05.06.2023)
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Overview of recent advancements in IFMIF-DONES neutronics activities
Qiu, Y., Ansorge, M., Álvarez, I., Ambrožič, K., Berry, T., Bieńkowska, B., Chohan, H., Čufar, A., Dworak, D., Dezsi, T., Eade, T., García, J., Jimenez-Rey, D., Lengar, I., Lopez-Revelles, A.J., Lopez, V., Mendoza, E., Mota, F., Martinez-Echevarria, M.J., Ogando, F., Park, J., Piotrowski, T., Serikov, A., Stankunas, G., Tidikas, A., Tracz, G., Žerovnik, G., Arbeiter, F., Arranz, F., Becerril, S., Cara, P., Bernardi, D., Castellanos, J., Gutiérrez, J., Ibarra, A., Królas, W., Maestre, J., Martín-Fuertes, F., Marugán, J.C., Micciché, G., Martínez-Serrano, J., Nitti, F.S., Podadera, I., Wiącek, U., Fischer, U.
Published in Fusion engineering and design (01.04.2024)
Published in Fusion engineering and design (01.04.2024)
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Anti-apoptotic and Matrix Remodeling Actions of a Small Molecule Agonist of the Human Relaxin Receptor, ML290 in Mice With Unilateral Ureteral Obstruction
Ng, Hooi Hooi, Soula, Mariluz, Rivas, Bryan, Wilson, Kenneth J., Marugan, Juan J., Agoulnik, Alexander I.
Published in Frontiers in physiology (07.07.2021)
Published in Frontiers in physiology (07.07.2021)
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